JP2023552490A5 - - Google Patents

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Publication number
JP2023552490A5
JP2023552490A5 JP2023548533A JP2023548533A JP2023552490A5 JP 2023552490 A5 JP2023552490 A5 JP 2023552490A5 JP 2023548533 A JP2023548533 A JP 2023548533A JP 2023548533 A JP2023548533 A JP 2023548533A JP 2023552490 A5 JP2023552490 A5 JP 2023552490A5
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JP
Japan
Prior art keywords
alkyl
ring
optionally substituted
cycloalkyl
independently selected
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023548533A
Other languages
English (en)
Japanese (ja)
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JP2023552490A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/055165 external-priority patent/WO2022093552A2/en
Publication of JP2023552490A publication Critical patent/JP2023552490A/ja
Publication of JP2023552490A5 publication Critical patent/JP2023552490A5/ja
Pending legal-status Critical Current

Links

JP2023548533A 2020-10-16 2021-10-15 Rev-erbアゴニスト Pending JP2023552490A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063092893P 2020-10-16 2020-10-16
US63/092,893 2020-10-16
PCT/US2021/055165 WO2022093552A2 (en) 2020-10-16 2021-10-15 Rev-erb agonists

Publications (2)

Publication Number Publication Date
JP2023552490A JP2023552490A (ja) 2023-12-15
JP2023552490A5 true JP2023552490A5 (cg-RX-API-DMAC7.html) 2024-10-21

Family

ID=81384462

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023548533A Pending JP2023552490A (ja) 2020-10-16 2021-10-15 Rev-erbアゴニスト

Country Status (7)

Country Link
US (1) US20240002380A1 (cg-RX-API-DMAC7.html)
EP (1) EP4228632A4 (cg-RX-API-DMAC7.html)
JP (1) JP2023552490A (cg-RX-API-DMAC7.html)
CN (1) CN116635029A (cg-RX-API-DMAC7.html)
AU (1) AU2021372389A1 (cg-RX-API-DMAC7.html)
CA (1) CA3195127A1 (cg-RX-API-DMAC7.html)
WO (1) WO2022093552A2 (cg-RX-API-DMAC7.html)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN114432302B (zh) * 2020-11-05 2024-08-27 中国科学院上海营养与健康研究所 小分子sr9009在抗衰老以及减轻衰老引起的慢性炎症中的用途
CN114907333B (zh) * 2022-05-11 2023-07-04 中国人民解放军军事科学院军事医学研究院 环丙甲酰胺衍生物及其制备方法和用途
WO2025024550A1 (en) * 2023-07-25 2025-01-30 University Of Florida Research Foundation, Incorporated Rev-erb antagonists

Family Cites Families (19)

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Publication number Priority date Publication date Assignee Title
US4472193A (en) * 1982-07-06 1984-09-18 The Dow Chemical Company Naphthyridinyloxy(or thio)phenoxy propanoic acids, derivatives thereof and methods of herbicidal use
ES2200617B1 (es) * 2001-01-19 2005-05-01 Almirall Prodesfarma, S.A. Derivados de urea como antagonistas de integrinas alfa 4.
WO2008057209A1 (en) * 2006-10-27 2008-05-15 Merck & Co., Inc. Hcv ns3 protease inhibitors
US8258301B2 (en) * 2007-05-15 2012-09-04 Boehringer Ingelheim International Gmbh Urotensin II receptor antagonists
UY31984A (es) * 2008-07-16 2010-02-26 Boehringer Ingelheim Int DERIVADOS DE 1-(3,4-difluorobencil)-6-oxo-1,6-dihidropirimidin-5-carboxamidas N-sustituidas y de 2-(3,4-difluorobencil)-3-oxo-2,3-dihidro-1H-pirazol-4-carboxamidas N-sustituidas.
TW201026667A (en) * 2008-09-30 2010-07-16 Merz Pharma Gmbh & Co Kgaa Glycine b antagonists
US9593108B2 (en) * 2009-04-06 2017-03-14 Ptc Therapeutics, Inc. Compounds and methods for antiviral treatment
AU2011253058A1 (en) * 2010-05-13 2012-12-06 Amgen Inc. Heteroaryloxycarbocyclyl compounds as PDE10 inhibitors
WO2013033310A1 (en) * 2011-08-31 2013-03-07 Theodore Mark Kamenecka Modulators of rev-erb
WO2013045519A1 (en) * 2011-09-27 2013-04-04 Genfit Derivatives of 6-substituted triazolopyridazines as rev-erb agonists
AU2013216354B2 (en) * 2012-02-02 2017-08-31 Idorsia Pharmaceuticals Ltd 4-(benzoimidazol-2-yl)-thiazole compounds and related aza derivatives
TW201348231A (zh) * 2012-02-29 2013-12-01 Amgen Inc 雜雙環化合物
JP6374384B2 (ja) * 2012-08-07 2018-08-15 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung プロテインキナーゼ阻害剤としてのピリドピリミジン誘導体
CA2894126A1 (en) * 2012-12-21 2014-06-26 Epizyme, Inc. Prmt5 inhibitors and uses thereof
WO2015103527A1 (en) * 2014-01-06 2015-07-09 The Scripps Research Institute Modulators of rev-erb
SG11201705192PA (en) * 2014-12-24 2017-07-28 Gilead Sciences Inc Fused pyrimidine compounds for the treatment of hiv
WO2017222951A1 (en) * 2016-06-23 2017-12-28 Merck Sharp & Dohme Corp. 3-aryl and heteroaryl substituted 5-trifluoromethyl oxadiazoles as histone deacetylase 6 (hdac6) inhibitors
CN109776335B (zh) * 2017-11-15 2022-03-18 武汉尚赛光电科技有限公司 芘的胺类衍生物及其制备方法、应用和器件
GB201810486D0 (en) * 2018-06-26 2018-08-08 Imperial Innovations Ltd Natural killer cells

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