JP5693951B2 - プロテインキナーゼの阻害剤 - Google Patents

プロテインキナーゼの阻害剤 Download PDF

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JP5693951B2
JP5693951B2 JP2010504681A JP2010504681A JP5693951B2 JP 5693951 B2 JP5693951 B2 JP 5693951B2 JP 2010504681 A JP2010504681 A JP 2010504681A JP 2010504681 A JP2010504681 A JP 2010504681A JP 5693951 B2 JP5693951 B2 JP 5693951B2
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alkyl
phenyl
compound
pain
methoxy
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JP2010504681A
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Japanese (ja)
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JP2011502956A (ja
JP2011502956A5 (enExample
Inventor
ワブニトズ プヒリププ
ワブニトズ プヒリププ
スチャウエルテ ヘイケ
スチャウエルテ ヘイケ
アルルゲイエル ハンス
アルルゲイエル ハンス
アウグストイン マルトイン
アウグストイン マルトイン
ゼイトルマンン ルトズ
ゼイトルマンン ルトズ
エー．プレイスス ミチャエル
エー．プレイスス ミチャエル
ストウムム ガブリエレ
ストウムム ガブリエレ
ムエルレル アンケ
ムエルレル アンケ
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アストラゼネカ エービー
アストラゼネカ エービー
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
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JP2010504681A 2007-04-24 2008-04-24 プロテインキナーゼの阻害剤 Expired - Fee Related JP5693951B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EPPCT/EP2007/003602 2007-04-24
EP2007003602 2007-04-24
PCT/EP2008/054975 WO2008129070A1 (en) 2007-04-24 2008-04-24 Inhibitors of protein kinases

Publications (3)

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JP2011502956A JP2011502956A (ja) 2011-01-27
JP2011502956A5 JP2011502956A5 (enExample) 2011-06-16
JP5693951B2 true JP5693951B2 (ja) 2015-04-01

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JP2010504681A Expired - Fee Related JP5693951B2 (ja) 2007-04-24 2008-04-24 プロテインキナーゼの阻害剤

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US (1) US8436007B2 (enExample)
JP (1) JP5693951B2 (enExample)
ES (1) ES2539518T3 (enExample)
WO (1) WO2008129070A1 (enExample)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
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EP2137166B1 (en) * 2007-04-24 2012-05-30 Ingenium Pharmaceuticals GmbH 4, 6-disubstituted aminopyrimidine derivatives as inhibitors of protein kinases
ES2539518T3 (es) 2007-04-24 2015-07-01 Astrazeneca Ab Inhibidores de proteínas quinasas
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