JP6670756B2 - ブルトン型チロシンキナーゼ(btk)インヒビターとしての多フルオロ置換化合物 - Google Patents

ブルトン型チロシンキナーゼ(btk)インヒビターとしての多フルオロ置換化合物 Download PDF

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JP6670756B2
JP6670756B2 JP2016565402A JP2016565402A JP6670756B2 JP 6670756 B2 JP6670756 B2 JP 6670756B2 JP 2016565402 A JP2016565402 A JP 2016565402A JP 2016565402 A JP2016565402 A JP 2016565402A JP 6670756 B2 JP6670756 B2 JP 6670756B2
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フー,ウェイ
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チョーチアン ディーティーアールエム バイオファーマ コーポレーション リミテッド
チョーチアン ディーティーアールエム バイオファーマ コーポレーション リミテッド
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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JP2016565402A 2014-04-29 2015-04-27 ブルトン型チロシンキナーゼ(btk)インヒビターとしての多フルオロ置換化合物 Active JP6670756B2 (ja)

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CN201410175783.7 2014-04-29
CN201410175783.7A CN105017256A (zh) 2014-04-29 2014-04-29 多氟化合物作为布鲁顿酪氨酸激酶抑制剂
PCT/CN2015/000290 WO2015165279A1 (zh) 2014-04-29 2015-04-27 多氟化合物作为布鲁顿酪氨酸激酶抑制剂

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JP2020040989A (ja) * 2014-04-29 2020-03-19 チョーチアン ディーティーアールエム バイオファーマ コーポレーション リミテッド ブルトン型チロシンキナーゼ(btk)インヒビターとしての多フルオロ置換化合物

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PT3023100T (pt) 2013-07-18 2019-05-29 Taiho Pharmaceutical Co Ltd Fármaco antitumoral para administração intermitente de inibidor de fgfr
ES2819398T3 (es) 2013-07-18 2021-04-15 Taiho Pharmaceutical Co Ltd Agente terapéutico para el cáncer resistente al inhibidor de FGFR
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