JP2021510376A5 - - Google Patents
Info
- Publication number
- JP2021510376A5 JP2021510376A5 JP2020538691A JP2020538691A JP2021510376A5 JP 2021510376 A5 JP2021510376 A5 JP 2021510376A5 JP 2020538691 A JP2020538691 A JP 2020538691A JP 2020538691 A JP2020538691 A JP 2020538691A JP 2021510376 A5 JP2021510376 A5 JP 2021510376A5
- Authority
- JP
- Japan
- Prior art keywords
- unsubstituted
- cancer
- substituted
- pharmaceutically acceptable
- acceptable salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2023156385A JP2024001052A (ja) | 2018-01-10 | 2023-09-21 | ベンズアミド化合物 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862615857P | 2018-01-10 | 2018-01-10 | |
| US62/615,857 | 2018-01-10 | ||
| PCT/US2019/012695 WO2019139899A1 (en) | 2018-01-10 | 2019-01-08 | Benzamide compounds |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023156385A Division JP2024001052A (ja) | 2018-01-10 | 2023-09-21 | ベンズアミド化合物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021510376A JP2021510376A (ja) | 2021-04-22 |
| JP2021510376A5 true JP2021510376A5 (enExample) | 2022-01-17 |
| JP7355741B2 JP7355741B2 (ja) | 2023-10-03 |
Family
ID=67218673
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020538692A Pending JP2021510165A (ja) | 2018-01-10 | 2019-01-08 | ベンズアミド化合物 |
| JP2020538644A Pending JP2021510163A (ja) | 2018-01-10 | 2019-01-08 | ベンズアミド化合物 |
| JP2020538691A Active JP7355741B2 (ja) | 2018-01-10 | 2019-01-08 | ベンズアミド化合物 |
| JP2023156385A Pending JP2024001052A (ja) | 2018-01-10 | 2023-09-21 | ベンズアミド化合物 |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020538692A Pending JP2021510165A (ja) | 2018-01-10 | 2019-01-08 | ベンズアミド化合物 |
| JP2020538644A Pending JP2021510163A (ja) | 2018-01-10 | 2019-01-08 | ベンズアミド化合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023156385A Pending JP2024001052A (ja) | 2018-01-10 | 2023-09-21 | ベンズアミド化合物 |
Country Status (16)
| Country | Link |
|---|---|
| US (7) | USRE50643E1 (enExample) |
| EP (4) | EP4556469A1 (enExample) |
| JP (4) | JP2021510165A (enExample) |
| KR (4) | KR20200108301A (enExample) |
| CN (5) | CN118084904A (enExample) |
| AR (4) | AR114998A1 (enExample) |
| AU (4) | AU2019207611A1 (enExample) |
| BR (3) | BR112020014169A2 (enExample) |
| CA (3) | CA3087261A1 (enExample) |
| ES (1) | ES3013457T3 (enExample) |
| IL (4) | IL275762B2 (enExample) |
| MX (4) | MX2020007014A (enExample) |
| RU (2) | RU2020120929A (enExample) |
| SG (3) | SG11202005785XA (enExample) |
| TW (5) | TW201930317A (enExample) |
| WO (4) | WO2019139902A1 (enExample) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3565815B1 (en) | 2017-01-07 | 2024-03-13 | Fochon Pharmaceuticals, Ltd. | Compounds as bcl-2-selective apoptosis-inducing agents |
| EP3612531B1 (en) | 2017-04-18 | 2022-08-24 | Shanghai Fochon Pharmaceutical Co., Ltd. | Apoptosis-inducing agents |
| KR20200108301A (ko) | 2018-01-10 | 2020-09-17 | 리커리엄 아이피 홀딩스, 엘엘씨 | 벤즈아미드 화합물 |
| KR20220034038A (ko) * | 2019-07-10 | 2022-03-17 | 리커리엄 아이피 홀딩스, 엘엘씨 | Bcl-2 억제제의 나노입자 제형 |
| AU2020310147A1 (en) * | 2019-07-10 | 2022-01-06 | Recurium Ip Holdings, Llc | Bcl-2 protein inhibitors |
| JP7142173B2 (ja) | 2019-12-06 | 2022-09-26 | ロクソ オンコロジー， インコーポレイテッド | ブルトン型チロシンキナーゼ阻害剤の投薬 |
| AU2020407070A1 (en) * | 2019-12-20 | 2022-07-14 | Recurium Ip Holdings, Llc | Combinations |
| IL294067A (en) * | 2019-12-20 | 2022-08-01 | Recurium Ip Holdings Llc | Combinations |
| AU2020404996A1 (en) * | 2019-12-20 | 2022-07-14 | Recurium Ip Holdings, Llc | Combinations |
| US20230065577A1 (en) * | 2019-12-20 | 2023-03-02 | Recurium Ip Holdings, Llc | Combinations |
| WO2021167987A1 (en) | 2020-02-21 | 2021-08-26 | Recurium Ip Holdings, Llc | Difluoromethyl iodo compounds and methods |
| US20230167105A1 (en) * | 2020-04-28 | 2023-06-01 | Recurium Ip Holdings, Llc | Bcl-2 protein inhibitors |
| JP2023525022A (ja) * | 2020-05-07 | 2023-06-14 | リキュリウム アイピー ホールディングス リミテッド ライアビリティー カンパニー | 組み合わせ |
| BR112022023486A2 (pt) * | 2020-05-19 | 2023-01-10 | Recurium Ip Holdings Llc | Tratamento para amiloidose |
| BR112023000320A2 (pt) * | 2020-07-10 | 2023-01-31 | Jiangsu Hengrui Pharmaceuticals Co Ltd | Derivado de sulfonilbenzamida e seu cojugado, método de preparação do mesmo e seu uso |
| US20230381172A1 (en) * | 2020-10-16 | 2023-11-30 | Recurium Ip Holdings, Llc | Combinations of bcl-2 inhibitors with chemotherapeutic agents |
| WO2022133446A1 (en) * | 2020-12-16 | 2022-06-23 | Recurium Ip Holdings, Llc | Combinations |
| CN113143930B (zh) * | 2021-04-08 | 2023-05-30 | 深圳湾实验室 | 化合物在制备SARS-Cov-2 E蛋白抑制剂中的用途 |
| CN113816889B (zh) * | 2021-10-11 | 2023-08-22 | 中国药科大学 | 一类4-磺酰亚胺-1H-吡咯类Mcl-1抑制剂及其抗肿瘤医药用途 |
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2019
- 2019-01-08 KR KR1020207022537A patent/KR20200108301A/ko not_active Withdrawn
- 2019-01-08 EP EP25150549.1A patent/EP4556469A1/en not_active Withdrawn
- 2019-01-08 CN CN202410225030.6A patent/CN118084904A/zh active Pending
- 2019-01-08 CN CN201980015896.1A patent/CN111801320A/zh active Pending
- 2019-01-08 US US18/212,692 patent/USRE50643E1/en active Active
- 2019-01-08 AU AU2019207611A patent/AU2019207611A1/en not_active Abandoned
- 2019-01-08 CN CN201980015923.5A patent/CN111788203A/zh active Pending
- 2019-01-08 EP EP19738922.4A patent/EP3737672A4/en not_active Withdrawn
- 2019-01-08 BR BR112020014169-0A patent/BR112020014169A2/pt active IP Right Grant
- 2019-01-08 WO PCT/US2019/012704 patent/WO2019139902A1/en not_active Ceased
- 2019-01-08 JP JP2020538692A patent/JP2021510165A/ja active Pending
- 2019-01-08 WO PCT/US2019/012699 patent/WO2019139900A1/en not_active Ceased
- 2019-01-08 BR BR112020014160-7A patent/BR112020014160A2/pt not_active Application Discontinuation
- 2019-01-08 IL IL275762A patent/IL275762B2/en unknown
- 2019-01-08 KR KR1020207022538A patent/KR102751751B1/ko active Active
- 2019-01-08 CN CN201980015882.XA patent/CN111801327B/zh active Active
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- 2019-01-08 IL IL316472A patent/IL316472A/en unknown
- 2019-01-08 JP JP2020538644A patent/JP2021510163A/ja active Pending
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- 2019-01-08 JP JP2020538691A patent/JP7355741B2/ja active Active
- 2019-01-08 ES ES19738996T patent/ES3013457T3/es active Active
- 2019-01-08 CN CN202410225032.5A patent/CN118084905A/zh active Pending
- 2019-01-08 RU RU2020120929A patent/RU2020120929A/ru unknown
- 2019-01-08 SG SG11202005785XA patent/SG11202005785XA/en unknown
- 2019-01-08 SG SG11202005985PA patent/SG11202005985PA/en unknown
- 2019-01-08 MX MX2020007014A patent/MX2020007014A/es unknown
- 2019-01-08 EP EP19738996.8A patent/EP3740487B1/en active Active
- 2019-01-08 US US16/957,865 patent/US11590126B2/en active Active
- 2019-01-08 CA CA3087262A patent/CA3087262A1/en active Pending
- 2019-01-08 US US16/957,862 patent/US11344546B2/en active Active
- 2019-01-08 RU RU2020120928A patent/RU2020120928A/ru unknown
- 2019-01-08 AU AU2019207616A patent/AU2019207616A1/en not_active Abandoned
- 2019-01-08 WO PCT/US2019/012719 patent/WO2019139907A1/en not_active Ceased
- 2019-01-08 US US16/957,861 patent/US11318134B2/en not_active Ceased
- 2019-01-08 CA CA3087263A patent/CA3087263A1/en active Pending
- 2019-01-08 KR KR1020247043033A patent/KR20250008139A/ko active Pending
- 2019-01-08 MX MX2020007392A patent/MX2020007392A/es unknown
- 2019-01-08 WO PCT/US2019/012695 patent/WO2019139899A1/en not_active Ceased
- 2019-01-08 MX MX2020007388A patent/MX2020007388A/es unknown
- 2019-01-08 SG SG11202005784YA patent/SG11202005784YA/en unknown
- 2019-01-08 BR BR112020014151-8A patent/BR112020014151A2/pt not_active Application Discontinuation
- 2019-01-08 KR KR1020207022443A patent/KR20200108298A/ko not_active Withdrawn
- 2019-01-10 AR ARP190100053A patent/AR114998A1/es unknown
- 2019-01-10 TW TW108101047A patent/TW201930317A/zh unknown
- 2019-01-10 TW TW113101066A patent/TW202417442A/zh unknown
- 2019-01-10 AR ARP190100051A patent/AR114949A1/es not_active Application Discontinuation
- 2019-01-10 TW TW108101046A patent/TW201934538A/zh unknown
- 2019-01-10 TW TW108101048A patent/TWI829664B/zh active
- 2019-01-10 TW TW108101045A patent/TW201934550A/zh unknown
- 2019-01-10 AR ARP190100050A patent/AR114948A1/es unknown
- 2019-01-10 AR ARP190100052A patent/AR114950A1/es not_active Application Discontinuation
-
2020
- 2020-06-30 IL IL275761A patent/IL275761A/en unknown
- 2020-06-30 IL IL275763A patent/IL275763A/en unknown
- 2020-07-13 MX MX2023009185A patent/MX2023009185A/es unknown
-
2022
- 2022-03-28 US US17/656,726 patent/US11813259B2/en active Active
-
2023
- 2023-05-26 US US18/202,622 patent/US11813260B1/en active Active
- 2023-09-20 US US18/471,017 patent/US20240180899A1/en not_active Abandoned
- 2023-09-21 JP JP2023156385A patent/JP2024001052A/ja active Pending
-
2024
- 2024-06-06 AU AU2024203833A patent/AU2024203833A1/en active Pending
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