JP2022507065A5 - - Google Patents

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Publication number
JP2022507065A5
JP2022507065A5 JP2021525223A JP2021525223A JP2022507065A5 JP 2022507065 A5 JP2022507065 A5 JP 2022507065A5 JP 2021525223 A JP2021525223 A JP 2021525223A JP 2021525223 A JP2021525223 A JP 2021525223A JP 2022507065 A5 JP2022507065 A5 JP 2022507065A5
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JP
Japan
Application number
JP2021525223A
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Japanese (ja)
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JP2022507065A (ja
JPWO2020102096A5 (https=
JP7730759B2 (ja
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Priority claimed from PCT/US2019/060770 external-priority patent/WO2020102096A1/en
Publication of JP2022507065A publication Critical patent/JP2022507065A/ja
Publication of JPWO2020102096A5 publication Critical patent/JPWO2020102096A5/ja
Publication of JP2022507065A5 publication Critical patent/JP2022507065A5/ja
Priority to JP2024091521A priority Critical patent/JP2024113083A/ja
Application granted granted Critical
Publication of JP7730759B2 publication Critical patent/JP7730759B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021525223A 2018-11-13 2019-11-11 Nlrp活性に関連する病態を治療するための化合物及び組成物 Active JP7730759B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024091521A JP2024113083A (ja) 2018-11-13 2024-06-05 Nlrp活性に関連する病態を治療するための化合物及び組成物

Applications Claiming Priority (27)

Application Number Priority Date Filing Date Title
US201862760248P 2018-11-13 2018-11-13
US201862760244P 2018-11-13 2018-11-13
US201862760209P 2018-11-13 2018-11-13
US62/760,209 2018-11-13
US62/760,244 2018-11-13
US62/760,248 2018-11-13
US201862768811P 2018-11-16 2018-11-16
US62/768,811 2018-11-16
US201862769151P 2018-11-19 2018-11-19
US201862769165P 2018-11-19 2018-11-19
US62/769,165 2018-11-19
US62/769,151 2018-11-19
US201962795919P 2019-01-23 2019-01-23
US62/795,919 2019-01-23
US201962796356P 2019-01-24 2019-01-24
US201962796361P 2019-01-24 2019-01-24
US62/796,361 2019-01-24
US62/796,356 2019-01-24
US201962836577P 2019-04-19 2019-04-19
US201962836585P 2019-04-19 2019-04-19
US201962836575P 2019-04-19 2019-04-19
US62/836,585 2019-04-19
US62/836,577 2019-04-19
US62/836,575 2019-04-19
US201962895595P 2019-09-04 2019-09-04
US62/895,595 2019-09-04
PCT/US2019/060770 WO2020102096A1 (en) 2018-11-13 2019-11-11 Compounds and compositions for treating conditions associated with nlrp activity

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024091521A Division JP2024113083A (ja) 2018-11-13 2024-06-05 Nlrp活性に関連する病態を治療するための化合物及び組成物

Publications (4)

Publication Number Publication Date
JP2022507065A JP2022507065A (ja) 2022-01-18
JPWO2020102096A5 JPWO2020102096A5 (https=) 2022-11-22
JP2022507065A5 true JP2022507065A5 (https=) 2022-11-22
JP7730759B2 JP7730759B2 (ja) 2025-08-28

Family

ID=68841175

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021525223A Active JP7730759B2 (ja) 2018-11-13 2019-11-11 Nlrp活性に関連する病態を治療するための化合物及び組成物
JP2024091521A Pending JP2024113083A (ja) 2018-11-13 2024-06-05 Nlrp活性に関連する病態を治療するための化合物及び組成物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024091521A Pending JP2024113083A (ja) 2018-11-13 2024-06-05 Nlrp活性に関連する病態を治療するための化合物及び組成物

Country Status (31)

Country Link
US (1) US20230031406A1 (https=)
EP (2) EP3880660B1 (https=)
JP (2) JP7730759B2 (https=)
KR (1) KR20210096123A (https=)
CN (2) CN113166065B (https=)
AU (1) AU2019379109B2 (https=)
BR (1) BR112021008969A2 (https=)
CA (1) CA3114918A1 (https=)
CL (1) CL2021001228A1 (https=)
CO (1) CO2021006075A2 (https=)
CR (1) CR20210235A (https=)
DK (1) DK3880660T3 (https=)
EC (2) ECSP21033236A (https=)
ES (1) ES3042546T3 (https=)
FI (1) FI3880660T3 (https=)
HR (1) HRP20251344T1 (https=)
HU (1) HUE073575T2 (https=)
IL (1) IL283042B2 (https=)
JO (1) JOP20210105B1 (https=)
LT (1) LT3880660T (https=)
MA (1) MA54229B1 (https=)
MX (1) MX2021005529A (https=)
MY (1) MY206733A (https=)
PE (1) PE20211698A1 (https=)
PH (1) PH12021500025A1 (https=)
PL (1) PL3880660T3 (https=)
PT (1) PT3880660T (https=)
RS (1) RS67257B1 (https=)
SG (1) SG11202103405TA (https=)
SI (1) SI3880660T1 (https=)
WO (1) WO2020102096A1 (https=)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3649112A1 (en) * 2017-07-07 2020-05-13 Inflazome Limited Sulfonylureas and sulfonylthioureas as nlrp3 inhibitors
EP3668843A1 (en) 2017-08-15 2020-06-24 Inflazome Limited Sulfonylureas and sulfonylthioureas as nlrp3 inhibitors
MA49903A (fr) 2017-08-15 2020-06-24 Inflazome Ltd Sulfonylureés et sulfonylthioureés en tant qu'inhibiteurs de nlrp3
UY37848A (es) 2017-08-15 2019-03-29 Inflazome Ltd Sulfonilureas y sulfoniltioureas útiles como inhibidores de nlrp3
WO2019092171A1 (en) 2017-11-09 2019-05-16 Inflazome Limited Novel sulfonamide carboxamide compounds
CN111315733A (zh) 2017-11-09 2020-06-19 英夫拉索姆有限公司 新颖磺酰胺甲酰胺化合物
US11905252B2 (en) 2018-03-02 2024-02-20 Inflazome Limited Compounds
CA3105521A1 (en) 2018-07-20 2020-01-23 F. Hoffmann-La Roche Ag Sulfonimidamide compounds as inhibitors of interleukin-1 activity
JP7392169B2 (ja) * 2019-11-12 2023-12-05 成都百裕制薬股▲ふん▼有限公司 アミド誘導体及びその調製方法並びに医薬における応用
PH12022551767A1 (en) * 2020-01-22 2023-11-29 Hoffmann La Roche Sulfonimidamide compounds as nlrp3 modulators
WO2022023907A1 (en) 2020-07-31 2022-02-03 Novartis Ag Methods of selecting and treating patients at elevated risk of major adverse cardiac events
CN117279903A (zh) * 2021-02-10 2023-12-22 杭州英创医药科技有限公司 作为nlrp3抑制剂的化合物
US11932630B2 (en) 2021-04-16 2024-03-19 Novartis Ag Heteroaryl aminopropanol derivatives
CN116635373A (zh) * 2021-05-10 2023-08-22 成都百裕制药股份有限公司 酰胺衍生物及其应用
CN116917282A (zh) * 2021-05-10 2023-10-20 成都百裕制药股份有限公司 酰胺衍生物及其应用
CN116635374B (zh) * 2021-05-10 2025-05-06 康百达(四川)生物医药科技有限公司 酰胺衍生物及其应用
CN114989058B (zh) * 2022-06-02 2024-04-16 中国科学院成都生物研究所 一种手性氯代砜亚胺类化合物及其衍生物的制备方法
CN115974745B (zh) * 2022-12-27 2025-06-03 瑞石生物医药有限公司 一类含引达省的化合物及其医药用途
CN116253664A (zh) * 2023-02-01 2023-06-13 山东海科创新研究院有限公司 基于双液相微乳化缩合工艺的accp制备方法
WO2025153532A1 (en) 2024-01-16 2025-07-24 NodThera Limited Nlrp3 inhibitors and glp-1 agonists combination therapies

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI3259253T1 (sl) * 2015-02-16 2020-07-31 The University Of Queensland Sulfonilsečnine in sorodne spojine ter njihova uporaba
US11339136B2 (en) * 2016-04-18 2022-05-24 Novartis Ag Compounds and compositions for treating conditions associated with NLRP activity
JP7349981B2 (ja) * 2017-07-24 2023-09-25 ノバルティス アーゲー Nlrp活性に関連する状態を治療するための化合物及び組成物
ES2988798T3 (es) * 2017-07-24 2024-11-21 Novartis Ag Compuestos y composiciones para el tratamiento de afecciones asociadas a la actividad de NLRP
CA3105521A1 (en) * 2018-07-20 2020-01-23 F. Hoffmann-La Roche Ag Sulfonimidamide compounds as inhibitors of interleukin-1 activity

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