JP2023551203A5 - - Google Patents

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Publication number
JP2023551203A5
JP2023551203A5 JP2023530743A JP2023530743A JP2023551203A5 JP 2023551203 A5 JP2023551203 A5 JP 2023551203A5 JP 2023530743 A JP2023530743 A JP 2023530743A JP 2023530743 A JP2023530743 A JP 2023530743A JP 2023551203 A5 JP2023551203 A5 JP 2023551203A5
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JP
Japan
Prior art keywords
substituted
alkyl
aryl
conjugate
cycloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023530743A
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English (en)
Japanese (ja)
Other versions
JP2023551203A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/060193 external-priority patent/WO2022109335A1/en
Publication of JP2023551203A publication Critical patent/JP2023551203A/ja
Publication of JP2023551203A5 publication Critical patent/JP2023551203A5/ja
Pending legal-status Critical Current

Links

JP2023530743A 2020-11-20 2021-11-19 抗体-薬物コンジュゲートのためのグリコシド二重切断リンカー Pending JP2023551203A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202063116632P 2020-11-20 2020-11-20
US63/116,632 2020-11-20
US202163139685P 2021-01-20 2021-01-20
US63/139,685 2021-01-20
PCT/US2021/060193 WO2022109335A1 (en) 2020-11-20 2021-11-19 Glycoside dual-cleavage linkers for antibody-drug conjugates

Publications (2)

Publication Number Publication Date
JP2023551203A JP2023551203A (ja) 2023-12-07
JP2023551203A5 true JP2023551203A5 (https=) 2024-11-26

Family

ID=81708155

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023530743A Pending JP2023551203A (ja) 2020-11-20 2021-11-19 抗体-薬物コンジュゲートのためのグリコシド二重切断リンカー

Country Status (8)

Country Link
US (2) US12187810B2 (https=)
EP (1) EP4247829A1 (https=)
JP (1) JP2023551203A (https=)
KR (1) KR20230122008A (https=)
AU (1) AU2021382033A1 (https=)
CA (1) CA3201005A1 (https=)
MX (1) MX2023005979A (https=)
WO (1) WO2022109335A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202440164A (zh) 2022-12-13 2024-10-16 美商克林提克斯醫藥股份有限公司 生長抑素亞型-2受體(sst2r)靶向治療劑及其用途

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