JP5412273B2 - ペプチド−ぺプチダーゼ阻害剤及びその使用 - Google Patents

ペプチド−ぺプチダーゼ阻害剤及びその使用 Download PDF

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Publication number
JP5412273B2
JP5412273B2 JP2009501566A JP2009501566A JP5412273B2 JP 5412273 B2 JP5412273 B2 JP 5412273B2 JP 2009501566 A JP2009501566 A JP 2009501566A JP 2009501566 A JP2009501566 A JP 2009501566A JP 5412273 B2 JP5412273 B2 JP 5412273B2
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peptide
seq
conjugate
glp
peptidase
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Expired - Fee Related
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JP2009501566A
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Japanese (ja)
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JP2009530395A5 (https=
JP2009530395A (ja
Inventor
サウミトラ・ゴーシュ
ジョズエ・アルファロ−ロペス
ローレンス・ドスーザ
オディール・レビー
リン・チン
クリス・ソアレス
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Amylin Pharmaceuticals LLC
AstraZeneca Pharmaceuticals LP
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Amylin Pharmaceuticals LLC
AstraZeneca Pharmaceuticals LP
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/545—Heterocyclic compounds
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  • Diabetes (AREA)
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  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Endocrinology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Physical Education & Sports Medicine (AREA)
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  • Molecular Biology (AREA)
  • Child & Adolescent Psychology (AREA)
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  • Psychiatry (AREA)
  • Vascular Medicine (AREA)
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  • Nutrition Science (AREA)
  • Reproductive Health (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2009501566A 2006-03-21 2007-03-21 ペプチド−ぺプチダーゼ阻害剤及びその使用 Expired - Fee Related JP5412273B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US78479506P 2006-03-21 2006-03-21
US60/784,795 2006-03-21
PCT/US2007/007163 WO2007109354A2 (en) 2006-03-21 2007-03-21 Peptide-peptidase inhibitor conjugates and methods of using same

Publications (3)

Publication Number Publication Date
JP2009530395A JP2009530395A (ja) 2009-08-27
JP2009530395A5 JP2009530395A5 (https=) 2010-05-06
JP5412273B2 true JP5412273B2 (ja) 2014-02-12

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JP2009501566A Expired - Fee Related JP5412273B2 (ja) 2006-03-21 2007-03-21 ペプチド−ぺプチダーゼ阻害剤及びその使用

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US (3) US20090186817A1 (https=)
EP (1) EP2004238A2 (https=)
JP (1) JP5412273B2 (https=)
CN (1) CN101432025B (https=)
AU (1) AU2007227202B2 (https=)
CA (1) CA2646598C (https=)
WO (1) WO2007109354A2 (https=)

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