JP4723242B2 - 炎症および免疫障害治療用ｃｃｒ１アンタゴニストとして使用するための１−アリール−４−置換ピペラジン誘導体 - Google Patents

炎症および免疫障害治療用ｃｃｒ１アンタゴニストとして使用するための１−アリール−４−置換ピペラジン誘導体 Download PDF

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JP4723242B2
JP4723242B2 JP2004512756A JP2004512756A JP4723242B2 JP 4723242 B2 JP4723242 B2 JP 4723242B2 JP 2004512756 A JP2004512756 A JP 2004512756A JP 2004512756 A JP2004512756 A JP 2004512756A JP 4723242 B2 JP4723242 B2 JP 4723242B2
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cycloalkyl
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JP2006508036A5 (enExample
JP2006508036A (ja
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アンドリュー エム． ケイ． ペンネル
ジェイムス ビー． アッゲン
ジェイ． ジェイ． キム ライト
スブハブラタ セン
ブライアン イー． マックマスター
ダニエル ジョセフ ダイラギ
バレリー ブイ． マルティチョノク
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JP2004512756A 2002-06-12 2003-06-11 炎症および免疫障害治療用ｃｃｒ１アンタゴニストとして使用するための１−アリール−４−置換ピペラジン誘導体 Expired - Lifetime JP4723242B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US45371102P 2002-06-12 2002-06-12
US60/453,711 2002-06-12
PCT/US2003/018660 WO2003105853A1 (en) 2002-06-12 2003-06-11 1-aryl-4-substituted piperazines derivatives for use as ccr1 antagonists for the treatment of inflammation and immune disorders

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JP2006508036A JP2006508036A (ja) 2006-03-09
JP2006508036A5 JP2006508036A5 (enExample) 2006-08-03
JP4723242B2 true JP4723242B2 (ja) 2011-07-13

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US (2) US7157464B2 (enExample)
EP (1) EP1531822B1 (enExample)
JP (1) JP4723242B2 (enExample)
KR (1) KR101255356B1 (enExample)
CN (1) CN1867336B (enExample)
AT (1) ATE438401T1 (enExample)
AU (1) AU2003236500B9 (enExample)
CA (1) CA2488202C (enExample)
DE (1) DE60328690D1 (enExample)
DK (1) DK1531822T3 (enExample)
ES (1) ES2329356T3 (enExample)
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JP4958787B2 (ja) 2004-09-20 2012-06-20 ゼノン・ファーマシューティカルズ・インコーポレイテッド ヒトステアロイル−ＣｏＡデサチュラーゼを阻害するためのピリジン誘導体
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