JP2024529527A5 - - Google Patents
Info
- Publication number
- JP2024529527A5 JP2024529527A5 JP2024506443A JP2024506443A JP2024529527A5 JP 2024529527 A5 JP2024529527 A5 JP 2024529527A5 JP 2024506443 A JP2024506443 A JP 2024506443A JP 2024506443 A JP2024506443 A JP 2024506443A JP 2024529527 A5 JP2024529527 A5 JP 2024529527A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- groups
- alkyl
- halogenated
- alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202110892791.3 | 2021-08-04 | ||
| CN202110892791 | 2021-08-04 | ||
| CN202111322097.4 | 2021-11-09 | ||
| CN202111322097 | 2021-11-09 | ||
| CN202210041958.X | 2022-01-14 | ||
| CN202210041958 | 2022-01-14 | ||
| CN202210540040 | 2022-05-17 | ||
| CN202210540040.X | 2022-05-17 | ||
| PCT/CN2022/110017 WO2023011539A1 (zh) | 2021-08-04 | 2022-08-03 | 环烯类衍生物调节剂、其制备方法和应用 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024529527A JP2024529527A (ja) | 2024-08-06 |
| JP2024529527A5 true JP2024529527A5 (https=) | 2025-07-31 |
Family
ID=85155248
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024506443A Pending JP2024529527A (ja) | 2021-08-04 | 2022-08-03 | シクロアルケン系誘導体調節剤、その製造方法及び応用 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20240360109A1 (https=) |
| EP (1) | EP4382525A4 (https=) |
| JP (1) | JP2024529527A (https=) |
| KR (1) | KR20240042624A (https=) |
| CN (1) | CN117751110A (https=) |
| AU (1) | AU2022321506A1 (https=) |
| CA (1) | CA3227366A1 (https=) |
| IL (1) | IL310400A (https=) |
| MX (1) | MX2024001331A (https=) |
| TW (1) | TW202321227A (https=) |
| WO (1) | WO2023011539A1 (https=) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA3188891A1 (en) | 2020-09-01 | 2022-01-13 | Fanglong Yang | Fused imidazole derivative, preparation method therefor, and medical use thereof |
| PT4408840T (pt) | 2021-09-27 | 2025-10-07 | Terns Pharmaceuticals Inc | Ácidos benzimidazolocarboxílicos como agonistas de glp-1r |
| CN118401519A (zh) | 2021-10-25 | 2024-07-26 | 拓臻制药公司 | 作为glp-1r激动剂的化合物 |
| CN119095843A (zh) | 2022-02-23 | 2024-12-06 | 拓臻制药公司 | 作为glp-1r激动剂的化合物 |
| TW202434574A (zh) * | 2023-02-02 | 2024-09-01 | 大陸商江蘇豪森藥業集團有限公司 | 一種環烯類化合物的鹽、晶型及其製備方法和應用 |
| EP4568664B1 (en) | 2023-04-07 | 2026-04-01 | Terns Pharmaceuticals, Inc. | Combination comprising a thr-beta agonist and a glp-1r agonist for use in treating obesity |
| CN120981457A (zh) | 2023-09-14 | 2025-11-18 | 歌礼制药(中国)有限公司 | Glp-1r激动剂及其治疗方法 |
| TW202521534A (zh) | 2023-11-24 | 2025-06-01 | 香港商歌禮製藥(中國)有限公司 | Glp-1r 激動劑及其治療方法 |
| WO2025247390A1 (zh) * | 2024-05-31 | 2025-12-04 | 福佑泰生物制药公司 | 可用作glp-1r激动剂的杂双环化合物 |
| WO2025252201A1 (zh) * | 2024-06-07 | 2025-12-11 | 江苏豪森药业集团有限公司 | 一种环烯类衍生物的制备方法 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2016022742A1 (en) * | 2014-08-08 | 2016-02-11 | Merck Sharp & Dohme Corp. | Antidiabetic bicyclic compounds |
| KR102314286B1 (ko) * | 2016-12-16 | 2021-10-21 | 화이자 인코포레이티드 | Glp-1 수용체 작용제 및 이의 용도 |
| US10934279B2 (en) * | 2018-06-13 | 2021-03-02 | Pfizer Inc. | GLP-1 receptor agonists and uses thereof |
| DK3806855T5 (da) * | 2018-06-15 | 2023-05-22 | Pfizer | GLP-1-receptoragonister og anvendelser deraf |
| MA54555A (fr) * | 2018-11-22 | 2021-09-29 | Qilu Regor Therapeutics Inc | Agonistes de glp-1r et leurs utilisations |
| EP3953344A4 (en) * | 2019-04-12 | 2023-08-09 | Qilu Regor Therapeutics Inc. | GLP-IR AGONISTS AND THEIR USES |
| WO2021018023A1 (zh) * | 2019-08-01 | 2021-02-04 | 济南泰达领创医药技术有限公司 | 小分子glp-1受体调节剂 |
| EP4048664A1 (en) * | 2019-10-25 | 2022-08-31 | Gilead Sciences, Inc. | Glp-1r modulating compounds |
| WO2021096284A1 (ko) * | 2019-11-15 | 2021-05-20 | 일동제약(주) | Glp-1 수용체 작용제 및 이의 용도 |
| TW202206429A (zh) * | 2020-04-29 | 2022-02-16 | 美商迦舒布魯姆生物有限公司 | 雜環glp—1促效劑 |
| CA3192601A1 (en) * | 2020-08-21 | 2022-02-24 | Terns Pharmaceuticals, Inc. | Compounds as glp-1r agonists |
| CA3188891A1 (en) * | 2020-09-01 | 2022-01-13 | Fanglong Yang | Fused imidazole derivative, preparation method therefor, and medical use thereof |
| EP4229050A4 (en) * | 2020-10-13 | 2024-12-11 | Gasherbrum Bio, Inc. | Heterocyclic glp-1 agonists |
| CN114805336B (zh) * | 2021-01-20 | 2026-04-14 | 江苏恒瑞医药股份有限公司 | 稠合咪唑类化合物、其制备方法及其在医药上的应用 |
-
2022
- 2022-08-03 WO PCT/CN2022/110017 patent/WO2023011539A1/zh not_active Ceased
- 2022-08-03 KR KR1020247006472A patent/KR20240042624A/ko active Pending
- 2022-08-03 IL IL310400A patent/IL310400A/en unknown
- 2022-08-03 JP JP2024506443A patent/JP2024529527A/ja active Pending
- 2022-08-03 MX MX2024001331A patent/MX2024001331A/es unknown
- 2022-08-03 CN CN202280053790.2A patent/CN117751110A/zh active Pending
- 2022-08-03 AU AU2022321506A patent/AU2022321506A1/en active Pending
- 2022-08-03 US US18/293,637 patent/US20240360109A1/en active Pending
- 2022-08-03 CA CA3227366A patent/CA3227366A1/en active Pending
- 2022-08-03 EP EP22852251.2A patent/EP4382525A4/en active Pending
- 2022-08-04 TW TW111129379A patent/TW202321227A/zh unknown
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