JP2024518447A5 - - Google Patents
Info
- Publication number
- JP2024518447A5 JP2024518447A5 JP2023568613A JP2023568613A JP2024518447A5 JP 2024518447 A5 JP2024518447 A5 JP 2024518447A5 JP 2023568613 A JP2023568613 A JP 2023568613A JP 2023568613 A JP2023568613 A JP 2023568613A JP 2024518447 A5 JP2024518447 A5 JP 2024518447A5
- Authority
- JP
- Japan
- Prior art keywords
- hydrogen
- alkyl
- haloalkyl
- halogen
- stereoisomers
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB2106486.0 | 2021-05-06 | ||
| GB202106486 | 2021-05-06 | ||
| PCT/GB2022/051167 WO2022234299A1 (en) | 2021-05-06 | 2022-05-06 | Pkc-theta modulators |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024518447A JP2024518447A (ja) | 2024-05-01 |
| JP2024518447A5 true JP2024518447A5 (https=) | 2025-11-18 |
Family
ID=82100804
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023568613A Pending JP2024518447A (ja) | 2021-05-06 | 2022-05-06 | PKC-θモジュレーター |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20240239794A1 (https=) |
| EP (1) | EP4334316A1 (https=) |
| JP (1) | JP2024518447A (https=) |
| KR (1) | KR20240024063A (https=) |
| CN (1) | CN117295738A (https=) |
| AU (1) | AU2022269348A1 (https=) |
| BR (1) | BR112023022883A2 (https=) |
| CA (1) | CA3214088A1 (https=) |
| CL (1) | CL2023003247A1 (https=) |
| CO (1) | CO2023015005A2 (https=) |
| IL (1) | IL307669A (https=) |
| MX (1) | MX2023013012A (https=) |
| PE (1) | PE20250019A1 (https=) |
| WO (1) | WO2022234299A1 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2022234298A1 (en) * | 2021-05-06 | 2022-11-10 | Exscientia Ai Limited | Pkc-theta modulators |
| CN118772140B (zh) * | 2023-04-07 | 2026-04-17 | 四川大学 | 一类化合物及其在治疗hDHODH介导的疾病中的用途 |
| WO2025255294A1 (en) * | 2024-06-06 | 2025-12-11 | Bristol-Myers Squibb Company | Pkc-theta inhibitors, compositions, and methods of use |
| WO2025255298A1 (en) * | 2024-06-06 | 2025-12-11 | Bristol-Myers Squibb Company | Pkc-theta inhibitors, compositions, and methods of use |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200924762A (en) * | 2007-11-02 | 2009-06-16 | Vertex Pharma | Kinase inhibitors |
| GB0920382D0 (en) | 2009-11-20 | 2010-01-06 | Univ Dundee | Design of molecules |
| CN102471342A (zh) * | 2010-05-05 | 2012-05-23 | 沃泰克斯药物股份有限公司 | 用作PKC-θ抑制剂的4取代的吡唑并吡啶类 |
| US9556126B2 (en) | 2013-12-20 | 2017-01-31 | Signal Pharmaceuticals, Llc | Substituted diaminopyrimidyl compounds, compositions thereof, and methods of treatment therewith |
| AU2020284742B2 (en) * | 2019-05-28 | 2026-03-05 | Mankind Pharma Ltd. | Novel compounds for inhibition of Janus Kinase 1 |
| WO2022234298A1 (en) * | 2021-05-06 | 2022-11-10 | Exscientia Ai Limited | Pkc-theta modulators |
-
2022
- 2022-05-06 PE PE2023002994A patent/PE20250019A1/es unknown
- 2022-05-06 AU AU2022269348A patent/AU2022269348A1/en active Pending
- 2022-05-06 IL IL307669A patent/IL307669A/en unknown
- 2022-05-06 JP JP2023568613A patent/JP2024518447A/ja active Pending
- 2022-05-06 CA CA3214088A patent/CA3214088A1/en active Pending
- 2022-05-06 BR BR112023022883A patent/BR112023022883A2/pt unknown
- 2022-05-06 US US18/557,865 patent/US20240239794A1/en active Pending
- 2022-05-06 WO PCT/GB2022/051167 patent/WO2022234299A1/en not_active Ceased
- 2022-05-06 CN CN202280033111.5A patent/CN117295738A/zh active Pending
- 2022-05-06 MX MX2023013012A patent/MX2023013012A/es unknown
- 2022-05-06 EP EP22731282.4A patent/EP4334316A1/en active Pending
- 2022-05-06 KR KR1020237041626A patent/KR20240024063A/ko active Pending
-
2023
- 2023-11-02 CL CL2023003247A patent/CL2023003247A1/es unknown
- 2023-11-03 CO CONC2023/0015005A patent/CO2023015005A2/es unknown
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