JP2023529001A5 - - Google Patents

Info

Publication number
JP2023529001A5
JP2023529001A5 JP2022576335A JP2022576335A JP2023529001A5 JP 2023529001 A5 JP2023529001 A5 JP 2023529001A5 JP 2022576335 A JP2022576335 A JP 2022576335A JP 2022576335 A JP2022576335 A JP 2022576335A JP 2023529001 A5 JP2023529001 A5 JP 2023529001A5
Authority
JP
Japan
Prior art keywords
solid oral
oral composition
rabeximod
composition according
dosage form
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022576335A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023529001A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2021/065705 external-priority patent/WO2021250204A1/en
Publication of JP2023529001A publication Critical patent/JP2023529001A/ja
Publication of JP2023529001A5 publication Critical patent/JP2023529001A5/ja
Pending legal-status Critical Current

Links

JP2022576335A 2020-06-10 2021-06-10 結晶形のラベキシモドを含む経口製剤 Pending JP2023529001A (ja)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
EP20179279.3 2020-06-10
EP20179279 2020-06-10
EP20179277.7 2020-06-10
EP20179239 2020-06-10
EP20179277 2020-06-10
EP20179239.7 2020-06-10
EP20180706 2020-06-18
EP20180706.2 2020-06-18
PCT/EP2021/065705 WO2021250204A1 (en) 2020-06-10 2021-06-10 Oral formulation comprising a crystalline form of rabeximod

Publications (2)

Publication Number Publication Date
JP2023529001A JP2023529001A (ja) 2023-07-06
JP2023529001A5 true JP2023529001A5 (https=) 2024-06-18

Family

ID=76305939

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2022576335A Pending JP2023529001A (ja) 2020-06-10 2021-06-10 結晶形のラベキシモドを含む経口製剤
JP2022575226A Pending JP2023529877A (ja) 2020-06-10 2021-06-10 結晶形のラベキシモドの調製方法
JP2022575829A Pending JP2023533662A (ja) 2020-06-10 2021-06-10 関節リウマチの治療におけるラベキシモド

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2022575226A Pending JP2023529877A (ja) 2020-06-10 2021-06-10 結晶形のラベキシモドの調製方法
JP2022575829A Pending JP2023533662A (ja) 2020-06-10 2021-06-10 関節リウマチの治療におけるラベキシモド

Country Status (8)

Country Link
US (3) US12594274B2 (https=)
EP (3) EP4164650A1 (https=)
JP (3) JP2023529001A (https=)
KR (3) KR20230022880A (https=)
CN (4) CN115768431A (https=)
AU (3) AU2021290174A1 (https=)
CA (3) CA3181629A1 (https=)
WO (3) WO2021250197A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20230022880A (ko) 2020-06-10 2023-02-16 사익손 아베 라벡시모드의 결정성 형태를 포함하는 경구 제형
US11643415B1 (en) 2021-12-09 2023-05-09 Cyxone Ab Rabeximod compounds

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE8600260D0 (sv) 1986-01-21 1986-01-21 Lundblad Leif Substituerade indolokinoxaliner
SE504289C2 (sv) * 1994-06-23 1996-12-23 Leif J I Lundblad Användning av vissa indolo-2,3b-kinoxaliner för framställning av ett läkemedel för inhibering av enzymet HIV-integras
JPH08165278A (ja) 1994-12-14 1996-06-25 Kawaken Fine Chem Co Ltd 1−置換トリプタミン化合物の製造方法
SE504862C2 (sv) 1994-12-27 1997-05-20 Leif J I Lundblad Användning av vissa indolo-§2,3b¤-kinoxaliner för framställning av ett läkemedel för skydd av DNA i initieringsfasen och/eller promotionsfasen av karcinogenes och för förhindrande av oxidativ stress i patienter med sjukdomar relaterade till fria radikaler
DE19516804A1 (de) * 1995-05-08 1996-11-14 Hoechst Ag Isoindolinpigmente auf Basis von Aminochinoxalindionen
US6333327B2 (en) 2000-02-18 2001-12-25 Leif J. I. Lundblad Method for the treatment of Multiple Sclerosis
SE516067C2 (sv) 2000-02-18 2001-11-12 Lundblad Leif J I Användning av en förening för framställning av ett läkemedel
TW200410921A (en) * 2002-11-25 2004-07-01 Hoffmann La Roche Mandelic acid derivatives
ATE382623T1 (de) * 2004-06-09 2008-01-15 Hoffmann La Roche Octahydropyrrolo(3,4-c)pyrrolderivate und deren verwendung als antivirale mitteln
SE527639C2 (sv) 2004-06-17 2006-05-02 Oxypharma Ab Alkylsubstituerade indolokinoxaliner
WO2008066151A1 (fr) * 2006-11-30 2008-06-05 Tokyo Institute Of Technology Nouveau dérivé curcumine
CN102115457B (zh) 2011-03-05 2012-11-21 太原理工大学 一种n-乙基咔唑的制备方法
US20150079111A1 (en) * 2012-06-05 2015-03-19 Jonas Axelsson Mechanism, diagnostic, and treatments for complications of renal failure
EA201500942A1 (ru) 2013-03-15 2016-03-31 Виронова Херпес Аб ПРОТИВОВИРУСНЫЙ ИНДОЛО[2,3-b]ХИНОКСАЛИН
AU2016272089B2 (en) 2015-06-03 2021-02-18 Triastek, Inc. Dosage forms and use thereof
CN105061432B (zh) * 2015-07-16 2017-09-29 河北大学 6H‑吲哚[2,3‑b]喹喔啉衍生物、药物组合物及其制备和应用
TWI842978B (zh) * 2018-07-13 2024-05-21 美商基利科學股份有限公司 衍生物
KR20230022880A (ko) 2020-06-10 2023-02-16 사익손 아베 라벡시모드의 결정성 형태를 포함하는 경구 제형
EP4164649A1 (en) 2020-06-10 2023-04-19 Cyxone AB New use of rabeximod
US11643415B1 (en) * 2021-12-09 2023-05-09 Cyxone Ab Rabeximod compounds

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