JP2007524704A5 - - Google Patents

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Publication number
JP2007524704A5
JP2007524704A5 JP2007500259A JP2007500259A JP2007524704A5 JP 2007524704 A5 JP2007524704 A5 JP 2007524704A5 JP 2007500259 A JP2007500259 A JP 2007500259A JP 2007500259 A JP2007500259 A JP 2007500259A JP 2007524704 A5 JP2007524704 A5 JP 2007524704A5
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JP
Japan
Prior art keywords
group
formula
alkyl
groups
cycloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2007500259A
Other languages
English (en)
Japanese (ja)
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JP2007524704A (ja
JP4787234B2 (ja
Filing date
Publication date
Priority claimed from FR0401953A external-priority patent/FR2866888B1/fr
Application filed filed Critical
Publication of JP2007524704A publication Critical patent/JP2007524704A/ja
Publication of JP2007524704A5 publication Critical patent/JP2007524704A5/ja
Application granted granted Critical
Publication of JP4787234B2 publication Critical patent/JP4787234B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2007500259A 2004-02-26 2005-02-25 アルキルピペラジン−及びアルキルホモピペラジン−カルボキシラートの誘導体、その調製方法及びfaah酵素阻害剤としての同使用 Expired - Fee Related JP4787234B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR0401953 2004-02-26
FR0401953A FR2866888B1 (fr) 2004-02-26 2004-02-26 Derives de alkylpiperazine- et alkylhomopiperazine- carboxylates, leur preparation et leur application en therapeutique
PCT/FR2005/000450 WO2005090322A1 (fr) 2004-02-26 2005-02-25 Derives de alkylpiperazine- et alkylhomopiperazine- carboxylates, leur preparation et leur application en tant qu’inhibiteurs de l’enzyme faah

Publications (3)

Publication Number Publication Date
JP2007524704A JP2007524704A (ja) 2007-08-30
JP2007524704A5 true JP2007524704A5 (enExample) 2008-04-03
JP4787234B2 JP4787234B2 (ja) 2011-10-05

Family

ID=34834070

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007500259A Expired - Fee Related JP4787234B2 (ja) 2004-02-26 2005-02-25 アルキルピペラジン−及びアルキルホモピペラジン−カルボキシラートの誘導体、その調製方法及びfaah酵素阻害剤としての同使用

Country Status (28)

Country Link
US (2) US7482346B2 (enExample)
EP (1) EP1720848B1 (enExample)
JP (1) JP4787234B2 (enExample)
KR (1) KR20060133592A (enExample)
CN (1) CN100567279C (enExample)
AR (1) AR047974A1 (enExample)
AT (1) ATE380184T1 (enExample)
AU (1) AU2005223422B2 (enExample)
BR (1) BRPI0508047A (enExample)
CA (1) CA2554855A1 (enExample)
CY (1) CY1107182T1 (enExample)
DE (1) DE602005003648T2 (enExample)
DK (1) DK1720848T3 (enExample)
ES (1) ES2296162T3 (enExample)
FR (1) FR2866888B1 (enExample)
HR (1) HRP20080024T3 (enExample)
IL (1) IL177422A (enExample)
MA (1) MA28370A1 (enExample)
NO (1) NO20064364L (enExample)
NZ (1) NZ549471A (enExample)
PL (1) PL1720848T3 (enExample)
PT (1) PT1720848E (enExample)
RS (1) RS50542B (enExample)
RU (1) RU2331637C2 (enExample)
SI (1) SI1720848T1 (enExample)
TW (1) TWI350286B (enExample)
WO (1) WO2005090322A1 (enExample)
ZA (1) ZA200607092B (enExample)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0102299D0 (sv) 2001-06-26 2001-06-26 Astrazeneca Ab Compounds
FR2866884B1 (fr) * 2004-02-26 2007-08-31 Sanofi Synthelabo Derives d'aryl-et d'heteroaryl-piperidinecarboxylates, leur preparation et leur application en therapeutique
US7269708B2 (en) * 2004-04-20 2007-09-11 Rambus Inc. Memory controller for non-homogenous memory system
TWI385152B (zh) 2005-02-17 2013-02-11 Astellas Pharma Inc Pyridyl non-aromatic nitrogen-containing heterocyclic-1-carboxylate derivatives (I)
US8197472B2 (en) 2005-03-25 2012-06-12 Maquet Cardiovascular, Llc Tissue welding and cutting apparatus and method
US7918848B2 (en) 2005-03-25 2011-04-05 Maquet Cardiovascular, Llc Tissue welding and cutting apparatus and method
WO2007005510A1 (en) 2005-06-30 2007-01-11 Janssen Pharmaceutica N.V. N-heteroarylpiperazinyl ureas as modulators of fatty acid amide hydrolase
EP2065369A4 (en) * 2006-08-23 2011-12-28 Astellas Pharma Inc UREA CONNECTION OR SALT THEREOF
US9402680B2 (en) 2008-05-27 2016-08-02 Maquet Cardiovasular, Llc Surgical instrument and method
JP2011521723A (ja) 2008-05-27 2011-07-28 マッケ カーディオバスキュラー,エルエルシー 外科用器具および方法
US9968396B2 (en) 2008-05-27 2018-05-15 Maquet Cardiovascular Llc Surgical instrument and method
CN101712655B (zh) * 2008-10-08 2012-05-23 秦引林 一种乙酰胺类衍生物及其在制药中的应用
CN101503394B (zh) * 2009-03-11 2010-05-12 深圳市湘雅生物医药研究院 高哌嗪乙酰肼类衍生物及其制备方法和用途
FR2945533B1 (fr) * 2009-05-12 2011-05-27 Sanofi Aventis Derives de cyclopenta°c!pyrrolyl-alkylcarbamates d'heterocycles a 5 chainons, leur preparation et leur application en therapeutique
FR2945531A1 (fr) * 2009-05-12 2010-11-19 Sanofi Aventis Derives de 7-aza-spiro°3,5!nonane-7-carboxylates, leur preparation et leur application en therapeutique
AR076687A1 (es) * 2009-05-18 2011-06-29 Infinity Pharmaceuticals Inc Isoxazolinas como inhibidores de la amidahidrolasa de acidos grasos y com-posiciones farmaceuticas que los contienen
TW201044234A (en) * 2009-06-08 2010-12-16 Chunghwa Picture Tubes Ltd Method of scanning touch panel
US9955858B2 (en) * 2009-08-21 2018-05-01 Maquet Cardiovascular Llc Surgical instrument and method for use
US20130150346A1 (en) 2010-01-08 2013-06-13 Quest Ventures Ltd. Use of FAAH Inhibitors for Treating Parkinson's Disease and Restless Legs Syndrome
WO2011123719A2 (en) 2010-03-31 2011-10-06 Ironwood Pharmaceuticals, Inc. Use of faah inhibitors for treating abdominal, visceral and pelvic pain
WO2012015704A2 (en) 2010-07-28 2012-02-02 The Regents Of The University Of California Peripherally restricted faah inhibitors
ES2708723T3 (es) 2011-08-19 2019-04-10 Univ California Inhibidores de FAAH restringidos de forma periférica sustituidos en posición meta por bifenilo
ES2908240T3 (es) 2014-04-07 2022-04-28 Univ California Inhibidores de la enzima amida hidrolasa de ácidos grasos (FAAH) con biodisponibilidad oral mejorada y su uso como medicamentos
CN104356082B (zh) * 2014-10-31 2016-07-13 厦门大学 一类取代杂环衍生物及其制备方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2142883A1 (en) * 1992-08-21 1994-03-03 Saizo Shibata Dioxacycloalkane compound having renin-inhibitory activity
FR2740134B1 (fr) * 1995-10-18 1998-01-09 Pf Medicament Derives d'amines cycliques d'aryl-piperazines, leur preparation et les compositions pharmaceutiques les contenant
DE19816889A1 (de) * 1998-04-16 1999-10-21 Boehringer Ingelheim Pharma Piperazinderivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung
EP1268455A2 (en) * 2000-03-31 2003-01-02 Pfizer Products Inc. Piperazine derivatives
AU2003237882B2 (en) * 2002-05-16 2010-04-08 Sunovion Pharmaceuticals Inc. Amines that inhibit a mammalian anandamide transporter, and methods of use thereof
JP4228587B2 (ja) * 2002-05-22 2009-02-25 昭和電工株式会社 アミノメチル基含有ベンズアミド化合物の製造方法
FR2843964B1 (fr) * 2002-08-29 2004-10-01 Sanofi Synthelabo Derives de dioxane-2-alkylcarbamates, leur preparation et leur application en therapeutique
FR2854633B1 (fr) * 2003-05-07 2005-06-24 Sanofi Synthelabo Derives de piperidinyl-et piperazinyl-alkylcarbamates, leur preparation et leur application en therapeutique
FR2864080B1 (fr) * 2003-12-23 2006-02-03 Sanofi Synthelabo Derives de 1-piperazine-et-1-homopiperazine-carboxylates, leur preparation et leur application en therapeutique
FR2865205B1 (fr) * 2004-01-16 2006-02-24 Sanofi Synthelabo Derives de type aryloxyalkylcarbamates, leur preparation et leur application en therapeutique
FR2866884B1 (fr) * 2004-02-26 2007-08-31 Sanofi Synthelabo Derives d'aryl-et d'heteroaryl-piperidinecarboxylates, leur preparation et leur application en therapeutique
FR2866885B1 (fr) * 2004-02-26 2007-08-31 Sanofi Synthelabo Derives de piperidinylalkylcarbamates, leur prepation et leur application en therapeutique

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