JP4612990B2 - ヒスタミン−３受容体リガンドとしての新規アミンおよびそれらの治療的適用 - Google Patents

ヒスタミン−３受容体リガンドとしての新規アミンおよびそれらの治療的適用 Download PDF

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JP4612990B2
JP4612990B2 JP2002573767A JP2002573767A JP4612990B2 JP 4612990 B2 JP4612990 B2 JP 4612990B2 JP 2002573767 A JP2002573767 A JP 2002573767A JP 2002573767 A JP2002573767 A JP 2002573767A JP 4612990 B2 JP4612990 B2 JP 4612990B2
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ethyl
benzofuran
methyl
pyrrolidinyl
pyrrolidin
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JP2005500986A (ja
JP2005500986A5 (https=
Inventor
コワート，マーロン・デイー
ベンナニ，ユセフ・エル
フアギー，ラミン
グフエサー，グレゴリー・エイ
ブラツク，ローレンス・エイ
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Abbott Laboratories
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Abbott Laboratories
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Priority claimed from US09/810,648 external-priority patent/US20020177589A1/en
Priority claimed from US10/044,495 external-priority patent/US20020183309A1/en
Priority claimed from US10/081,207 external-priority patent/US6969730B2/en
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Publication of JP2005500986A publication Critical patent/JP2005500986A/ja
Publication of JP2005500986A5 publication Critical patent/JP2005500986A5/ja
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JP2002573767A 2001-03-16 2002-03-11 ヒスタミン−３受容体リガンドとしての新規アミンおよびそれらの治療的適用 Expired - Fee Related JP4612990B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US09/810,648 US20020177589A1 (en) 2001-03-16 2001-03-16 Novel amines as histamine-3 receptor ligands and their therapeutic applications
US10/044,495 US20020183309A1 (en) 2001-03-16 2002-01-11 Novel amines as histamine-3 receptor ligands and their therapeutic applications
US10/081,207 US6969730B2 (en) 2001-03-16 2002-02-25 Amines as histamine-3 receptor ligands and their therapeutic applications
PCT/US2002/007107 WO2002074758A2 (en) 2001-03-16 2002-03-11 Novel amines as histamine-3 receptor ligands and their therapeutic applications

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JP2005500986A JP2005500986A (ja) 2005-01-13
JP2005500986A5 JP2005500986A5 (https=) 2005-12-22
JP4612990B2 true JP4612990B2 (ja) 2011-01-12

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EP (2) EP2258694A1 (https=)
JP (1) JP4612990B2 (https=)
AR (1) AR035783A1 (https=)
BR (1) BR0205829A (https=)
CA (1) CA2440238C (https=)
MX (1) MXPA03008319A (https=)
WO (1) WO2002074758A2 (https=)

Families Citing this family (40)

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US7314937B2 (en) 2002-03-21 2008-01-01 Eli Lilly And Company Non-imidazole aryl alkylamines compounds as histamine H3 receptor antagonists, preparation and therapeutic uses
US6822101B2 (en) 2002-09-16 2004-11-23 Abbott Laboratories Process for preparing amine-substituted benzofurans
US7153889B2 (en) 2002-11-12 2006-12-26 Abbott Laboratories Bicyclic-substituted amines as histamine-3 receptor ligands
JP4820094B2 (ja) * 2002-11-12 2011-11-24 アボット・ラボラトリーズ ヒスタミン−３受容体リガンドとしての２環式置換アミン
US7244852B2 (en) 2003-02-27 2007-07-17 Abbott Laboratories Process for preparing 2-methylpyrrolidine and specific enantiomers thereof
WO2004080966A1 (ja) 2003-03-14 2004-09-23 Ono Pharmaceutical Co., Ltd. 含窒素複素環誘導体およびそれらを有効成分とする薬剤
WO2004089410A1 (ja) * 2003-04-03 2004-10-21 Kyowa Hakko Kogyo Co., Ltd. 神経因性疼痛の予防及び／または治療剤
US20040224952A1 (en) * 2003-05-07 2004-11-11 Cowart Marlon D. Fused bicyclic-substituted amines as histamine-3 receptor ligands
WO2004101559A1 (en) * 2003-05-07 2004-11-25 Abbott Laboratories Fused bicyclic-substituted amines as histamine-3 receptor ligands
US7094790B2 (en) 2003-05-07 2006-08-22 Abbott Laboratories Fused bicyclic-substituted amines as histamine-3 receptor ligands
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