JP2022521413A5 - - Google Patents

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Publication number
JP2022521413A5
JP2022521413A5 JP2021549463A JP2021549463A JP2022521413A5 JP 2022521413 A5 JP2022521413 A5 JP 2022521413A5 JP 2021549463 A JP2021549463 A JP 2021549463A JP 2021549463 A JP2021549463 A JP 2021549463A JP 2022521413 A5 JP2022521413 A5 JP 2022521413A5
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compound
item
ray powder
powder diffractogram
crystalline form
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JP2021549463A
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English (en)
Japanese (ja)
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JP2022521413A (ja
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Priority claimed from PCT/US2020/019071 external-priority patent/WO2020172431A1/en
Publication of JP2022521413A publication Critical patent/JP2022521413A/ja
Publication of JP2022521413A5 publication Critical patent/JP2022521413A5/ja
Pending legal-status Critical Current

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JP2021549463A 2019-02-22 2020-02-20 Syk阻害剤としての縮合ピラジンの固体形態 Pending JP2022521413A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962809337P 2019-02-22 2019-02-22
US62/809,337 2019-02-22
PCT/US2020/019071 WO2020172431A1 (en) 2019-02-22 2020-02-20 Solid forms of condensed pyrazines as syk inhibitors

Publications (2)

Publication Number Publication Date
JP2022521413A JP2022521413A (ja) 2022-04-07
JP2022521413A5 true JP2022521413A5 (enExample) 2023-02-28

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ID=69845599

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Application Number Title Priority Date Filing Date
JP2021549463A Pending JP2022521413A (ja) 2019-02-22 2020-02-20 Syk阻害剤としての縮合ピラジンの固体形態

Country Status (11)

Country Link
US (3) US11339168B2 (enExample)
EP (1) EP3927708A1 (enExample)
JP (1) JP2022521413A (enExample)
KR (1) KR20210131372A (enExample)
CN (1) CN113950479A (enExample)
AU (1) AU2020225455A1 (enExample)
CA (1) CA3130848A1 (enExample)
MX (1) MX2021010131A (enExample)
TW (1) TW202045510A (enExample)
WO (1) WO2020172431A1 (enExample)
ZA (1) ZA202106014B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI735853B (zh) 2013-12-23 2021-08-11 美商克洛諾斯生技有限公司 脾酪胺酸激酶抑制劑
US20240285621A1 (en) 2020-09-23 2024-08-29 Nerviano Medical Sciences S.R.L. Pyrazolyl-pyrimidine derivatives as kinase inhibitors
CN112939983A (zh) * 2021-02-01 2021-06-11 暨明医药科技(苏州)有限公司 一种SYK激酶抑制剂Lanraplenib的合成方法
EP4646412A1 (en) * 2022-12-09 2025-11-12 Kronos Bio, Inc. Crystalline forms of lanraplenib and methods of making and using the same

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