JP2025500917A5 - - Google Patents
Info
- Publication number
- JP2025500917A5 JP2025500917A5 JP2024536124A JP2024536124A JP2025500917A5 JP 2025500917 A5 JP2025500917 A5 JP 2025500917A5 JP 2024536124 A JP2024536124 A JP 2024536124A JP 2024536124 A JP2024536124 A JP 2024536124A JP 2025500917 A5 JP2025500917 A5 JP 2025500917A5
- Authority
- JP
- Japan
- Prior art keywords
- optionally substituted
- alkyl
- pharmaceutically acceptable
- solvate
- acceptable salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163290291P | 2021-12-16 | 2021-12-16 | |
| US63/290,291 | 2021-12-16 | ||
| US202263301267P | 2022-01-20 | 2022-01-20 | |
| US63/301,267 | 2022-01-20 | ||
| US202263380049P | 2022-10-18 | 2022-10-18 | |
| US63/380,049 | 2022-10-18 | ||
| US202263386647P | 2022-12-08 | 2022-12-08 | |
| US63/386,647 | 2022-12-08 | ||
| PCT/US2022/081504 WO2023114809A1 (en) | 2021-12-16 | 2022-12-14 | Inhibitors of met kinase |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2025500917A JP2025500917A (ja) | 2025-01-15 |
| JP2025500917A5 true JP2025500917A5 (https=) | 2025-12-23 |
Family
ID=85199244
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024536124A Pending JP2025500917A (ja) | 2021-12-16 | 2022-12-14 | Metキナーゼの阻害剤 |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US11753395B2 (https=) |
| EP (1) | EP4448510A1 (https=) |
| JP (1) | JP2025500917A (https=) |
| KR (1) | KR20240121851A (https=) |
| AU (1) | AU2022413540A1 (https=) |
| CA (1) | CA3240907A1 (https=) |
| CL (1) | CL2024001756A1 (https=) |
| CO (1) | CO2024009144A2 (https=) |
| IL (1) | IL313548A (https=) |
| MX (1) | MX2024007444A (https=) |
| TW (1) | TW202333709A (https=) |
| WO (1) | WO2023114809A1 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2023114809A1 (en) | 2021-12-16 | 2023-06-22 | Kinnate Biopharma Inc. | Inhibitors of met kinase |
| CN121038792A (zh) * | 2023-04-17 | 2025-11-28 | 赛琳治疗公司 | 用met激酶抑制剂治疗癌症 |
| WO2024259060A1 (en) * | 2023-06-16 | 2024-12-19 | Kinnate Biopharma Inc. | Inhibitors of met kinase |
| WO2025096463A1 (en) * | 2023-10-30 | 2025-05-08 | Vibliome Therapeutics, Llc | Plk4 modulators |
Family Cites Families (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6334997B1 (en) | 1994-03-25 | 2002-01-01 | Isotechnika, Inc. | Method of using deuterated calcium channel blockers |
| ES2293638T3 (es) | 1994-03-25 | 2008-03-16 | Isotechnika, Inc. | Mejora de la eficacia de farmacos por deuteracion. |
| EP0860433B1 (en) | 1995-11-07 | 2002-07-03 | Kirin Beer Kabushiki Kaisha | Quinoline derivatives and quinazoline derivatives inhibiting autophosphorylation of growth factor receptor originating in platelet and pharmaceutical compositions containing the same |
| JO2785B1 (en) | 2003-05-27 | 2014-03-15 | شركة جانسين فارماسوتيكا ان. في | Quinazoline derivatives |
| US7459562B2 (en) | 2004-04-23 | 2008-12-02 | Bristol-Myers Squibb Company | Monocyclic heterocycles as kinase inhibitors |
| US7439246B2 (en) | 2004-06-28 | 2008-10-21 | Bristol-Myers Squibb Company | Fused heterocyclic kinase inhibitors |
| US20070155746A1 (en) | 2005-12-23 | 2007-07-05 | Kalypsys, Inc. | Novel substituted pyridinyloxy and pyrimidinyloxy amides useful as inhibitors of protein kinases |
| JP2009539878A (ja) | 2006-06-08 | 2009-11-19 | アレイ バイオファーマ、インコーポレイテッド | キノリン化合物および使用方法 |
| US20090049035A1 (en) | 2007-08-14 | 2009-02-19 | International Business Machines Corporation | System and method for indexing type-annotated web documents |
| JP2010126530A (ja) | 2008-12-01 | 2010-06-10 | Takeda Chem Ind Ltd | 縮合複素環誘導体およびその用途 |
| CN102573994B (zh) | 2009-08-06 | 2015-06-24 | 默克专利有限公司 | 双环脲化合物 |
| EP2423208A1 (en) | 2010-08-28 | 2012-02-29 | Lead Discovery Center GmbH | Pharmaceutically active compounds as Axl inhibitors |
| CN102827186A (zh) | 2011-06-16 | 2012-12-19 | 中国科学院上海药物研究所 | 一类吡啶并五元杂环衍生物及其制备方法和用途 |
| JP2015507606A (ja) | 2011-11-22 | 2015-03-12 | デシフェラ ファーマシューティカルズ,エルエルシー | 抗癌および抗増殖作用を示すピリドンアミドおよび類似体 |
| WO2013180949A1 (en) * | 2012-05-27 | 2013-12-05 | Ning Xi | Substituted quinoline compounds and methods of use |
| CN103508961B (zh) | 2012-06-26 | 2015-07-22 | 中美冠科生物技术(太仓)有限公司 | 抗肿瘤药物 |
| EP3003315B1 (en) | 2013-06-06 | 2018-01-17 | Lead Discovery Center GmbH | A quinoline inhibitor of the macrophage stimulating 1 receptor mst1r |
| KR101505783B1 (ko) | 2014-08-01 | 2015-03-25 | 씨제이헬스케어 주식회사 | 신규한 피롤로피리디닐옥시페닐아미드 유도체 및 이의 용도 |
| SG11201707638UA (en) | 2015-04-14 | 2017-10-30 | Qurient Co Ltd | Quinoline derivatives as tam rtk inhibitors |
| CN105153026B (zh) | 2015-08-21 | 2018-02-02 | 江西科技师范大学 | 含联芳基酰胺结构的索拉非尼衍生物及其制备方法和应用 |
| CN105732616B (zh) | 2016-01-08 | 2018-07-27 | 江西科技师范大学 | 含联芳基酰胺结构的吡咯并吡啶类化合物及其制备方法和应用 |
| CN109896997A (zh) | 2017-12-08 | 2019-06-18 | 中国药科大学 | N-酰基苯胺类c-Met激酶抑制剂的制备方法及其用途 |
| UY38349A (es) | 2018-08-30 | 2020-03-31 | Array Biopharma Inc | Compuestos de pirazolo[3,4-b]piridina como inhibidores de cinasas tam y met |
| CN111196814B (zh) | 2018-11-19 | 2022-12-06 | 北京赛特明强医药科技有限公司 | 芳环连二噁烷并喹唑啉或喹啉类化合物、组合物及其应用 |
| JP2022551422A (ja) * | 2019-09-26 | 2022-12-09 | エグゼリクシス, インコーポレイテッド | ピリドン化合物およびタンパク質キナーゼの調節における使用の方法 |
| WO2023114809A1 (en) | 2021-12-16 | 2023-06-22 | Kinnate Biopharma Inc. | Inhibitors of met kinase |
-
2022
- 2022-12-14 WO PCT/US2022/081504 patent/WO2023114809A1/en not_active Ceased
- 2022-12-14 MX MX2024007444A patent/MX2024007444A/es unknown
- 2022-12-14 JP JP2024536124A patent/JP2025500917A/ja active Pending
- 2022-12-14 CA CA3240907A patent/CA3240907A1/en active Pending
- 2022-12-14 TW TW111148006A patent/TW202333709A/zh unknown
- 2022-12-14 EP EP22854688.3A patent/EP4448510A1/en active Pending
- 2022-12-14 US US18/066,056 patent/US11753395B2/en active Active
- 2022-12-14 IL IL313548A patent/IL313548A/en unknown
- 2022-12-14 AU AU2022413540A patent/AU2022413540A1/en active Pending
- 2022-12-14 KR KR1020247023755A patent/KR20240121851A/ko active Pending
-
2023
- 2023-06-26 US US18/341,503 patent/US12595245B2/en active Active
-
2024
- 2024-06-13 CL CL2024001756A patent/CL2024001756A1/es unknown
- 2024-07-11 CO CONC2024/0009144A patent/CO2024009144A2/es unknown
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