AU2015252654C1 - Polyfluorinated compounds acting as Bruton's tyrosine kinase inhibitors - Google Patents

Polyfluorinated compounds acting as Bruton's tyrosine kinase inhibitors Download PDF

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AU2015252654C1
AU2015252654C1 AU2015252654A AU2015252654A AU2015252654C1 AU 2015252654 C1 AU2015252654 C1 AU 2015252654C1 AU 2015252654 A AU2015252654 A AU 2015252654A AU 2015252654 A AU2015252654 A AU 2015252654A AU 2015252654 C1 AU2015252654 C1 AU 2015252654C1
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fluoro
pyrazolo
pyrimidin
phenyl
mmol
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AU2015252654A1 (en
AU2015252654B2 (en
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Wei He
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ZHEJIANG DTRM BIOPHARMA Co Ltd
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ZHEJIANG DTRM BIOPHARMA CO Ltd
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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AU2015252654A 2014-04-29 2015-04-27 Polyfluorinated compounds acting as Bruton's tyrosine kinase inhibitors Active AU2015252654C1 (en)

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Application Number Priority Date Filing Date Title
CN201410175783.7 2014-04-29
CN201410175783.7A CN105017256A (zh) 2014-04-29 2014-04-29 多氟化合物作为布鲁顿酪氨酸激酶抑制剂
PCT/CN2015/000290 WO2015165279A1 (zh) 2014-04-29 2015-04-27 多氟化合物作为布鲁顿酪氨酸激酶抑制剂

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AU2015252654A1 AU2015252654A1 (en) 2016-11-03
AU2015252654B2 AU2015252654B2 (en) 2019-10-03
AU2015252654C1 true AU2015252654C1 (en) 2020-01-23

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KR (2) KR20160144378A (enExample)
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WO2015008844A1 (ja) 2013-07-18 2015-01-22 大鵬薬品工業株式会社 Ｆｇｆｒ阻害剤耐性癌の治療薬
TR201907147T4 (tr) 2013-07-18 2019-06-21 Taiho Pharmaceutical Co Ltd Fgfr inhibitörünün aralıklı uygulanmasına yönelik anti-tümör ilaç.
CN105017256A (zh) * 2014-04-29 2015-11-04 浙江导明医药科技有限公司 多氟化合物作为布鲁顿酪氨酸激酶抑制剂
WO2016079693A1 (en) * 2014-11-19 2016-05-26 Sun Pharmaceutical Industries Limited A process for the preparation of ibrutinib
JP6681922B2 (ja) * 2015-02-12 2020-04-15 上▲海▼度▲徳▼医▲藥▼科技有限公司 イブルチニブの製造方法
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