JP2021511360A5 - - Google Patents
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- Publication number
- JP2021511360A5 JP2021511360A5 JP2020540751A JP2020540751A JP2021511360A5 JP 2021511360 A5 JP2021511360 A5 JP 2021511360A5 JP 2020540751 A JP2020540751 A JP 2020540751A JP 2020540751 A JP2020540751 A JP 2020540751A JP 2021511360 A5 JP2021511360 A5 JP 2021511360A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- optionally substituted
- alkylene
- cycloalkyl
- heterocycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2023083168A JP7690517B2 (ja) | 2018-01-26 | 2023-05-19 | キナーゼ依存的障害を処置するための化合物 |
| JP2025089864A JP2025128208A (ja) | 2018-01-26 | 2025-05-29 | キナーゼ依存的障害を処置するための化合物 |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862622702P | 2018-01-26 | 2018-01-26 | |
| US62/622,702 | 2018-01-26 | ||
| US201862758321P | 2018-11-09 | 2018-11-09 | |
| US62/758,321 | 2018-11-09 | ||
| PCT/US2019/015297 WO2019148044A1 (en) | 2018-01-26 | 2019-01-25 | Compounds for the treatment of kinase-dependent disorders |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023083168A Division JP7690517B2 (ja) | 2018-01-26 | 2023-05-19 | キナーゼ依存的障害を処置するための化合物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021511360A JP2021511360A (ja) | 2021-05-06 |
| JP2021511360A5 true JP2021511360A5 (https=) | 2022-02-01 |
| JP7321165B2 JP7321165B2 (ja) | 2023-08-04 |
Family
ID=65409544
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020540751A Active JP7321165B2 (ja) | 2018-01-26 | 2019-01-25 | キナーゼ依存的障害を処置するための化合物 |
| JP2023083168A Active JP7690517B2 (ja) | 2018-01-26 | 2023-05-19 | キナーゼ依存的障害を処置するための化合物 |
| JP2025089864A Pending JP2025128208A (ja) | 2018-01-26 | 2025-05-29 | キナーゼ依存的障害を処置するための化合物 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023083168A Active JP7690517B2 (ja) | 2018-01-26 | 2023-05-19 | キナーゼ依存的障害を処置するための化合物 |
| JP2025089864A Pending JP2025128208A (ja) | 2018-01-26 | 2025-05-29 | キナーゼ依存的障害を処置するための化合物 |
Country Status (34)
| Country | Link |
|---|---|
| US (2) | US11542259B2 (https=) |
| EP (2) | EP3743070B1 (https=) |
| JP (3) | JP7321165B2 (https=) |
| KR (2) | KR102721118B1 (https=) |
| CN (5) | CN117402114A (https=) |
| AU (2) | AU2019212801B2 (https=) |
| BR (1) | BR112020015201A2 (https=) |
| CA (1) | CA3088200A1 (https=) |
| CL (2) | CL2020001931A1 (https=) |
| CO (1) | CO2020010465A2 (https=) |
| CR (2) | CR20230287A (https=) |
| DK (1) | DK3743070T3 (https=) |
| ES (1) | ES3048989T3 (https=) |
| FI (1) | FI3743070T3 (https=) |
| GE (2) | GEP20257770B (https=) |
| HR (1) | HRP20251184T1 (https=) |
| HU (1) | HUE073371T2 (https=) |
| IL (3) | IL321138A (https=) |
| LT (1) | LT3743070T (https=) |
| MA (1) | MA51673B1 (https=) |
| MD (1) | MD3743070T2 (https=) |
| MX (2) | MX2020007765A (https=) |
| MY (1) | MY210421A (https=) |
| PE (2) | PE20242219A1 (https=) |
| PH (1) | PH12020551208A1 (https=) |
| PL (1) | PL3743070T3 (https=) |
| PT (1) | PT3743070T (https=) |
| RS (1) | RS67317B1 (https=) |
| SA (1) | SA520412500B1 (https=) |
| SG (1) | SG11202006921PA (https=) |
| SI (1) | SI3743070T1 (https=) |
| SM (1) | SMT202500395T1 (https=) |
| UA (1) | UA128476C2 (https=) |
| WO (1) | WO2019148044A1 (https=) |
Families Citing this family (24)
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| KR20210108367A (ko) | 2018-11-09 | 2021-09-02 | 비바체 테라퓨틱스, 인크. | 비시클릭 화합물 |
| KR102828472B1 (ko) | 2018-12-13 | 2025-07-03 | 엑셀리시스, 인코포레이티드 | 키나아제 억제제의 결정질 형태 및 염 형태 |
| BR112021014504A2 (pt) * | 2019-01-25 | 2021-09-28 | Exelixis, Inc. | Compostos para o tratamento de transtornos dependentes de cinase |
| CN109761899B (zh) * | 2019-02-14 | 2022-11-15 | 广州六顺生物科技股份有限公司 | 喹啉衍生物、其药学上可接受的盐或其溶剂合物、其应用、药物及药物组合物 |
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| CN110845406B (zh) * | 2019-12-04 | 2021-07-20 | 广州安岩仁医药科技有限公司 | 喹啉类化合物的制备方法 |
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| CN115461328B (zh) * | 2020-04-30 | 2025-11-07 | 埃克塞里艾克西斯公司 | 用于制备激酶抑制剂的方法 |
| IL300151A (en) * | 2020-07-31 | 2023-03-01 | Exelixis Inc | Combinations for cancer treatment |
| JP2023548855A (ja) * | 2020-11-05 | 2023-11-21 | エグゼリクシス, インコーポレイテッド | キナーゼ阻害剤の医薬組成物 |
| TW202334090A (zh) * | 2021-11-03 | 2023-09-01 | 美商艾克塞里克斯公司 | 用於治療激酶依賴性病症之化合物 |
| US20250368606A1 (en) * | 2021-12-22 | 2025-12-04 | Exelixis, Inc. | Crystalline forms and salt forms of a kinase inhibitor |
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2019
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2022
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2023
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