AU2003291329A1 - Bicyclic-substituted amines as histamine-3 receptor ligands - Google Patents
Bicyclic-substituted amines as histamine-3 receptor ligandsInfo
- Publication number
- AU2003291329A1 AU2003291329A1 AU2003291329A AU2003291329A AU2003291329A1 AU 2003291329 A1 AU2003291329 A1 AU 2003291329A1 AU 2003291329 A AU2003291329 A AU 2003291329A AU 2003291329 A AU2003291329 A AU 2003291329A AU 2003291329 A1 AU2003291329 A1 AU 2003291329A1
- Authority
- AU
- Australia
- Prior art keywords
- histamine
- bicyclic
- receptor ligands
- substituted amines
- amines
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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- C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C255/58—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
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GB1166538A (en) * | 1967-06-10 | 1969-10-08 | Pfizer Ltd | Substituted Tetrahydroquinolines |
US3489756A (en) * | 1967-07-10 | 1970-01-13 | Merck & Co Inc | 2-carbocyclic-6-tertiary amino alkoxy naphthalenes and tetralins |
JPS5649357A (en) * | 1979-09-28 | 1981-05-02 | Otsuka Pharmaceut Co Ltd | Quinoline derivative |
JP2551298B2 (en) * | 1991-04-25 | 1996-11-06 | 田辺製薬株式会社 | Antidepressant |
US5480883A (en) * | 1991-05-10 | 1996-01-02 | Rhone-Poulenc Rorer Pharmaceuticals Inc. | Bis mono- and bicyclic aryl and heteroaryl compounds which inhibit EGF and/or PDGF receptor tyrosine kinase |
EP1019375A1 (en) * | 1997-03-25 | 2000-07-19 | Astra Pharmaceuticals Limited | Novel pyridine derivatives and pharmaceutical compositions containing them |
IL131846A0 (en) * | 1997-03-25 | 2001-03-19 | Astra Pharma Prod | Novel pyridine derivatives and pharmaceutical compositions containing them |
JP4370002B2 (en) * | 1997-08-08 | 2009-11-25 | 富山化学工業株式会社 | Quinolone carboxylic acid derivative or salt thereof |
EP0982300A3 (en) * | 1998-07-29 | 2000-03-08 | Societe Civile Bioprojet | Non-imidazole alkylamines as histamine H3 - receptor ligands and their therapeutic applications |
AU4058399A (en) * | 1998-11-20 | 2000-06-13 | Torii Pharmaceutical Co., Ltd. | Naphthalene derivatives |
JP2002275157A (en) * | 1998-11-20 | 2002-09-25 | Torii Yakuhin Kk | New naphthalene derivative |
WO2002018335A1 (en) * | 2000-08-28 | 2002-03-07 | Yamanouchi Pharmaceutical Co., Ltd. | Cyclic amine derivatives |
DE60134762D1 (en) * | 2000-10-02 | 2008-08-21 | Janssen Pharmaceutica Nv | METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS |
CA2440238C (en) * | 2001-03-16 | 2011-09-13 | Abbott Laboratories | Novel amines as histamine-3 receptor ligands and their therapeutic applications |
-
2003
- 2003-11-05 WO PCT/US2003/035365 patent/WO2004043458A1/en active Application Filing
- 2003-11-05 AU AU2003291329A patent/AU2003291329A1/en not_active Abandoned
- 2003-11-05 JP JP2004551799A patent/JP4820094B2/en not_active Expired - Fee Related
- 2003-11-05 EP EP03768721A patent/EP1569637A1/en not_active Withdrawn
- 2003-11-05 CA CA2505427A patent/CA2505427C/en not_active Expired - Fee Related
- 2003-11-05 CA CA2765093A patent/CA2765093A1/en not_active Abandoned
- 2003-11-05 PL PL376751A patent/PL376751A1/en not_active Application Discontinuation
- 2003-11-05 MX MXPA05005116A patent/MXPA05005116A/en active IP Right Grant
- 2003-11-12 TW TW092131661A patent/TWI359658B/en not_active IP Right Cessation
-
2010
- 2010-10-20 JP JP2010235798A patent/JP2011063594A/en active Pending
Also Published As
Publication number | Publication date |
---|---|
TW200418454A (en) | 2004-10-01 |
CA2505427A1 (en) | 2004-05-27 |
MXPA05005116A (en) | 2005-07-01 |
PL376751A1 (en) | 2006-01-09 |
JP4820094B2 (en) | 2011-11-24 |
CA2505427C (en) | 2012-04-03 |
EP1569637A1 (en) | 2005-09-07 |
JP2006514926A (en) | 2006-05-18 |
CA2765093A1 (en) | 2004-05-27 |
JP2011063594A (en) | 2011-03-31 |
WO2004043458A1 (en) | 2004-05-27 |
TWI359658B (en) | 2012-03-11 |
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MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |