JP4787234B2 - アルキルピペラジン−及びアルキルホモピペラジン−カルボキシラートの誘導体、その調製方法及びｆａａｈ酵素阻害剤としての同使用 - Google Patents

アルキルピペラジン−及びアルキルホモピペラジン−カルボキシラートの誘導体、その調製方法及びｆａａｈ酵素阻害剤としての同使用 Download PDF

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JP4787234B2
JP4787234B2 JP2007500259A JP2007500259A JP4787234B2 JP 4787234 B2 JP4787234 B2 JP 4787234B2 JP 2007500259 A JP2007500259 A JP 2007500259A JP 2007500259 A JP2007500259 A JP 2007500259A JP 4787234 B2 JP4787234 B2 JP 4787234B2
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JP2007524704A5 (enExample
JP2007524704A (ja
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アブアブデラ，アメツド
アルマリオ・ガルシア，アントニオ
オールナエール，クリスチヤン
リ，アドリアン・タク
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Sanofi SA
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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
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  • Animal Behavior & Ethology (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Communicable Diseases (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Epidemiology (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
JP2007500259A 2004-02-26 2005-02-25 アルキルピペラジン−及びアルキルホモピペラジン−カルボキシラートの誘導体、その調製方法及びｆａａｈ酵素阻害剤としての同使用 Expired - Fee Related JP4787234B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR0401953A FR2866888B1 (fr) 2004-02-26 2004-02-26 Derives de alkylpiperazine- et alkylhomopiperazine- carboxylates, leur preparation et leur application en therapeutique
FR0401953 2004-02-26
PCT/FR2005/000450 WO2005090322A1 (fr) 2004-02-26 2005-02-25 Derives de alkylpiperazine- et alkylhomopiperazine- carboxylates, leur preparation et leur application en tant qu’inhibiteurs de l’enzyme faah

Publications (3)

Publication Number Publication Date
JP2007524704A JP2007524704A (ja) 2007-08-30
JP2007524704A5 JP2007524704A5 (enExample) 2008-04-03
JP4787234B2 true JP4787234B2 (ja) 2011-10-05

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JP2007500259A Expired - Fee Related JP4787234B2 (ja) 2004-02-26 2005-02-25 アルキルピペラジン−及びアルキルホモピペラジン−カルボキシラートの誘導体、その調製方法及びｆａａｈ酵素阻害剤としての同使用

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US (2) US7482346B2 (enExample)
EP (1) EP1720848B1 (enExample)
JP (1) JP4787234B2 (enExample)
KR (1) KR20060133592A (enExample)
CN (1) CN100567279C (enExample)
AR (1) AR047974A1 (enExample)
AT (1) ATE380184T1 (enExample)
AU (1) AU2005223422B2 (enExample)
BR (1) BRPI0508047A (enExample)
CA (1) CA2554855A1 (enExample)
CY (1) CY1107182T1 (enExample)
DE (1) DE602005003648T2 (enExample)
DK (1) DK1720848T3 (enExample)
ES (1) ES2296162T3 (enExample)
FR (1) FR2866888B1 (enExample)
HR (1) HRP20080024T3 (enExample)
IL (1) IL177422A (enExample)
MA (1) MA28370A1 (enExample)
NO (1) NO20064364L (enExample)
NZ (1) NZ549471A (enExample)
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PT (1) PT1720848E (enExample)
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RU (1) RU2331637C2 (enExample)
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US9968396B2 (en) 2008-05-27 2018-05-15 Maquet Cardiovascular Llc Surgical instrument and method
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CN101712655B (zh) * 2008-10-08 2012-05-23 秦引林 一种乙酰胺类衍生物及其在制药中的应用
CN101503394B (zh) * 2009-03-11 2010-05-12 深圳市湘雅生物医药研究院 高哌嗪乙酰肼类衍生物及其制备方法和用途
FR2945533B1 (fr) 2009-05-12 2011-05-27 Sanofi Aventis Derives de cyclopenta°c!pyrrolyl-alkylcarbamates d'heterocycles a 5 chainons, leur preparation et leur application en therapeutique
FR2945531A1 (fr) * 2009-05-12 2010-11-19 Sanofi Aventis Derives de 7-aza-spiro°3,5!nonane-7-carboxylates, leur preparation et leur application en therapeutique
AR076687A1 (es) * 2009-05-18 2011-06-29 Infinity Pharmaceuticals Inc Isoxazolinas como inhibidores de la amidahidrolasa de acidos grasos y com-posiciones farmaceuticas que los contienen
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WO2011123719A2 (en) 2010-03-31 2011-10-06 Ironwood Pharmaceuticals, Inc. Use of faah inhibitors for treating abdominal, visceral and pelvic pain
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