JP2022552445A5 - - Google Patents
Info
- Publication number
- JP2022552445A5 JP2022552445A5 JP2022546591A JP2022546591A JP2022552445A5 JP 2022552445 A5 JP2022552445 A5 JP 2022552445A5 JP 2022546591 A JP2022546591 A JP 2022546591A JP 2022546591 A JP2022546591 A JP 2022546591A JP 2022552445 A5 JP2022552445 A5 JP 2022552445A5
- Authority
- JP
- Japan
- Prior art keywords
- optionally substituted
- alkyl
- group
- pharmaceutically acceptable
- occurrence
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962911653P | 2019-10-07 | 2019-10-07 | |
| US62/911,653 | 2019-10-07 | ||
| PCT/US2020/054373 WO2021071821A1 (en) | 2019-10-07 | 2020-10-06 | Arylmethylene aromatic compounds as kv1.3 potassium shaker channel blockers |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022552445A JP2022552445A (ja) | 2022-12-15 |
| JP2022552445A5 true JP2022552445A5 (enExample) | 2024-09-06 |
| JP7697954B2 JP7697954B2 (ja) | 2025-06-24 |
Family
ID=75438313
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022546591A Active JP7697954B2 (ja) | 2019-10-07 | 2020-10-06 | Ｋｖ１．３カリウムシェーカーチャネル遮断薬としてのアリールメチレン芳香族化合物 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20230131535A1 (enExample) |
| EP (1) | EP4041230A4 (enExample) |
| JP (1) | JP7697954B2 (enExample) |
| KR (1) | KR20220079879A (enExample) |
| CN (1) | CN114727992A (enExample) |
| AU (1) | AU2020363366A1 (enExample) |
| BR (1) | BR112022006242A2 (enExample) |
| CA (1) | CA3157026A1 (enExample) |
| IL (1) | IL291733A (enExample) |
| MX (1) | MX2022004168A (enExample) |
| WO (1) | WO2021071821A1 (enExample) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA3193554A1 (en) | 2020-10-06 | 2022-04-14 | D.E. Shaw Research, Llc | Lactam compounds as kv1.3 potassium shaker channel blockers |
| EP4253383A4 (en) * | 2020-12-31 | 2024-07-17 | Tsinghua University | PYRIDINE-2-AMINE DERIVATIVE, PHARMACEUTICAL COMPOSITION AND ASSOCIATED USE |
| WO2022198196A1 (en) | 2021-03-15 | 2022-09-22 | Maze Therapeutics, Inc. | Inhibitors of glycogen synthase 1 (gys1) and methods of use thereof |
| CN115703734B (zh) * | 2021-08-05 | 2024-08-09 | 重庆文理学院 | 二芳基甲基吡啶类化合物及其制备方法和应用 |
| TW202345806A (zh) | 2022-03-31 | 2023-12-01 | 美商艾伯維有限公司 | 噻唑并〔５，４－ｂ〕吡啶ｍａｌｔ－１抑制劑 |
| WO2024104815A1 (en) | 2022-11-16 | 2024-05-23 | Basf Se | Substituted benzodiazepines as fungicides |
| CN120202194A (zh) | 2022-11-16 | 2025-06-24 | 巴斯夫欧洲公司 | 作为杀真菌剂的取代的四氢苯并二氮杂䓬 |
| CN120957986A (zh) | 2023-03-17 | 2025-11-14 | 巴斯夫欧洲公司 | 用于对抗植物病原性真菌的取代的吡啶基/吡嗪基二氢苯并硫氮杂䓬化合物 |
| TW202521512A (zh) | 2023-07-31 | 2025-06-01 | 美商美國禮來大藥廠 | Kv1.3鉀shaker通道阻斷劑之固體形式及其使用方法 |
| WO2026057374A1 (en) | 2024-09-11 | 2026-03-19 | Basf Se | Fungicidal mixture comprising substituted pyridyl/pyrazidyl dihydrobenzothiazepine compounds |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH540009A (de) * | 1970-07-23 | 1973-09-28 | Ciba Geigy Ag | Verwendung von Monohydroxyphenylcarbinolen zum antimikrobiellen Ausrüsten bzw. zum Schützen von textilen Materialien gegen schädliche Mikroorganismen |
| JPH07309837A (ja) * | 1993-04-28 | 1995-11-28 | Takeda Chem Ind Ltd | ピリジン誘導体、その製造法および剤 |
| JPH09278757A (ja) * | 1996-04-15 | 1997-10-28 | Takeda Chem Ind Ltd | ヒドラゾン誘導体および剤 |
| TW467902B (en) | 1996-07-31 | 2001-12-11 | Bristol Myers Squibb Co | Diphenyl heterocycles as potassium channel modulators |
| AU736712B2 (en) | 1998-01-29 | 2001-08-02 | Bristol-Myers Squibb Company | Benzoate derivatives of diaryl 1,3,4-oxadiazolone |
| KR20070092297A (ko) * | 2004-12-21 | 2007-09-12 | 데브젠 엔브이 | Ｋｖ4 이온 채널 활성을 갖는 화합물 |
| NZ584480A (en) * | 2007-10-04 | 2011-08-26 | Bionomics Ltd | Novel aryl potassium channel blockers and uses thereof |
| GB0815784D0 (en) | 2008-08-29 | 2008-10-08 | Xention Ltd | Novel potassium channel blockers |
| GB0909672D0 (en) | 2009-06-04 | 2009-07-22 | Xention Discovery Ltd | Compounds |
| KR20130100300A (ko) * | 2010-08-27 | 2013-09-10 | 그뤼넨탈 게엠베하 | Ｋｃｎｑ２／３ 조절제로서의 치환된 ２-옥시-퀴놀린-３-카복스아미드 |
| BR112015022504A2 (pt) * | 2013-03-13 | 2017-07-18 | A Reichard Gregory | compostos de triazina e composições dos mesmos e métodos para tratar malária e quimioprofilaxia |
| RS61719B1 (sr) * | 2015-08-27 | 2021-05-31 | Pfizer | Biciklična fuzionisana hetaroaril ili aril jedinjenja kao modulatori irak4 |
| EP3490581A4 (en) * | 2016-07-26 | 2020-10-14 | Flagship Pioneering Innovations V, Inc. | NEUROMODULATORY COMPOSITIONS AND ASSOCIATED CANCER TREATMENT METHODS |
-
2020
- 2020-10-06 BR BR112022006242A patent/BR112022006242A2/pt not_active IP Right Cessation
- 2020-10-06 AU AU2020363366A patent/AU2020363366A1/en not_active Abandoned
- 2020-10-06 WO PCT/US2020/054373 patent/WO2021071821A1/en not_active Ceased
- 2020-10-06 EP EP20875222.0A patent/EP4041230A4/en active Pending
- 2020-10-06 CN CN202080084417.4A patent/CN114727992A/zh active Pending
- 2020-10-06 US US17/766,879 patent/US20230131535A1/en active Pending
- 2020-10-06 KR KR1020227013504A patent/KR20220079879A/ko not_active Withdrawn
- 2020-10-06 JP JP2022546591A patent/JP7697954B2/ja active Active
- 2020-10-06 MX MX2022004168A patent/MX2022004168A/es unknown
- 2020-10-06 CA CA3157026A patent/CA3157026A1/en active Pending
-
2022
- 2022-03-27 IL IL291733A patent/IL291733A/en unknown
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