JP2024518554A5 - - Google Patents

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Publication number
JP2024518554A5
JP2024518554A5 JP2023570165A JP2023570165A JP2024518554A5 JP 2024518554 A5 JP2024518554 A5 JP 2024518554A5 JP 2023570165 A JP2023570165 A JP 2023570165A JP 2023570165 A JP2023570165 A JP 2023570165A JP 2024518554 A5 JP2024518554 A5 JP 2024518554A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
alkyl
diluent
acceptable salt
pharmaceutical composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023570165A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024518554A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/029102 external-priority patent/WO2022241171A1/en
Publication of JP2024518554A publication Critical patent/JP2024518554A/ja
Publication of JP2024518554A5 publication Critical patent/JP2024518554A5/ja
Pending legal-status Critical Current

Links

JP2023570165A 2021-05-14 2022-05-13 置換ヘテロ環化合物 Pending JP2024518554A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202163188498P 2021-05-14 2021-05-14
US63/188,498 2021-05-14
US202263318149P 2022-03-09 2022-03-09
US63/318,149 2022-03-09
PCT/US2022/029102 WO2022241171A1 (en) 2021-05-14 2022-05-13 Substituted heterocyclic compounds

Publications (2)

Publication Number Publication Date
JP2024518554A JP2024518554A (ja) 2024-05-01
JP2024518554A5 true JP2024518554A5 (enExample) 2025-03-12

Family

ID=81927926

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023570165A Pending JP2024518554A (ja) 2021-05-14 2022-05-13 置換ヘテロ環化合物

Country Status (13)

Country Link
US (3) US11866414B2 (enExample)
EP (1) EP4337655A1 (enExample)
JP (1) JP2024518554A (enExample)
KR (1) KR20240008336A (enExample)
AU (1) AU2022271794A1 (enExample)
CA (1) CA3217332A1 (enExample)
CL (1) CL2023003308A1 (enExample)
CO (1) CO2023015226A2 (enExample)
IL (1) IL308421A (enExample)
MX (1) MX2023013445A (enExample)
PE (1) PE20250262A1 (enExample)
TW (1) TW202311247A (enExample)
WO (1) WO2022241171A1 (enExample)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102858043B1 (ko) * 2018-10-30 2025-09-10 브리스톨-마이어스 스큅 컴퍼니 Il-12, il-23 및/또는 ifn-알파의 조정과 관련된 상태의 치료를 위한 아미드-치환된 헤테로시클릭 화합물
WO2021226208A2 (en) 2020-05-05 2021-11-11 Nuvalent, Inc. Heteroaromatic macrocyclic ether chemotherapeutic agents
KR102698413B1 (ko) 2020-05-05 2024-08-26 뉴베일런트, 아이엔씨. 헤테로방향족 거대환식 에터 화학치료제
CN122520625A (zh) 2020-12-22 2026-08-07 益方生物科技(上海)股份有限公司 杂芳基化合物及其制备方法和用途
US12668594B2 (en) 2020-12-23 2026-06-30 Sudo Biosciences Limited TYK2 inhibitors and uses thereof
KR20230159421A (ko) 2021-02-19 2023-11-21 수도 바이오사이언시즈 리미티드 Tyk2 억제제 및 이의 용도
TW202302583A (zh) 2021-02-19 2023-01-16 英商蘇多生物科學有限公司 Tyk2抑制劑及其用途
IL305119A (en) 2021-02-19 2023-10-01 Sudo Biosciences Ltd Tyk2 inhibitors and uses thereof
WO2022212489A1 (en) 2021-03-31 2022-10-06 Xinthera, Inc. Mk2 inhibitors and uses thereof
EP4337650A1 (en) * 2021-05-14 2024-03-20 Bristol-Myers Squibb Company Substituted heterocyclic compounds
PE20250262A1 (es) * 2021-05-14 2025-01-29 Bristol Myers Squibb Co Compuestos heterociclicos sustituidos
US20240317718A1 (en) * 2021-05-14 2024-09-26 Bristol-Myers Squibb Company Substituted heterocyclic compounds
KR20240008338A (ko) * 2021-05-14 2024-01-18 브리스톨-마이어스 스큅 컴퍼니 치환된 헤테로시클릭 화합물
KR20240007242A (ko) * 2021-05-14 2024-01-16 브리스톨-마이어스 스큅 컴퍼니 치환된 헤테로시클릭 화합물
CN115724830A (zh) * 2021-08-31 2023-03-03 浙江文达医药科技有限公司 作为tyk2/jak1假激酶结构域(jh2)抑制剂的化合物及合成和使用方法
TW202320768A (zh) 2021-10-01 2023-06-01 美商努法倫特公司 雜芳族大環醚化合物之固體形式、醫藥組成物及製備
CN117263913A (zh) 2022-06-20 2023-12-22 益方生物科技(上海)股份有限公司 杂芳基化合物、固体形式、制备方法及其用途
WO2024044486A1 (en) * 2022-08-22 2024-02-29 Ajax Therapeutics, Inc. Jak2 inhibitor compounds
CN120152968A (zh) * 2022-11-08 2025-06-13 百时美施贵宝公司 取代的杂环化合物
CN118812511A (zh) * 2023-04-21 2024-10-22 浙江文达医药科技有限公司 作为tyk2抑制剂的杂环化合物及合成和应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP20220766T1 (hr) * 2012-11-08 2022-09-16 Bristol-Myers Squibb Company Amidom-supstituirani heterociklički spojevi korisni kao modulatori il-12, il-23 i/ili ifn alfa odgovora
LT3601268T (lt) 2017-03-30 2021-05-25 Bristol-Myers Squibb Company 6-(ciklopropanamido)-4-((2-metoksi-3-(1-metil-1h-1,2,4-triazol-3-il)fenil)amino)-n-(metil-d3)piridazino-3-karboksamido gavimo būdas
PE20250262A1 (es) * 2021-05-14 2025-01-29 Bristol Myers Squibb Co Compuestos heterociclicos sustituidos

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