JP2021512913A5 - - Google Patents
Info
- Publication number
- JP2021512913A5 JP2021512913A5 JP2020542775A JP2020542775A JP2021512913A5 JP 2021512913 A5 JP2021512913 A5 JP 2021512913A5 JP 2020542775 A JP2020542775 A JP 2020542775A JP 2020542775 A JP2020542775 A JP 2020542775A JP 2021512913 A5 JP2021512913 A5 JP 2021512913A5
- Authority
- JP
- Japan
- Prior art keywords
- pharmaceutically acceptable
- alkoxybenzo
- membered heterocyclic
- heterocyclic amine
- amine compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN201810124854.9 | 2018-02-07 | ||
| CN201810124854.9A CN110117278B (zh) | 2018-02-07 | 2018-02-07 | 烷氧基苯并五元(六元)杂环胺类化合物及其药物用途 |
| PCT/CN2019/072468 WO2019154047A1 (zh) | 2018-02-07 | 2019-01-21 | 烷氧基苯并五元(六元)杂环胺类化合物及其药物用途 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021512913A JP2021512913A (ja) | 2021-05-20 |
| JP2021512913A5 true JP2021512913A5 (https=) | 2023-01-10 |
| JP7475049B2 JP7475049B2 (ja) | 2024-04-26 |
Family
ID=67519628
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020542775A Active JP7475049B2 (ja) | 2018-02-07 | 2019-01-21 | アルコキシベンゾ五員（六員）複素環式アミン化合物およびその医薬用途 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US11396504B2 (https=) |
| EP (1) | EP3750890B1 (https=) |
| JP (1) | JP7475049B2 (https=) |
| CN (1) | CN110117278B (https=) |
| WO (1) | WO2019154047A1 (https=) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2764243C2 (ru) | 2017-09-22 | 2022-01-14 | ДЖУБИЛАНТ ЭПИПЭД ЭлЭлСи | Гетероциклические соединения в качестве ингибиторов PAD |
| AU2018352142B2 (en) | 2017-10-18 | 2022-08-25 | Jubilant Epipad LLC | Imidazo-pyridine compounds as PAD inhibitors |
| US11629135B2 (en) | 2017-11-06 | 2023-04-18 | Jubilant Prodell Llc | Pyrimidine derivatives as inhibitors of PD1/PD-L1 activation |
| PT3704120T (pt) | 2017-11-24 | 2024-07-03 | Jubilant Episcribe Llc | Compostos heterocíclicos como inibidores de prmt5 |
| CN110117278B (zh) | 2018-02-07 | 2022-07-19 | 石家庄以岭药业股份有限公司 | 烷氧基苯并五元(六元)杂环胺类化合物及其药物用途 |
| MX2020009517A (es) | 2018-03-13 | 2021-01-20 | Jubilant Prodel LLC | Compuestos biciclicos como inhibidores de la interaccion/activacio n de pdl/pd-l1. |
| CN111481548A (zh) * | 2019-01-29 | 2020-08-04 | 复旦大学 | 4-(2,6-二氯苄氧基)-3-(3-氨基吡啶)苯并[d]异噁唑在制药中的用途 |
| CN113616652A (zh) * | 2020-05-06 | 2021-11-09 | 石家庄以岭药业股份有限公司 | Sms2抑制剂在制备治疗高侵袭性乳腺癌药物中的应用 |
| CN116854670A (zh) * | 2022-03-28 | 2023-10-10 | 中国科学院上海药物研究所 | 一类二氢喹喔啉类选择性溴结构域识别蛋白抑制剂及其制备方法和用途 |
| CN119320385A (zh) * | 2023-07-17 | 2025-01-17 | 复旦大学 | 烷氧基噻吩甲酰芳胺类化合物及其应用 |
Family Cites Families (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3755332A (en) * | 1971-07-01 | 1973-08-28 | Ciba Geigy Corp | Substituted 4 indazolaminoquinolines |
| HUP9802492A3 (en) * | 1995-06-06 | 1999-10-28 | Hoechst Marion Roussel Inc Cin | Benzisoxazole and indazole derivatives as antipsychotic agents, process for their preparation and pharmaceutical compositions containing the same |
| US5668154A (en) * | 1995-06-06 | 1997-09-16 | Hoechst Marion Roussel Inc. | Pyridiniminyl-1,2-benzisoxazoles and -benzisothiazoles |
| GB9914486D0 (en) * | 1999-06-21 | 1999-08-18 | Smithkline Beecham Plc | Medicaments |
| FR2836915B1 (fr) * | 2002-03-11 | 2008-01-11 | Aventis Pharma Sa | Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant |
| RU2006134022A (ru) * | 2004-02-27 | 2008-04-10 | Ф.Хоффманн-Ля Рош Аг (Ch) | Производные индазола и содержащие их фармацевтические композиции |
| EP1647549A1 (en) * | 2004-10-14 | 2006-04-19 | Laboratoire Theramex | Indazoles, benzisoxazoles and benzisothiazoles as estrogenic agents |
| JP5314244B2 (ja) * | 2004-10-27 | 2013-10-16 | 富山化学工業株式会社 | 新規な含窒素複素環化合物およびその塩 |
| EP1856099A2 (en) * | 2005-03-03 | 2007-11-21 | Sirtris Pharmaceuticals, Inc. | Acridine and quinoline derivatives as sirtuin modulators |
| WO2006094235A1 (en) * | 2005-03-03 | 2006-09-08 | Sirtris Pharmaceuticals, Inc. | Fused heterocyclic compounds and their use as sirtuin modulators |
| DE102005026194A1 (de) * | 2005-06-06 | 2006-12-07 | Grünenthal GmbH | Substituierte N-Benzo[d]isoxazol-3-yl-amin-Derivate und deren Verwendung zur Herstellung von Arzneimitteln |
| CN101213187B (zh) * | 2005-06-28 | 2012-06-06 | 塞诺菲-安万特股份有限公司 | 作为rho-激酶抑制剂的异喹啉衍生物 |
| JP2009520825A (ja) * | 2005-12-20 | 2009-05-28 | 武田薬品工業株式会社 | グルコキナーゼ活性剤 |
| WO2008089310A2 (en) * | 2007-01-18 | 2008-07-24 | Lexicon Pharmaceuticals, Inc. | Delta 5 desaturase inhibitors for the treatment of obesity |
| US20080194557A1 (en) * | 2007-01-18 | 2008-08-14 | Joseph Barbosa | Methods and compositions for the treatment of pain, inflammation and cancer |
| ATE549325T1 (de) * | 2007-01-26 | 2012-03-15 | Basf Se | 3-amino-1,2-benzisothiazol-verbindungen zur bekämpfung von tierpest ii |
| MX2009008531A (es) * | 2007-02-16 | 2009-08-26 | Amgen Inc | Cetonas de heterociclilo que contienen nitrogeno y su uso como inhibidores de c-met. |
| WO2008156757A1 (en) * | 2007-06-19 | 2008-12-24 | Takeda Pharmaceutical Company Limited | Indazole compounds for activating glucokinase |
| JP2010111624A (ja) * | 2008-11-06 | 2010-05-20 | Shionogi & Co Ltd | Ｔｔｋ阻害作用を有するインダゾール誘導体 |
| CN101993382B (zh) * | 2009-08-21 | 2014-10-29 | 复旦大学 | 芳香胺类衍生物或其类似物及其应用 |
| CN105348182B (zh) * | 2014-08-24 | 2018-04-13 | 复旦大学 | 2‑烷氧基苯甲酰芳胺类化合物及其药物用途 |
| JP6661192B2 (ja) | 2016-01-19 | 2020-03-11 | 国立大学法人北海道大学 | Ｓｍｓ２阻害活性を有するセラミド誘導体 |
| CN110117278B (zh) | 2018-02-07 | 2022-07-19 | 石家庄以岭药业股份有限公司 | 烷氧基苯并五元(六元)杂环胺类化合物及其药物用途 |
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2018
- 2018-02-07 CN CN201810124854.9A patent/CN110117278B/zh active Active
-
2019
- 2019-01-21 WO PCT/CN2019/072468 patent/WO2019154047A1/zh not_active Ceased
- 2019-01-21 EP EP19751009.2A patent/EP3750890B1/en active Active
- 2019-01-21 US US16/967,118 patent/US11396504B2/en active Active
- 2019-01-21 JP JP2020542775A patent/JP7475049B2/ja active Active