JP2020528889A5 - - Google Patents

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JP2020528889A5
JP2020528889A5 JP2020502955A JP2020502955A JP2020528889A5 JP 2020528889 A5 JP2020528889 A5 JP 2020528889A5 JP 2020502955 A JP2020502955 A JP 2020502955A JP 2020502955 A JP2020502955 A JP 2020502955A JP 2020528889 A5 JP2020528889 A5 JP 2020528889A5
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JP
Japan
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alkyl
membered
aryl
hydroxy
alkoxy
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JP2020502955A
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Japanese (ja)
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JP7349981B2 (ja
JP2020528889A (ja
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Priority claimed from PCT/US2018/043330 external-priority patent/WO2019023145A1/en
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JP2020502955A 2017-07-24 2018-07-23 Nlrp活性に関連する状態を治療するための化合物及び組成物 Active JP7349981B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201762536352P 2017-07-24 2017-07-24
US62/536,352 2017-07-24
US201762573935P 2017-10-18 2017-10-18
US62/573,935 2017-10-18
PCT/US2018/043330 WO2019023145A1 (en) 2017-07-24 2018-07-23 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PATHOLOGICAL CONDITIONS ASSOCIATED WITH NLRP ACTIVITY

Publications (3)

Publication Number Publication Date
JP2020528889A JP2020528889A (ja) 2020-10-01
JP2020528889A5 true JP2020528889A5 (enExample) 2021-09-02
JP7349981B2 JP7349981B2 (ja) 2023-09-25

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ID=63143409

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JP2020502955A Active JP7349981B2 (ja) 2017-07-24 2018-07-23 Nlrp活性に関連する状態を治療するための化合物及び組成物

Country Status (6)

Country Link
US (2) US11370763B2 (enExample)
EP (1) EP3658538B1 (enExample)
JP (1) JP7349981B2 (enExample)
CN (1) CN111094242B (enExample)
ES (1) ES2949404T3 (enExample)
WO (1) WO2019023145A1 (enExample)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN117209447A (zh) 2017-07-24 2023-12-12 诺华股份有限公司 用于治疗与nlrp活性相关的病症的化合物和组合物
PE20200758A1 (es) 2017-08-15 2020-07-27 Inflazome Ltd Sulfonilureas y sulfoniltioureas como inhibidores de nlrp3
WO2019068772A1 (en) 2017-10-03 2019-04-11 Inflazome Limited NEW COMPOUNDS
US20210395241A1 (en) * 2018-07-03 2021-12-23 Novartis Ag Nlrp modulators
CA3103664A1 (en) * 2018-07-03 2020-01-09 Novartis Ag Methods of treating or selecting a treatment for a subject resistant to tnf inhibitor using a nlrp3 antagonist
GB201902327D0 (en) 2019-02-20 2019-04-03 Inflazome Ltd Novel compounds
PE20211333A1 (es) 2018-08-15 2021-07-22 Inflazome Ltd Compuestos de sulfonamidaurea novedosos
CN120531732A (zh) * 2018-11-13 2025-08-26 诺华股份有限公司 用于治疗与nlrp活性相关的病症的化合物和组合物
US12134611B2 (en) 2018-11-13 2024-11-05 Novartis Ag Compounds and compositions for treating conditions associated with NLRP activity
CN113227055A (zh) * 2018-11-16 2021-08-06 诺华股份有限公司 用于治疗与nlrp活性相关的病症的化合物和组合物
GB201819083D0 (en) 2018-11-23 2019-01-09 Inflazome Ltd Novel compounds
GB201905265D0 (en) 2019-04-12 2019-05-29 Inflazome Ltd Inflammasome inhibition
US20220378801A1 (en) 2019-06-21 2022-12-01 Ac Immune Sa Novel compounds
WO2021002887A1 (en) * 2019-07-02 2021-01-07 Novartis Inflammasome Research, Inc. Gut-targeted nlrp3 antagonists and their use in therapy
EP4013762A1 (en) 2019-08-16 2022-06-22 Inflazome Limited Macrocyclic sulfonylamide derivatives useful as nlrp3 inhibitors
JP2022545400A (ja) 2019-08-16 2022-10-27 インフレイゾーム リミテッド Nlrp3阻害剤として有用な大環状スルホニル尿素誘導体
JP2022547882A (ja) 2019-09-06 2022-11-16 インフレイゾーム リミテッド Nlrp3阻害剤
JP2023513935A (ja) 2020-02-18 2023-04-04 インフレイゾーム リミテッド 化合物
AU2021244313A1 (en) 2020-03-25 2022-11-17 Olatec Therapeutics Llc Method for treating diabetes
CA3178361A1 (en) 2020-06-19 2021-12-23 Emanuele Gabellieri Dihydrooxazole and thiourea derivatives modulating the nlrp3 inflammasome pathway
WO2022023907A1 (en) 2020-07-31 2022-02-03 Novartis Ag Methods of selecting and treating patients at elevated risk of major adverse cardiac events
US11932630B2 (en) 2021-04-16 2024-03-19 Novartis Ag Heteroaryl aminopropanol derivatives
WO2022237781A1 (zh) * 2021-05-10 2022-11-17 成都百裕制药股份有限公司 酰胺衍生物及其应用
US20250109126A1 (en) 2021-12-22 2025-04-03 Ac Immune Sa Dihydro-oxazol derivative compounds
JP2025524640A (ja) 2022-07-14 2025-07-30 エーシー・イミューン・エス・アー Nlrp3インフラマソーム経路の調節剤としてのピロロトリアジン及びイミダゾトリアジン誘導体
CN119998284A (zh) 2022-07-28 2025-05-13 Ac免疫有限公司 新化合物
WO2024249539A1 (en) 2023-06-02 2024-12-05 Merck Sharp & Dohme Llc 5,6 unsaturated bicyclic heterocyles useful as inhibitors of nod-like receptor protein 3
WO2025133307A1 (en) 2023-12-22 2025-06-26 Ac Immune Sa Heterocyclic modulators of the nlrp3 inflammasome pathway
TW202545527A (zh) 2024-01-16 2025-12-01 英商諾得瑟拉公司 Nlrp3及glp-1a組合療法
WO2025153624A1 (en) 2024-01-17 2025-07-24 Ac Immune Sa Imidazo[1,2-d][1,2,4]triazine derivatives for use as inhibitors of the nlrp3 inflammasome pathway
WO2025153625A1 (en) 2024-01-17 2025-07-24 Ac Immune Sa Imidazo[1,2-d][1,2,4]triazine derivatives for use as inhibitors of the nlrp3 inflammasome pathway
WO2025163069A1 (en) 2024-01-31 2025-08-07 Ac Immune Sa Novel compounds
CN119680348A (zh) * 2025-02-05 2025-03-25 上海惠志环保科技有限公司 一种应用于含高浓度二氯甲烷废气处理方法及其系统

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ245458A (en) * 1991-12-20 1995-04-27 Lilly Co Eli Sulphonimidamide derivatives and pharmaceutical compositions
MY193765A (en) * 2015-02-16 2022-10-27 Univ Queensland Sulfonylureas and related compounds and use of same
US11447460B2 (en) * 2016-04-18 2022-09-20 Novartis Ag Compounds and compositions for treating conditions associated with NLRP activity
JP7050751B2 (ja) 2016-04-18 2022-04-08 ノバルティス アーゲー Nlrp活性に関連する状態を処置するための化合物および組成物
CA3103664A1 (en) * 2018-07-03 2020-01-09 Novartis Ag Methods of treating or selecting a treatment for a subject resistant to tnf inhibitor using a nlrp3 antagonist

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