JP2022517189A5 - - Google Patents

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Publication number
JP2022517189A5
JP2022517189A5 JP2021539020A JP2021539020A JP2022517189A5 JP 2022517189 A5 JP2022517189 A5 JP 2022517189A5 JP 2021539020 A JP2021539020 A JP 2021539020A JP 2021539020 A JP2021539020 A JP 2021539020A JP 2022517189 A5 JP2022517189 A5 JP 2022517189A5
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JP
Japan
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JP2021539020A
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JP7539892B2 (ja
JPWO2020142612A5 (https=
JP2022517189A (ja
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JP2021539020A 2019-01-03 2020-01-02 癌疾患の処置のためのエンドリボヌクレアーゼのイノシトール要求酵素i(ireiアルファ)の阻害剤としてのピリド-ピリミジノン化合物及びプテリジノン化合物 Active JP7539892B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
CNPCT/CN2019/070275 2019-01-03
CN2019070275 2019-01-03
CNPCT/CN2019/081673 2019-04-08
CN2019081673 2019-04-08
PCT/US2020/012058 WO2020142612A1 (en) 2019-01-03 2020-01-02 Pyrido-pyrimidinone and pteridinone compounds as inhibitors of endoribonuclease inositol requiring enzyme i (ire i alpha) for the treatment of cancer diseases.

Publications (4)

Publication Number Publication Date
JP2022517189A JP2022517189A (ja) 2022-03-07
JP2022517189A5 true JP2022517189A5 (https=) 2023-01-04
JPWO2020142612A5 JPWO2020142612A5 (https=) 2023-01-04
JP7539892B2 JP7539892B2 (ja) 2024-08-26

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JP2021539020A Active JP7539892B2 (ja) 2019-01-03 2020-01-02 癌疾患の処置のためのエンドリボヌクレアーゼのイノシトール要求酵素i(ireiアルファ)の阻害剤としてのピリド-ピリミジノン化合物及びプテリジノン化合物

Country Status (6)

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US (1) US12344603B2 (https=)
EP (1) EP3941919B1 (https=)
JP (1) JP7539892B2 (https=)
CN (1) CN113508115A (https=)
TW (1) TWI748317B (https=)
WO (1) WO2020142612A1 (https=)

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