JP5148499B2 - Ｖｅｇｆ受容体およびｈｇｆ受容体シグナル伝達の阻害剤 - Google Patents

Ｖｅｇｆ受容体およびｈｇｆ受容体シグナル伝達の阻害剤 Download PDF

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JP5148499B2
JP5148499B2 JP2008537239A JP2008537239A JP5148499B2 JP 5148499 B2 JP5148499 B2 JP 5148499B2 JP 2008537239 A JP2008537239 A JP 2008537239A JP 2008537239 A JP2008537239 A JP 2008537239A JP 5148499 B2 JP5148499 B2 JP 5148499B2
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thieno
pyridin
yloxy
phenyl
imidazol
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Japanese (ja)
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JP2009504804A5 (https=
JP2009504804A (ja
Inventor
サーヴェドゥラ，オスカー，マリオ
クラリッジ，ステフェン，ウィリアム
ツァン，リジー
ラエッペル，フランク
ヴァイスブルク，アルカディー
ラエッペル，ステファン
ドゥジエル，ロベール
マンニオン，ミヒャエル
ツー，ナンシー
ゴデット，フレデリック
イサコヴィック，リュボミール
ワーブ，アマル
グランジャー，マリー−クロード
ベルンスタイン，ナオミー
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メチルジーン インコーポレイテッド
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
JP2008537239A 2005-05-20 2006-05-19 Ｖｅｇｆ受容体およびｈｇｆ受容体シグナル伝達の阻害剤 Active JP5148499B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US68303605P 2005-05-20 2005-05-20
US60/683,036 2005-05-20
US75490205P 2005-12-29 2005-12-29
US60/754,902 2005-12-29
US78505406P 2006-03-22 2006-03-22
US60/785,054 2006-03-22
PCT/IB2006/004306 WO2008041053A2 (en) 2005-05-20 2006-05-19 Inhibitors of vegf receptor and hgf receptor signaling

Publications (3)

Publication Number Publication Date
JP2009504804A JP2009504804A (ja) 2009-02-05
JP2009504804A5 JP2009504804A5 (https=) 2009-07-09
JP5148499B2 true JP5148499B2 (ja) 2013-02-20

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JP2008537239A Active JP5148499B2 (ja) 2005-05-20 2006-05-19 Ｖｅｇｆ受容体およびｈｇｆ受容体シグナル伝達の阻害剤

Country Status (13)

Country Link
US (2) US8093264B2 (https=)
EP (1) EP1957498B1 (https=)
JP (1) JP5148499B2 (https=)
KR (1) KR101378716B1 (https=)
CN (1) CN101796055B (https=)
AU (1) AU2006343808B2 (https=)
BR (1) BRPI0610322B8 (https=)
CA (1) CA2611370C (https=)
ES (1) ES2623221T3 (https=)
IL (1) IL187484A (https=)
MX (1) MX2007014616A (https=)
NZ (1) NZ564283A (https=)
WO (1) WO2008041053A2 (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010536887A (ja) * 2007-08-29 2010-12-02 メチルジーン インコーポレイテッド タンパク質チロシンキナーゼ活性の阻害剤

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JP2010536887A (ja) * 2007-08-29 2010-12-02 メチルジーン インコーポレイテッド タンパク質チロシンキナーゼ活性の阻害剤

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IL187484A (en) 2014-04-30
BRPI0610322B1 (pt) 2020-12-01
CN101796055A (zh) 2010-08-04
CN101796055B (zh) 2013-09-04
KR20080059112A (ko) 2008-06-26
EP1957498A4 (en) 2010-10-27
AU2006343808A1 (en) 2008-04-10
US8329726B2 (en) 2012-12-11
IL187484A0 (en) 2011-08-01
WO2008041053A2 (en) 2008-04-10
MX2007014616A (es) 2009-08-12
US20120083482A1 (en) 2012-04-05
KR101378716B1 (ko) 2014-04-10
JP2009504804A (ja) 2009-02-05
BRPI0610322A2 (pt) 2010-06-15
EP1957498B1 (en) 2017-02-15
US20070004675A1 (en) 2007-01-04
NZ564283A (en) 2011-07-29
CA2611370C (en) 2014-11-25
EP1957498A2 (en) 2008-08-20
WO2008041053A3 (en) 2009-12-23
AU2006343808B2 (en) 2012-03-29
US8093264B2 (en) 2012-01-10
CA2611370A1 (en) 2006-11-20
BRPI0610322B8 (pt) 2021-05-25
ES2623221T3 (es) 2017-07-10

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