JP2024525368A5 - - Google Patents
Info
- Publication number
- JP2024525368A5 JP2024525368A5 JP2023578050A JP2023578050A JP2024525368A5 JP 2024525368 A5 JP2024525368 A5 JP 2024525368A5 JP 2023578050 A JP2023578050 A JP 2023578050A JP 2023578050 A JP2023578050 A JP 2023578050A JP 2024525368 A5 JP2024525368 A5 JP 2024525368A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- alkylene
- disease
- condition
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163217607P | 2021-07-01 | 2021-07-01 | |
| US63/217,607 | 2021-07-01 | ||
| PCT/US2022/073385 WO2023279105A1 (en) | 2021-07-01 | 2022-07-01 | Azetidinyl pyrimidines and uses thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024525368A JP2024525368A (ja) | 2024-07-12 |
| JP2024525368A5 true JP2024525368A5 (https=) | 2025-06-27 |
Family
ID=82799923
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023578050A Pending JP2024525368A (ja) | 2021-07-01 | 2022-07-01 | アゼチジニルピリミジンおよびその使用 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20240425496A1 (https=) |
| EP (1) | EP4363058A1 (https=) |
| JP (1) | JP2024525368A (https=) |
| KR (1) | KR20240031347A (https=) |
| CN (1) | CN117642395A (https=) |
| AU (2) | AU2022304597C1 (https=) |
| CA (1) | CA3225872A1 (https=) |
| IL (1) | IL309892A (https=) |
| MX (1) | MX2024000273A (https=) |
| WO (1) | WO2023279105A1 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA3260763A1 (en) * | 2022-06-29 | 2024-01-04 | Alcon Inc. | AZETIDINYL PYRIMIDINES AND THEIR USES AS JAK INHIBITORS |
| WO2024148184A1 (en) * | 2023-01-04 | 2024-07-11 | Aerie Pharmaceuticals, Inc. | Compounds and processes for the preparation of jak inhibitors |
| WO2024148186A1 (en) | 2023-01-04 | 2024-07-11 | Aerie Pharmaceuticals, Inc. | Polymorphs of a jak1/tyk2 inhibitor and uses thereof |
| CN116903592B (zh) * | 2023-07-13 | 2025-08-01 | 特科罗生物科技(成都)有限公司 | 一种嘧啶胺类nuak抑制剂及其制备方法和用途 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2634646C (en) * | 2005-12-21 | 2012-04-10 | Pfizer Products Inc. | Pyrimidine derivatives for the treatment of abnormal cell growth |
| WO2008132502A1 (en) * | 2007-04-25 | 2008-11-06 | Astrazeneca Ab | Pyrazolyl-amino-substituted pyrimidines and their use for the treatment of cancer |
| MX2010013726A (es) * | 2008-06-12 | 2011-01-14 | Janssen Pharmaceutica Nv | Moduladores de diamino-piridina, pirimidina, y piridazina del receptor h4 de histamina. |
| CN110621316B (zh) * | 2017-04-21 | 2024-01-26 | Epizyme股份有限公司 | 用ehmt2抑制剂进行的组合疗法 |
| WO2020108516A1 (zh) * | 2018-11-27 | 2020-06-04 | 江苏豪森药业集团有限公司 | 含氮杂芳类衍生物调节剂、其制备方法和应用 |
| CN110317176A (zh) * | 2019-07-04 | 2019-10-11 | 沈阳药科大学 | 2-氨基嘧啶类化合物及其用途 |
| TW202227418A (zh) * | 2020-10-12 | 2022-07-16 | 大陸商四川海思科製藥有限公司 | 一種雜環衍生物及其在醫藥上的應用 |
| KR102585193B1 (ko) * | 2021-04-08 | 2023-10-06 | 주식회사 스탠다임 | 신규한 lrrk2 억제제 |
-
2022
- 2022-07-01 JP JP2023578050A patent/JP2024525368A/ja active Pending
- 2022-07-01 WO PCT/US2022/073385 patent/WO2023279105A1/en not_active Ceased
- 2022-07-01 KR KR1020247003795A patent/KR20240031347A/ko active Pending
- 2022-07-01 CA CA3225872A patent/CA3225872A1/en active Pending
- 2022-07-01 EP EP22751232.4A patent/EP4363058A1/en active Pending
- 2022-07-01 IL IL309892A patent/IL309892A/en unknown
- 2022-07-01 US US18/573,305 patent/US20240425496A1/en active Pending
- 2022-07-01 AU AU2022304597A patent/AU2022304597C1/en active Active
- 2022-07-01 MX MX2024000273A patent/MX2024000273A/es unknown
- 2022-07-01 CN CN202280047279.1A patent/CN117642395A/zh active Pending
-
2025
- 2025-10-20 AU AU2025252656A patent/AU2025252656A1/en active Pending
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