JP2023513373A5 - - Google Patents

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Publication number
JP2023513373A5
JP2023513373A5 JP2022548875A JP2022548875A JP2023513373A5 JP 2023513373 A5 JP2023513373 A5 JP 2023513373A5 JP 2022548875 A JP2022548875 A JP 2022548875A JP 2022548875 A JP2022548875 A JP 2022548875A JP 2023513373 A5 JP2023513373 A5 JP 2023513373A5
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JP
Japan
Application number
JP2022548875A
Other languages
Japanese (ja)
Other versions
JPWO2021161105A5 (https=
JP2023513373A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2021/000091 external-priority patent/WO2021161105A1/en
Publication of JP2023513373A publication Critical patent/JP2023513373A/ja
Publication of JPWO2021161105A5 publication Critical patent/JPWO2021161105A5/ja
Publication of JP2023513373A5 publication Critical patent/JP2023513373A5/ja
Ceased legal-status Critical Current

Links

JP2022548875A 2020-02-14 2021-02-12 P2x3修飾薬 Ceased JP2023513373A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062977008P 2020-02-14 2020-02-14
US62/977,008 2020-02-14
PCT/IB2021/000091 WO2021161105A1 (en) 2020-02-14 2021-02-12 P2x3 modulators

Publications (3)

Publication Number Publication Date
JP2023513373A JP2023513373A (ja) 2023-03-30
JPWO2021161105A5 JPWO2021161105A5 (https=) 2024-02-20
JP2023513373A5 true JP2023513373A5 (https=) 2024-02-20

Family

ID=77292083

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022548875A Ceased JP2023513373A (ja) 2020-02-14 2021-02-12 P2x3修飾薬

Country Status (11)

Country Link
US (1) US20230312557A1 (https=)
EP (1) EP4103564A4 (https=)
JP (1) JP2023513373A (https=)
KR (1) KR20220141331A (https=)
CN (2) CN119039290A (https=)
AU (1) AU2021219097A1 (https=)
BR (1) BR112022015858A2 (https=)
CA (1) CA3170664A1 (https=)
IL (1) IL295393A (https=)
MX (1) MX2022009762A (https=)
WO (1) WO2021161105A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2020228760A1 (en) 2019-02-25 2021-09-23 Glaxosmithkline Intellectual Property (No. 3) Limited Treatment with P2X3 modulators
EP4103572A4 (en) * 2020-02-14 2024-03-06 Bellus Health Cough Inc. MAKING A P2X3 ANTAGONIST
WO2021244634A1 (zh) * 2020-06-05 2021-12-09 武汉人福创新药物研发中心有限公司 咪唑并吡啶类化合物及其用途
CN114805237B (zh) * 2021-01-22 2026-04-21 武汉人福创新药物研发中心有限公司 杂环类化合物的制备方法及其中间体
CN114805340A (zh) * 2021-01-22 2022-07-29 武汉人福创新药物研发中心有限公司 咪唑并吡啶类化合物的制备方法及其中间体
CN116635389A (zh) * 2021-01-29 2023-08-22 上海海雁医药科技有限公司 吗啉衍生物及其药物组合物和用途
CN115043836B (zh) * 2021-08-20 2023-07-18 苏州璞正医药有限公司 一种咪唑并吡啶衍生物的p2x3受体选择性调节剂及其药物用途

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112012011518B8 (pt) * 2009-11-18 2023-01-10 Astrazeneca Ab Compostos, composição farmacêutica, kit e usos de um composto
US9598409B2 (en) * 2013-01-31 2017-03-21 Neomed Institute Imidazopyridine compounds and uses thereof
US9907795B2 (en) * 2016-01-08 2018-03-06 Nerre Therapeutics Limited Method of treatment of chronic cough administering orvepitant in combination with other therapeutic agents
US10111883B1 (en) * 2017-09-18 2018-10-30 Bellus Health Cough Inc. Selective P2X3 modulators
CA3115939A1 (en) * 2018-10-10 2020-04-16 Bellus Health Cough Inc. Treatment of pruritus with p2x3 antagonists
WO2020135771A1 (zh) * 2018-12-29 2020-07-02 武汉朗来科技发展有限公司 杂环类化合物、中间体、其制备方法及应用
AU2020228760A1 (en) * 2019-02-25 2021-09-23 Glaxosmithkline Intellectual Property (No. 3) Limited Treatment with P2X3 modulators
CN112409331B (zh) * 2019-08-21 2024-02-20 上海翰森生物医药科技有限公司 杂环类衍生物抑制剂、其制备方法和应用

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