JP2024524658A5 - - Google Patents
Info
- Publication number
- JP2024524658A5 JP2024524658A5 JP2024501708A JP2024501708A JP2024524658A5 JP 2024524658 A5 JP2024524658 A5 JP 2024524658A5 JP 2024501708 A JP2024501708 A JP 2024501708A JP 2024501708 A JP2024501708 A JP 2024501708A JP 2024524658 A5 JP2024524658 A5 JP 2024524658A5
- Authority
- JP
- Japan
- Prior art keywords
- hydrochloride salt
- reaction
- alkyl
- mixture
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EPPCT/EP2021/069486 | 2021-07-13 | ||
| EP2021069486 | 2021-07-13 | ||
| PCT/EP2022/069238 WO2023285342A2 (en) | 2021-07-13 | 2022-07-11 | A process for the synthesis of 4-((r)-2-{[6-((s)-3-methoxy-pyrrolidin-1-yl)-2-phenyl- pyrimidine-4-carbonyl]-amino}-3-phosphono-propionyl)-piperazine-1 -carboxylic acid butyl ester |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024524658A JP2024524658A (ja) | 2024-07-05 |
| JP2024524658A5 true JP2024524658A5 (https=) | 2025-07-02 |
Family
ID=82748669
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024501708A Pending JP2024524658A (ja) | 2021-07-13 | 2022-07-11 | 4-((r)-2-{[6-((s)-3-メトキシ-ピロリジン-1-イル)-2-フェニル-ピリミジン-4-カルボニル]-アミノ}-3-ホスホノ-プロピオニル)-ピペラジン-1-カルボン酸ブチルエステルの合成方法 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20240317784A1 (https=) |
| EP (1) | EP4370525A2 (https=) |
| JP (1) | JP2024524658A (https=) |
| KR (1) | KR20240033005A (https=) |
| CN (1) | CN117616033A (https=) |
| CA (1) | CA3223733A1 (https=) |
| IL (1) | IL309948A (https=) |
| MX (1) | MX2024000653A (https=) |
| TW (1) | TW202317140A (https=) |
| WO (1) | WO2023285342A2 (https=) |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2225253B1 (en) * | 2007-11-29 | 2012-06-27 | Actelion Pharmaceuticals Ltd. | Phosphonic acid derivates and their use as p2y12 receptor antagonists |
| EP3515924B1 (en) * | 2016-09-22 | 2021-12-15 | Idorsia Pharmaceuticals Ltd | Crystalline forms |
| MA49887A (fr) | 2017-03-15 | 2020-06-24 | Idorsia Pharmaceuticals Ltd | Administration sous-cutanée d'un antagoniste du récepteur p2y12 |
-
2022
- 2022-07-11 MX MX2024000653A patent/MX2024000653A/es unknown
- 2022-07-11 JP JP2024501708A patent/JP2024524658A/ja active Pending
- 2022-07-11 US US18/579,110 patent/US20240317784A1/en active Pending
- 2022-07-11 KR KR1020247004672A patent/KR20240033005A/ko active Pending
- 2022-07-11 WO PCT/EP2022/069238 patent/WO2023285342A2/en not_active Ceased
- 2022-07-11 EP EP22748321.1A patent/EP4370525A2/en active Pending
- 2022-07-11 CA CA3223733A patent/CA3223733A1/en active Pending
- 2022-07-11 CN CN202280048853.5A patent/CN117616033A/zh active Pending
- 2022-07-11 IL IL309948A patent/IL309948A/en unknown
- 2022-07-12 TW TW111126010A patent/TW202317140A/zh unknown
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