JP2022119852A5 - - Google Patents
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- JP2022119852A5 JP2022119852A5 JP2022081736A JP2022081736A JP2022119852A5 JP 2022119852 A5 JP2022119852 A5 JP 2022119852A5 JP 2022081736 A JP2022081736 A JP 2022081736A JP 2022081736 A JP2022081736 A JP 2022081736A JP 2022119852 A5 JP2022119852 A5 JP 2022119852A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- pharmaceutically acceptable
- tautomer
- stereoisomer
- geometric isomer
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN201611204309.8A CN108239074B (zh) | 2016-12-26 | 2016-12-26 | 喹唑啉类化合物及其制备方法、用途和药物组合物 |
| CN201611214102.9 | 2016-12-26 | ||
| CN201611211589.5A CN108239075B (zh) | 2016-12-26 | 2016-12-26 | 喹唑啉类化合物及其制备方法、用途和药物组合物 |
| CN201611204309.8 | 2016-12-26 | ||
| CN201611211589.5 | 2016-12-26 | ||
| CN201611214102.9A CN108239076B (zh) | 2016-12-26 | 2016-12-26 | 喹唑啉类化合物及其制备方法、用途和药物组合物 |
| JP2019534817A JP7077323B2 (ja) | 2016-12-26 | 2017-12-26 | キナゾリン化合物並びにその調製方法、使用及び医薬組成物 |
| PCT/CN2017/118771 WO2018121550A1 (zh) | 2016-12-26 | 2017-12-26 | 喹唑啉类化合物及其制备方法、用途和药物组合物 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019534817A Division JP7077323B2 (ja) | 2016-12-26 | 2017-12-26 | キナゾリン化合物並びにその調製方法、使用及び医薬組成物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022119852A JP2022119852A (ja) | 2022-08-17 |
| JP2022119852A5 true JP2022119852A5 (https=) | 2022-11-09 |
| JP7384535B2 JP7384535B2 (ja) | 2023-11-21 |
Family
ID=62707834
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019534817A Active JP7077323B2 (ja) | 2016-12-26 | 2017-12-26 | キナゾリン化合物並びにその調製方法、使用及び医薬組成物 |
| JP2022081738A Active JP7384536B2 (ja) | 2016-12-26 | 2022-05-18 | キナゾリン化合物並びにその調製方法、使用及び医薬組成物 |
| JP2022081736A Active JP7384535B2 (ja) | 2016-12-26 | 2022-05-18 | キナゾリン化合物並びにその調製方法、使用及び医薬組成物 |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019534817A Active JP7077323B2 (ja) | 2016-12-26 | 2017-12-26 | キナゾリン化合物並びにその調製方法、使用及び医薬組成物 |
| JP2022081738A Active JP7384536B2 (ja) | 2016-12-26 | 2022-05-18 | キナゾリン化合物並びにその調製方法、使用及び医薬組成物 |
Country Status (7)
| Country | Link |
|---|---|
| US (3) | US11534443B2 (https=) |
| EP (3) | EP4169917B1 (https=) |
| JP (3) | JP7077323B2 (https=) |
| CN (1) | CN110382490A (https=) |
| AU (3) | AU2017389818B2 (https=) |
| CA (3) | CA3174865A1 (https=) |
| WO (1) | WO2018121550A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11534443B2 (en) * | 2016-12-26 | 2022-12-27 | Institute Of Materia Medica, Chinese Academy Of Medical Sciences | Quinazoline compounds, preparation method, use, and pharmaceutical composition thereof |
| WO2021088787A1 (zh) * | 2019-11-07 | 2021-05-14 | 南京正大天晴制药有限公司 | 作为axl抑制剂的喹唑啉类化合物 |
| CN113620976B (zh) * | 2020-05-09 | 2023-09-26 | 中国医学科学院药物研究所 | 噻唑并嘧啶类化合物及其制备方法、用途和药物组合物 |
| MX2023005747A (es) | 2020-11-18 | 2023-07-28 | Deciphera Pharmaceuticals Llc | Inhibidores de gcn2 y perk quinasas y metodos de uso de los mismos. |
| KR20240113496A (ko) | 2021-12-03 | 2024-07-22 | 데시페라 파마슈티칼스, 엘엘씨. | Gcn2 및 perk 키나아제 억제제로서의 헤테로고리 화합물 |
| CN119630431A (zh) * | 2022-08-26 | 2025-03-14 | 卫材R&D管理有限公司 | 抗体药物缀合物 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR960008781B1 (ko) * | 1993-08-05 | 1996-07-03 | 김하운 | 연소효율 증강장치 |
| ES2788383T3 (es) | 2000-04-25 | 2020-10-21 | Icos Corp | Inhibidores de delta fosfatidilo-inositol 3-quinasa humana |
| PE20090288A1 (es) | 2007-05-10 | 2009-04-03 | Smithkline Beecham Corp | Derivados de quinoxalina como inhibidores de la pi3 quinasa |
| PE20090717A1 (es) | 2007-05-18 | 2009-07-18 | Smithkline Beecham Corp | Derivados de quinolina como inhibidores de la pi3 quinasa |
| UY31137A1 (es) | 2007-06-14 | 2009-01-05 | Smithkline Beecham Corp | Derivados de quinazolina como inhibidores de la pi3 quinasa |
| US20100311736A1 (en) | 2007-10-22 | 2010-12-09 | Glaxosmithkline Llc | Pyridosulfonamide derivatives as p13 kinase inhibitors |
| EP2984088B1 (en) * | 2013-04-12 | 2019-03-20 | Asana BioSciences, LLC | Quinazolines and azaquinazolines as dual inhibitors of ras/raf/mek/erk and pi3k/akt/pten/mtor pathways |
| US11534443B2 (en) * | 2016-12-26 | 2022-12-27 | Institute Of Materia Medica, Chinese Academy Of Medical Sciences | Quinazoline compounds, preparation method, use, and pharmaceutical composition thereof |
| CN108239074B (zh) | 2016-12-26 | 2021-07-06 | 中国医学科学院药物研究所 | 喹唑啉类化合物及其制备方法、用途和药物组合物 |
| CN108239075B (zh) | 2016-12-26 | 2021-07-02 | 中国医学科学院药物研究所 | 喹唑啉类化合物及其制备方法、用途和药物组合物 |
| CN108239076B (zh) | 2016-12-26 | 2021-07-06 | 中国医学科学院药物研究所 | 喹唑啉类化合物及其制备方法、用途和药物组合物 |
-
2017
- 2017-12-26 US US16/473,901 patent/US11534443B2/en active Active
- 2017-12-26 CA CA3174865A patent/CA3174865A1/en active Pending
- 2017-12-26 WO PCT/CN2017/118771 patent/WO2018121550A1/zh not_active Ceased
- 2017-12-26 CN CN201780075753.0A patent/CN110382490A/zh active Pending
- 2017-12-26 EP EP22213583.2A patent/EP4169917B1/en active Active
- 2017-12-26 CA CA3174890A patent/CA3174890A1/en active Pending
- 2017-12-26 AU AU2017389818A patent/AU2017389818B2/en active Active
- 2017-12-26 JP JP2019534817A patent/JP7077323B2/ja active Active
- 2017-12-26 EP EP22213594.9A patent/EP4169918B8/en active Active
- 2017-12-26 CA CA3048546A patent/CA3048546A1/en active Pending
- 2017-12-26 EP EP17886474.0A patent/EP3560921B1/en active Active
-
2022
- 2022-04-30 AU AU2022202885A patent/AU2022202885B2/en active Active
- 2022-04-30 AU AU2022202886A patent/AU2022202886B2/en active Active
- 2022-05-18 JP JP2022081738A patent/JP7384536B2/ja active Active
- 2022-05-18 JP JP2022081736A patent/JP7384535B2/ja active Active
- 2022-09-13 US US17/944,151 patent/US12508264B2/en active Active
- 2022-09-13 US US17/944,149 patent/US12508263B2/en active Active
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