JP2023521116A5 - - Google Patents
Info
- Publication number
- JP2023521116A5 JP2023521116A5 JP2022561396A JP2022561396A JP2023521116A5 JP 2023521116 A5 JP2023521116 A5 JP 2023521116A5 JP 2022561396 A JP2022561396 A JP 2022561396A JP 2022561396 A JP2022561396 A JP 2022561396A JP 2023521116 A5 JP2023521116 A5 JP 2023521116A5
- Authority
- JP
- Japan
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202063008183P | 2020-04-10 | 2020-04-10 | |
| US63/008,183 | 2020-04-10 | ||
| US202063027495P | 2020-05-20 | 2020-05-20 | |
| US63/027,495 | 2020-05-20 | ||
| PCT/US2021/022656 WO2021206876A1 (en) | 2020-04-10 | 2021-03-17 | Inhibitors of norovirus and coronavirus replication |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2023521116A JP2023521116A (ja) | 2023-05-23 |
| JPWO2021206876A5 JPWO2021206876A5 (https=) | 2024-03-26 |
| JP2023521116A5 true JP2023521116A5 (https=) | 2024-03-26 |
| JP7721561B2 JP7721561B2 (ja) | 2025-08-12 |
Family
ID=75439538
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022561396A Active JP7721561B2 (ja) | 2020-04-10 | 2021-03-17 | ノロウイルス及びコロナウイルス複製の阻害剤 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20230159453A1 (https=) |
| EP (1) | EP4132944A1 (https=) |
| JP (1) | JP7721561B2 (https=) |
| KR (1) | KR20230008079A (https=) |
| CN (1) | CN115698035A (https=) |
| AU (1) | AU2021254045A1 (https=) |
| BR (1) | BR112022019557A2 (https=) |
| CA (1) | CA3179697A1 (https=) |
| IL (1) | IL297069A (https=) |
| MX (1) | MX2022012714A (https=) |
| PH (1) | PH12022552486A1 (https=) |
| TW (1) | TW202204318A (https=) |
| WO (1) | WO2021206876A1 (https=) |
Families Citing this family (29)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4126816A4 (en) * | 2020-03-30 | 2024-07-31 | Kansas State University Research Foundation | BROAD-SPECTRUM ANTIVIRALS AGAINST CORONAVIRUS |
| US11124497B1 (en) | 2020-04-17 | 2021-09-21 | Pardes Biosciences, Inc. | Inhibitors of cysteine proteases and methods of use thereof |
| US11174231B1 (en) | 2020-06-09 | 2021-11-16 | Pardes Biosciences, Inc. | Inhibitors of cysteine proteases and methods of use thereof |
| GB2607514B (en) | 2020-07-20 | 2023-06-21 | Enanta Pharm Inc | Functionalized peptides as antiviral agents |
| US11351149B2 (en) * | 2020-09-03 | 2022-06-07 | Pfizer Inc. | Nitrile-containing antiviral compounds |
| US11352363B1 (en) | 2020-11-23 | 2022-06-07 | Enanta Pharmaceuticals, Inc. | Spiropyrrolidine derived antiviral agents |
| US11384090B2 (en) | 2020-11-23 | 2022-07-12 | Enanta Pharmaceuticals, Inc. | Spiropyrrolidine derived antiviral agents |
| US12540141B2 (en) | 2020-11-23 | 2026-02-03 | Enanta Pharmaceuticals, Inc. | Spiropyrrolidine derived antiviral agents |
| KR20230124583A (ko) | 2020-11-23 | 2023-08-25 | 이난타 파마슈티칼스, 인코포레이티드 | 신규한 스피로피롤리딘 유래 항바이러스제 |
| CN116685573B (zh) * | 2021-01-19 | 2025-12-12 | 中国人民解放军军事科学院军事医学研究院 | 含有n-(取代磺酰基)乙酰胺结构的病毒蛋白酶抑制剂，及其在抗病毒药物中的应用 |
| WO2022165220A1 (en) * | 2021-01-29 | 2022-08-04 | Kansas State University Research Foundation | Conformationally-constrained inhibitors of 3c or 3c-like proteases |
| WO2022235605A1 (en) | 2021-05-04 | 2022-11-10 | Enanta Pharmaceuticals, Inc. | Novel macrocyclic antiviral agents |
| US12398147B2 (en) | 2021-05-11 | 2025-08-26 | Enanta Pharmaceuticals, Inc. | Macrocyclic spiropyrrolidine derived antiviral agents |
| US11319325B1 (en) | 2021-05-11 | 2022-05-03 | Enanta Pharmaceuticals, Inc. | Macrocyclic spiropyrrolidine derived antiviral agents |
| JP2024522990A (ja) * | 2021-06-02 | 2024-06-25 | エイシア セラピューティクス， インコーポレイテッド | 抗ウイルス薬としてのプロテアーゼ阻害剤 |
| WO2022266363A1 (en) * | 2021-06-16 | 2022-12-22 | The Scripps Research Institute | Protease inhibitors for the treatment of coronavirus infections |
| US11325916B1 (en) | 2021-07-29 | 2022-05-10 | Enanta Pharmaceuticals, Inc. | Spiropyrrolidine derived antiviral agents |
| US11339170B1 (en) | 2021-07-23 | 2022-05-24 | Enanta Pharmaceuticals, Inc. | Spiropyrrolidine derived antiviral agents |
| US12479854B2 (en) | 2021-07-29 | 2025-11-25 | Enanta Pharmaceuticals, Inc. | Spiropyrrolidine derived antiviral agents |
| JP2024530920A (ja) * | 2021-08-03 | 2024-08-27 | コクリスタル ファーマ，インコーポレイテッド | コロナウイルスに対する阻害剤 |
| WO2023086352A1 (en) | 2021-11-12 | 2023-05-19 | Enanta Pharmaceuticals, Inc. | Novel spiropyrrolidine derived antiviral agents |
| WO2023086350A1 (en) | 2021-11-12 | 2023-05-19 | Enanta Pharmaceuticals, Inc. | Alkyne-containing antiviral agents |
| US11919910B2 (en) | 2021-11-12 | 2024-03-05 | Enanta Pharmaceuticals, Inc. | Spiropyrrolidine derived antiviral agents |
| US11993600B2 (en) | 2021-12-08 | 2024-05-28 | Enanta Pharmaceuticals, Inc. | Saturated spirocyclics as antiviral agents |
| US12145941B2 (en) | 2021-12-08 | 2024-11-19 | Enanta Pharmaceuticals, Inc. | Heterocyclic antiviral agents |
| EP4460508A4 (en) * | 2022-01-07 | 2025-12-24 | Merck Sharp & Dohme Llc | PROTEASE INHIBITORS TO TREAT OR PREVENT CORONAVIRUS INFECTION |
| EP4488264A4 (en) * | 2022-03-01 | 2026-03-04 | Westvac Biopharma Co Ltd | CETO AMIDE DERIVATIVES AND THEIR PHARMACEUTICAL USE |
| WO2023196307A1 (en) | 2022-04-05 | 2023-10-12 | Enanta Pharmaceuticals, Inc. | Novel spiropyrrolidine derived antiviral agents |
| CN115260074B (zh) * | 2022-08-02 | 2024-06-21 | 爱斯特（成都）生物制药股份有限公司 | 一种口服抗病毒药物Paxlovid中间体的制备方法 |
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| CN106928206B (zh) * | 2015-12-31 | 2022-02-18 | 中国科学院上海药物研究所 | 醛基类化合物及其制法和用途 |
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| CN110105348A (zh) * | 2019-03-08 | 2019-08-09 | 南开大学 | 新型迈克尔受体类肠病毒71型抑制剂的制备及用途 |
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2021
- 2021-03-17 CN CN202180027505.5A patent/CN115698035A/zh active Pending
- 2021-03-17 TW TW110109546A patent/TW202204318A/zh unknown
- 2021-03-17 US US17/912,749 patent/US20230159453A1/en active Pending
- 2021-03-17 BR BR112022019557A patent/BR112022019557A2/pt unknown
- 2021-03-17 PH PH1/2022/552486A patent/PH12022552486A1/en unknown
- 2021-03-17 MX MX2022012714A patent/MX2022012714A/es unknown
- 2021-03-17 JP JP2022561396A patent/JP7721561B2/ja active Active
- 2021-03-17 KR KR1020227039096A patent/KR20230008079A/ko active Pending
- 2021-03-17 WO PCT/US2021/022656 patent/WO2021206876A1/en not_active Ceased
- 2021-03-17 CA CA3179697A patent/CA3179697A1/en active Pending
- 2021-03-17 AU AU2021254045A patent/AU2021254045A1/en active Pending
- 2021-03-17 EP EP21717692.4A patent/EP4132944A1/en active Pending
- 2021-03-17 IL IL297069A patent/IL297069A/en unknown