JP2021533087A5 - - Google Patents
Info
- Publication number
- JP2021533087A5 JP2021533087A5 JP2020571842A JP2020571842A JP2021533087A5 JP 2021533087 A5 JP2021533087 A5 JP 2021533087A5 JP 2020571842 A JP2020571842 A JP 2020571842A JP 2020571842 A JP2020571842 A JP 2020571842A JP 2021533087 A5 JP2021533087 A5 JP 2021533087A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- substituted
- unsubstituted
- alkyl
- cyano
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024096077A JP2024133496A (ja) | 2018-06-26 | 2024-06-13 | 神経炎症におけるマクロファージコロニー刺激因子１受容体（ｃｓｆ１ｒ）をイメージングするための陽電子放射断層撮影（ｐｅｔ）放射性トレーサー |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862689958P | 2018-06-26 | 2018-06-26 | |
| US62/689,958 | 2018-06-26 | ||
| PCT/US2019/039234 WO2020006075A1 (en) | 2018-06-26 | 2019-06-26 | Positron emission tomography (pet) radiotracers for imaging macrophage colony-stimulating factor 1 receptor (csf1r) in neuroinflammation |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024096077A Division JP2024133496A (ja) | 2018-06-26 | 2024-06-13 | 神経炎症におけるマクロファージコロニー刺激因子１受容体（ｃｓｆ１ｒ）をイメージングするための陽電子放射断層撮影（ｐｅｔ）放射性トレーサー |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021533087A JP2021533087A (ja) | 2021-12-02 |
| JP2021533087A5 true JP2021533087A5 (enExample) | 2022-07-25 |
| JP7884818B2 JP7884818B2 (ja) | 2026-07-06 |
Family
ID=68985080
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020571842A Active JP7884818B2 (ja) | 2018-06-26 | 2019-06-26 | 神経炎症におけるマクロファージコロニー刺激因子１受容体（ｃｓｆ１ｒ）をイメージングするための陽電子放射断層撮影（ｐｅｔ）放射性トレーサー |
| JP2024096077A Pending JP2024133496A (ja) | 2018-06-26 | 2024-06-13 | 神経炎症におけるマクロファージコロニー刺激因子１受容体（ｃｓｆ１ｒ）をイメージングするための陽電子放射断層撮影（ｐｅｔ）放射性トレーサー |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024096077A Pending JP2024133496A (ja) | 2018-06-26 | 2024-06-13 | 神経炎症におけるマクロファージコロニー刺激因子１受容体（ｃｓｆ１ｒ）をイメージングするための陽電子放射断層撮影（ｐｅｔ）放射性トレーサー |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20210290784A1 (enExample) |
| EP (1) | EP3813890A4 (enExample) |
| JP (2) | JP7884818B2 (enExample) |
| KR (1) | KR20210013769A (enExample) |
| CN (2) | CN112638431A (enExample) |
| AU (1) | AU2019294699B2 (enExample) |
| BR (1) | BR112020026602A2 (enExample) |
| CA (1) | CA3104520A1 (enExample) |
| EA (1) | EA202092843A1 (enExample) |
| IL (1) | IL279768B2 (enExample) |
| MX (1) | MX2021000141A (enExample) |
| WO (1) | WO2020006075A1 (enExample) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MA54550A (fr) | 2018-12-20 | 2022-03-30 | Amgen Inc | Inhibiteurs de kif18a |
| AU2019401495B2 (en) * | 2018-12-20 | 2025-06-26 | Amgen Inc. | Heteroaryl amides useful as KIF18A inhibitors |
| AU2019404576B2 (en) | 2018-12-20 | 2025-07-17 | Amgen Inc. | Heteroaryl amides useful as KIF18A inhibitors |
| AU2020325115B2 (en) | 2019-08-02 | 2026-03-12 | Amgen Inc. | Pyridine derivatives as KIF18A inhibitors |
| JP7699100B2 (ja) | 2019-08-02 | 2025-06-26 | アムジエン・インコーポレーテツド | Ｋｉｆ１８ａ阻害剤 |
| EP4269404A4 (en) * | 2020-12-25 | 2024-12-04 | Xizang Haisco Pharmaceutical Co., Ltd. | KETOHEXOKINASE INHIBITORS AND USE THEREOF |
| US20240237960A1 (en) * | 2021-06-11 | 2024-07-18 | Jubilant Draximage Inc. | Expert scoring system for measurement of severity, treatment response and prognosis of peripheral arterial disease |
| US20250275730A1 (en) * | 2022-04-06 | 2025-09-04 | University Of Virginia Patent Foundation | Automation of the blood input function computation pipeline for dynamic fdg pet for human brain using machine learning |
| AU2024214768A1 (en) * | 2023-01-30 | 2025-08-07 | The Johns Hopkins University | 18 f-labeled pet radiotracers for imaging macrophage colony stimulating factor 1 receptor |
| CN118021811A (zh) * | 2023-12-28 | 2024-05-14 | 复旦大学附属华山医院 | 一种靶向于csf1r激酶的6-氟吡啶甲酰苯胺类抑制剂、药物组合物及其核素成像试剂 |
| CN118027009B (zh) * | 2024-04-15 | 2024-07-12 | 北京师范大学 | 一类靶向于csf1r激酶的苯基酰胺类化合物及其应用 |
| CN119498255B (zh) * | 2024-10-24 | 2025-11-25 | 香港理工大学深圳研究院 | 一种抑郁症小鼠模型及其构建方法与应用 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101084208A (zh) * | 2004-10-22 | 2007-12-05 | 詹森药业有限公司 | 作为c－fms激酶抑制剂的芳族酰胺 |
| AU2017258415B2 (en) * | 2016-04-29 | 2023-03-30 | Cornell University | Compositions and methods for targeted particle penetration, distribution, and response in malignant brain tumors |
-
2019
- 2019-06-26 WO PCT/US2019/039234 patent/WO2020006075A1/en not_active Ceased
- 2019-06-26 CA CA3104520A patent/CA3104520A1/en active Pending
- 2019-06-26 IL IL279768A patent/IL279768B2/en unknown
- 2019-06-26 CN CN201980056945.6A patent/CN112638431A/zh active Pending
- 2019-06-26 BR BR112020026602-7A patent/BR112020026602A2/pt unknown
- 2019-06-26 KR KR1020217002632A patent/KR20210013769A/ko not_active Ceased
- 2019-06-26 AU AU2019294699A patent/AU2019294699B2/en active Active
- 2019-06-26 EP EP19825817.0A patent/EP3813890A4/en active Pending
- 2019-06-26 EA EA202092843A patent/EA202092843A1/ru unknown
- 2019-06-26 JP JP2020571842A patent/JP7884818B2/ja active Active
- 2019-06-26 US US17/253,336 patent/US20210290784A1/en active Pending
- 2019-06-26 MX MX2021000141A patent/MX2021000141A/es unknown
- 2019-06-26 CN CN202410732670.6A patent/CN118743770A/zh active Pending
-
2024
- 2024-06-13 JP JP2024096077A patent/JP2024133496A/ja active Pending
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