JP4553487B2 - ヒスタミンｈ３−受容体リガンドとしての非イミダゾールアルキルアミンと、その治療への応用。 - Google Patents

ヒスタミンｈ３−受容体リガンドとしての非イミダゾールアルキルアミンと、その治療への応用。 Download PDF

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JP4553487B2
JP4553487B2 JP2000562103A JP2000562103A JP4553487B2 JP 4553487 B2 JP4553487 B2 JP 4553487B2 JP 2000562103 A JP2000562103 A JP 2000562103A JP 2000562103 A JP2000562103 A JP 2000562103A JP 4553487 B2 JP4553487 B2 JP 4553487B2
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propyl
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piperidine
pyrrolidine
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JP2002521463A (ja
JP2002521463A5 (https=
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ジャン−シャール シュワルツ，
ジャン−ミシェル アラン，
モニック ガルバーク，
ジャンヌ−マリー ルコント，
イクサビル リノー，
ヴァルター ゲー． シュナック，
ホルガー スターク，
シャロン ロビン ガネリーン，
ファビアン ルールクイン，
エルツ シグード，
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ソシエテ シヴィル ビオプロジェ
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07C217/14—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring
    • C07C217/16—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring the six-membered aromatic ring or condensed ring system containing that ring not being further substituted
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