JP2023535409A5 - - Google Patents

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Publication number
JP2023535409A5
JP2023535409A5 JP2023504258A JP2023504258A JP2023535409A5 JP 2023535409 A5 JP2023535409 A5 JP 2023535409A5 JP 2023504258 A JP2023504258 A JP 2023504258A JP 2023504258 A JP2023504258 A JP 2023504258A JP 2023535409 A5 JP2023535409 A5 JP 2023535409A5
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JP
Japan
Prior art keywords
formula
conjugate according
brm
alkyl
following
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023504258A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023535409A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/042280 external-priority patent/WO2022020288A1/en
Publication of JP2023535409A publication Critical patent/JP2023535409A/ja
Publication of JP2023535409A5 publication Critical patent/JP2023535409A5/ja
Pending legal-status Critical Current

Links

JP2023504258A 2020-07-21 2021-07-20 Brm分解の抗体コンジュゲート化化学的誘導物質及びbrm分解の方法 Pending JP2023535409A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063054757P 2020-07-21 2020-07-21
US63/054,757 2020-07-21
PCT/US2021/042280 WO2022020288A1 (en) 2020-07-21 2021-07-20 Antibody-conjugated chemical inducers of degradation of brm and methods thereof

Publications (2)

Publication Number Publication Date
JP2023535409A JP2023535409A (ja) 2023-08-17
JP2023535409A5 true JP2023535409A5 (enExample) 2024-07-25

Family

ID=77265314

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023504258A Pending JP2023535409A (ja) 2020-07-21 2021-07-20 Brm分解の抗体コンジュゲート化化学的誘導物質及びbrm分解の方法

Country Status (18)

Country Link
US (1) US20230330249A1 (enExample)
EP (1) EP4185328A1 (enExample)
JP (1) JP2023535409A (enExample)
KR (1) KR20230042032A (enExample)
CN (1) CN116249556A (enExample)
AR (1) AR123019A1 (enExample)
AU (1) AU2021312225A1 (enExample)
BR (1) BR112023001143A2 (enExample)
CA (1) CA3188649A1 (enExample)
CL (2) CL2023000193A1 (enExample)
CO (1) CO2023000679A2 (enExample)
CR (1) CR20230017A (enExample)
IL (1) IL299860A (enExample)
MX (1) MX2023000888A (enExample)
PE (1) PE20231104A1 (enExample)
PH (1) PH12023550129A1 (enExample)
TW (1) TW202216215A (enExample)
WO (1) WO2022020288A1 (enExample)

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US12606568B2 (en) 2020-12-09 2026-04-21 Kymera Therapeutics, Inc. SMARCA degraders and uses thereof
JP2024533990A (ja) * 2021-08-09 2024-09-18 ジェネンテック, インコーポレイテッド Brmの調節に使用するためのフェノール誘導体
AR128331A1 (es) * 2022-01-26 2024-04-17 Genentech Inc Inductores químicos de degradación conjugados con anticuerpos y métodos de estos
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