JP2023546352A5 - - Google Patents

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Publication number
JP2023546352A5
JP2023546352A5 JP2023521087A JP2023521087A JP2023546352A5 JP 2023546352 A5 JP2023546352 A5 JP 2023546352A5 JP 2023521087 A JP2023521087 A JP 2023521087A JP 2023521087 A JP2023521087 A JP 2023521087A JP 2023546352 A5 JP2023546352 A5 JP 2023546352A5
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Japan
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alkylene
alkyl
leukemia
pharmaceutically acceptable
independently
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JP2023521087A
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Japanese (ja)
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JP2023546352A (ja
JP7588224B2 (ja
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Priority claimed from PCT/US2021/071695 external-priority patent/WO2022076975A1/en
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Priority to JP2024128215A priority Critical patent/JP2024153884A/ja
Publication of JP2023546352A5 publication Critical patent/JP2023546352A5/ja
Priority to JP2024198167A priority patent/JP2025020388A/ja
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Publication of JP7588224B2 publication Critical patent/JP7588224B2/ja
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JP2023521087A 2020-10-05 2021-10-04 Bcr-ablチロシンキナーゼの阻害のための5-及び6-アザインドール化合物 Active JP7588224B2 (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2024128215A JP2024153884A (ja) 2020-10-05 2024-08-02 Bcr-ablチロシンキナーゼの阻害のための5-及び6-アザインドール化合物
JP2024198167A JP2025020388A (ja) 2020-10-05 2024-11-13 Bcr-ablチロシンキナーゼの阻害のための5-及び6-アザインドール化合物

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202063087763P 2020-10-05 2020-10-05
US63/087,763 2020-10-05
US202163224236P 2021-07-21 2021-07-21
US63/224,236 2021-07-21
PCT/US2021/071695 WO2022076975A1 (en) 2020-10-05 2021-10-04 5- and 6-azaindole compounds for inhibition of bcr-abl tyrosine kinases

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Publications (3)

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JP2023546352A JP2023546352A (ja) 2023-11-02
JP2023546352A5 true JP2023546352A5 (enExample) 2024-08-14
JP7588224B2 JP7588224B2 (ja) 2024-11-21

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JP2023521087A Active JP7588224B2 (ja) 2020-10-05 2021-10-04 Bcr-ablチロシンキナーゼの阻害のための5-及び6-アザインドール化合物
JP2024128215A Withdrawn JP2024153884A (ja) 2020-10-05 2024-08-02 Bcr-ablチロシンキナーゼの阻害のための5-及び6-アザインドール化合物
JP2024198167A Withdrawn JP2025020388A (ja) 2020-10-05 2024-11-13 Bcr-ablチロシンキナーゼの阻害のための5-及び6-アザインドール化合物

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JP2024128215A Withdrawn JP2024153884A (ja) 2020-10-05 2024-08-02 Bcr-ablチロシンキナーゼの阻害のための5-及び6-アザインドール化合物
JP2024198167A Withdrawn JP2025020388A (ja) 2020-10-05 2024-11-13 Bcr-ablチロシンキナーゼの阻害のための5-及び6-アザインドール化合物

Country Status (10)

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US (4) US11767321B2 (enExample)
EP (1) EP4225742A4 (enExample)
JP (3) JP7588224B2 (enExample)
KR (1) KR20230104781A (enExample)
CN (1) CN119019388B (enExample)
AU (1) AU2021358123A1 (enExample)
CA (1) CA3196620A1 (enExample)
IL (1) IL301739A (enExample)
MX (1) MX2023003995A (enExample)
WO (1) WO2022076975A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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WO2026084950A1 (en) 2024-10-16 2026-04-23 Enliven Inc. 5- and 6-azaindole compounds for inhibition of bcr-abl tyrosine kinases for use in the treatment of cancer

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