JP2021522327A5 - - Google Patents

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Publication number
JP2021522327A5
JP2021522327A5 JP2021506388A JP2021506388A JP2021522327A5 JP 2021522327 A5 JP2021522327 A5 JP 2021522327A5 JP 2021506388 A JP2021506388 A JP 2021506388A JP 2021506388 A JP2021506388 A JP 2021506388A JP 2021522327 A5 JP2021522327 A5 JP 2021522327A5
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JP
Japan
Prior art keywords
alkyl
alkynyl
alkenyl
cycloalkyl
amino
Prior art date
Application number
JP2021506388A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021522327A (ja
JPWO2019204813A5 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/028544 external-priority patent/WO2019204813A1/en
Publication of JP2021522327A publication Critical patent/JP2021522327A/ja
Publication of JP2021522327A5 publication Critical patent/JP2021522327A5/ja
Publication of JPWO2019204813A5 publication Critical patent/JPWO2019204813A5/ja
Pending legal-status Critical Current

Links

JP2021506388A 2018-04-20 2019-04-22 ミトコンドリア脱共役剤として有用なオキサジアゾロピラジンおよびオキサジアゾロピリジン Pending JP2021522327A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862660880P 2018-04-20 2018-04-20
US62/660,880 2018-04-20
PCT/US2019/028544 WO2019204813A1 (en) 2018-04-20 2019-04-22 Oxadiazolopyrazines and oxadiazolopyridines useful as mitochondrial uncouplers

Publications (3)

Publication Number Publication Date
JP2021522327A JP2021522327A (ja) 2021-08-30
JP2021522327A5 true JP2021522327A5 (https=) 2022-05-02
JPWO2019204813A5 JPWO2019204813A5 (https=) 2022-05-02

Family

ID=67139787

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2021506388A Pending JP2021522327A (ja) 2018-04-20 2019-04-22 ミトコンドリア脱共役剤として有用なオキサジアゾロピラジンおよびオキサジアゾロピリジン
JP2021506390A Pending JP2021523933A (ja) 2018-04-20 2019-04-22 ミトコンドリア脱共役剤として有用なイミダゾピリジン
JP2021506391A Pending JP2021523934A (ja) 2018-04-20 2019-04-22 ミトコンドリア脱共役剤として有用なアミノピラジンおよび関連化合物

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2021506390A Pending JP2021523933A (ja) 2018-04-20 2019-04-22 ミトコンドリア脱共役剤として有用なイミダゾピリジン
JP2021506391A Pending JP2021523934A (ja) 2018-04-20 2019-04-22 ミトコンドリア脱共役剤として有用なアミノピラジンおよび関連化合物

Country Status (12)

Country Link
US (3) US20210253594A1 (https=)
EP (3) EP3781572A1 (https=)
JP (3) JP2021522327A (https=)
KR (3) KR20210003831A (https=)
CN (3) CN112262141A (https=)
AU (2) AU2019256722A1 (https=)
BR (2) BR112020021466A2 (https=)
CA (2) CA3097751A1 (https=)
IL (2) IL278070A (https=)
MX (2) MX2020011050A (https=)
WO (3) WO2019204813A1 (https=)
ZA (2) ZA202006295B (https=)

Families Citing this family (5)

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CN112262141A (zh) * 2018-04-20 2021-01-22 弗吉尼亚理工大学知识产权有限公司 可用作线粒体解偶联剂的咪唑吡啶
WO2020191503A1 (en) * 2019-03-27 2020-10-01 Algernon Pharmaceuticals Inc. Methods and uses of bromantane and derivatives thereof for treating lung disease, fatty liver disease, and kidney disorders
CA3189027A1 (en) 2020-07-11 2022-01-20 Pfizer Inc. Antiviral heteroaryl ketone derivatives
US11351149B2 (en) 2020-09-03 2022-06-07 Pfizer Inc. Nitrile-containing antiviral compounds
EP4482494A4 (en) * 2022-02-21 2026-02-25 Univ Colorado Regents RE-SENSITIZATION OF MULTI-DRUG-RESISTANT GRAM-NEGATIVE (MDR) BACTERIA TO COLISTIN USING IONOPHORES

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CN112262141A (zh) * 2018-04-20 2021-01-22 弗吉尼亚理工大学知识产权有限公司 可用作线粒体解偶联剂的咪唑吡啶

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