JP2024518554A5 - - Google Patents
Info
- Publication number
- JP2024518554A5 JP2024518554A5 JP2023570165A JP2023570165A JP2024518554A5 JP 2024518554 A5 JP2024518554 A5 JP 2024518554A5 JP 2023570165 A JP2023570165 A JP 2023570165A JP 2023570165 A JP2023570165 A JP 2023570165A JP 2024518554 A5 JP2024518554 A5 JP 2024518554A5
- Authority
- JP
- Japan
- Prior art keywords
- pharmaceutically acceptable
- alkyl
- diluent
- acceptable salt
- pharmaceutical composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163188498P | 2021-05-14 | 2021-05-14 | |
| US63/188,498 | 2021-05-14 | ||
| US202263318149P | 2022-03-09 | 2022-03-09 | |
| US63/318,149 | 2022-03-09 | ||
| PCT/US2022/029102 WO2022241171A1 (en) | 2021-05-14 | 2022-05-13 | Substituted heterocyclic compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024518554A JP2024518554A (ja) | 2024-05-01 |
| JP2024518554A5 true JP2024518554A5 (enExample) | 2025-03-12 |
Family
ID=81927926
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023570165A Pending JP2024518554A (ja) | 2021-05-14 | 2022-05-13 | 置換ヘテロ環化合物 |
Country Status (13)
| Country | Link |
|---|---|
| US (3) | US11866414B2 (enExample) |
| EP (1) | EP4337655A1 (enExample) |
| JP (1) | JP2024518554A (enExample) |
| KR (1) | KR20240008336A (enExample) |
| AU (1) | AU2022271794A1 (enExample) |
| CA (1) | CA3217332A1 (enExample) |
| CL (1) | CL2023003308A1 (enExample) |
| CO (1) | CO2023015226A2 (enExample) |
| IL (1) | IL308421A (enExample) |
| MX (1) | MX2023013445A (enExample) |
| PE (1) | PE20250262A1 (enExample) |
| TW (1) | TW202311247A (enExample) |
| WO (1) | WO2022241171A1 (enExample) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102858043B1 (ko) * | 2018-10-30 | 2025-09-10 | 브리스톨-마이어스 스큅 컴퍼니 | Il-12, il-23 및/또는 ifn-알파의 조정과 관련된 상태의 치료를 위한 아미드-치환된 헤테로시클릭 화합물 |
| WO2021226208A2 (en) | 2020-05-05 | 2021-11-11 | Nuvalent, Inc. | Heteroaromatic macrocyclic ether chemotherapeutic agents |
| KR102698413B1 (ko) | 2020-05-05 | 2024-08-26 | 뉴베일런트, 아이엔씨. | 헤테로방향족 거대환식 에터 화학치료제 |
| CN122520625A (zh) | 2020-12-22 | 2026-08-07 | 益方生物科技(上海)股份有限公司 | 杂芳基化合物及其制备方法和用途 |
| US12668594B2 (en) | 2020-12-23 | 2026-06-30 | Sudo Biosciences Limited | TYK2 inhibitors and uses thereof |
| KR20230159421A (ko) | 2021-02-19 | 2023-11-21 | 수도 바이오사이언시즈 리미티드 | Tyk2 억제제 및 이의 용도 |
| TW202302583A (zh) | 2021-02-19 | 2023-01-16 | 英商蘇多生物科學有限公司 | Tyk2抑制劑及其用途 |
| IL305119A (en) | 2021-02-19 | 2023-10-01 | Sudo Biosciences Ltd | Tyk2 inhibitors and uses thereof |
| WO2022212489A1 (en) | 2021-03-31 | 2022-10-06 | Xinthera, Inc. | Mk2 inhibitors and uses thereof |
| EP4337650A1 (en) * | 2021-05-14 | 2024-03-20 | Bristol-Myers Squibb Company | Substituted heterocyclic compounds |
| PE20250262A1 (es) * | 2021-05-14 | 2025-01-29 | Bristol Myers Squibb Co | Compuestos heterociclicos sustituidos |
| US20240317718A1 (en) * | 2021-05-14 | 2024-09-26 | Bristol-Myers Squibb Company | Substituted heterocyclic compounds |
| KR20240008338A (ko) * | 2021-05-14 | 2024-01-18 | 브리스톨-마이어스 스큅 컴퍼니 | 치환된 헤테로시클릭 화합물 |
| KR20240007242A (ko) * | 2021-05-14 | 2024-01-16 | 브리스톨-마이어스 스큅 컴퍼니 | 치환된 헤테로시클릭 화합물 |
| CN115724830A (zh) * | 2021-08-31 | 2023-03-03 | 浙江文达医药科技有限公司 | 作为tyk2/jak1假激酶结构域(jh2)抑制剂的化合物及合成和使用方法 |
| TW202320768A (zh) | 2021-10-01 | 2023-06-01 | 美商努法倫特公司 | 雜芳族大環醚化合物之固體形式、醫藥組成物及製備 |
| CN117263913A (zh) | 2022-06-20 | 2023-12-22 | 益方生物科技(上海)股份有限公司 | 杂芳基化合物、固体形式、制备方法及其用途 |
| WO2024044486A1 (en) * | 2022-08-22 | 2024-02-29 | Ajax Therapeutics, Inc. | Jak2 inhibitor compounds |
| CN120152968A (zh) * | 2022-11-08 | 2025-06-13 | 百时美施贵宝公司 | 取代的杂环化合物 |
| CN118812511A (zh) * | 2023-04-21 | 2024-10-22 | 浙江文达医药科技有限公司 | 作为tyk2抑制剂的杂环化合物及合成和应用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HRP20220766T1 (hr) * | 2012-11-08 | 2022-09-16 | Bristol-Myers Squibb Company | Amidom-supstituirani heterociklički spojevi korisni kao modulatori il-12, il-23 i/ili ifn alfa odgovora |
| LT3601268T (lt) | 2017-03-30 | 2021-05-25 | Bristol-Myers Squibb Company | 6-(ciklopropanamido)-4-((2-metoksi-3-(1-metil-1h-1,2,4-triazol-3-il)fenil)amino)-n-(metil-d3)piridazino-3-karboksamido gavimo būdas |
| PE20250262A1 (es) * | 2021-05-14 | 2025-01-29 | Bristol Myers Squibb Co | Compuestos heterociclicos sustituidos |
-
2022
- 2022-05-13 PE PE2023003027A patent/PE20250262A1/es unknown
- 2022-05-13 US US17/743,557 patent/US11866414B2/en active Active
- 2022-05-13 AU AU2022271794A patent/AU2022271794A1/en active Pending
- 2022-05-13 TW TW111118122A patent/TW202311247A/zh unknown
- 2022-05-13 MX MX2023013445A patent/MX2023013445A/es unknown
- 2022-05-13 IL IL308421A patent/IL308421A/en unknown
- 2022-05-13 CA CA3217332A patent/CA3217332A1/en active Pending
- 2022-05-13 EP EP22727672.2A patent/EP4337655A1/en active Pending
- 2022-05-13 WO PCT/US2022/029102 patent/WO2022241171A1/en not_active Ceased
- 2022-05-13 KR KR1020237042720A patent/KR20240008336A/ko active Pending
- 2022-05-13 JP JP2023570165A patent/JP2024518554A/ja active Pending
-
2023
- 2023-11-07 CL CL2023003308A patent/CL2023003308A1/es unknown
- 2023-11-09 CO CONC2023/0015226A patent/CO2023015226A2/es unknown
- 2023-11-30 US US18/524,426 patent/US20240190829A1/en not_active Abandoned
-
2024
- 2024-12-11 US US18/976,869 patent/US20250163004A1/en active Pending
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