JP2020519684A5 - - Google Patents

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JP2020519684A5
JP2020519684A5 JP2020512764A JP2020512764A JP2020519684A5 JP 2020519684 A5 JP2020519684 A5 JP 2020519684A5 JP 2020512764 A JP2020512764 A JP 2020512764A JP 2020512764 A JP2020512764 A JP 2020512764A JP 2020519684 A5 JP2020519684 A5 JP 2020519684A5
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oxy
oxo
diazabicyclo
octane
substituted
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JP2020512764A
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Japanese (ja)
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JP6909924B2 (ja
JP2020519684A (ja
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Priority claimed from US15/934,497 external-priority patent/US10085999B1/en
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Priority to JP2021111184A priority Critical patent/JP2021165298A/ja
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JP2020512764A 2017-05-10 2018-05-02 ベータ−ラクタマーゼ阻害剤およびその使用 Active JP6909924B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2021111184A JP2021165298A (ja) 2017-05-10 2021-07-05 ベータ−ラクタマーゼ阻害剤およびその使用

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201762504523P 2017-05-10 2017-05-10
US62/504,523 2017-05-10
US201762551043P 2017-08-28 2017-08-28
US62/551,043 2017-08-28
US15/934,497 2018-03-23
US15/934,497 US10085999B1 (en) 2017-05-10 2018-03-23 Beta-lactamase inhibitors and uses thereof
PCT/US2018/030652 WO2018208557A1 (en) 2017-05-10 2018-05-02 3-(((((2s,5r)-2-carbamoyl-7-oxo-1,6-diazabicyclo[3.2.1]octan-6-yl)oxy)sulfonyl)oxy)-2,2-dimethylprop noate derivatives and related compounds as perorally administered profrugs of beta-lactamase inhibitors for treating bacterial infections

Related Child Applications (1)

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JP2021111184A Division JP2021165298A (ja) 2017-05-10 2021-07-05 ベータ−ラクタマーゼ阻害剤およびその使用

Publications (3)

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JP2020519684A JP2020519684A (ja) 2020-07-02
JP2020519684A5 true JP2020519684A5 (https=) 2021-02-04
JP6909924B2 JP6909924B2 (ja) 2021-07-28

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ID=63639355

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JP2020512764A Active JP6909924B2 (ja) 2017-05-10 2018-05-02 ベータ−ラクタマーゼ阻害剤およびその使用
JP2021111184A Pending JP2021165298A (ja) 2017-05-10 2021-07-05 ベータ−ラクタマーゼ阻害剤およびその使用

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JP2021111184A Pending JP2021165298A (ja) 2017-05-10 2021-07-05 ベータ−ラクタマーゼ阻害剤およびその使用

Country Status (22)

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US (6) US10085999B1 (https=)
EP (1) EP3625233B9 (https=)
JP (2) JP6909924B2 (https=)
KR (1) KR102411517B1 (https=)
CN (1) CN110662746B (https=)
AU (2) AU2018266566B2 (https=)
CA (2) CA3062619C (https=)
DK (1) DK3625233T5 (https=)
ES (1) ES2955871T3 (https=)
FI (1) FI3625233T5 (https=)
HR (1) HRP20230977T1 (https=)
HU (1) HUE062752T2 (https=)
IL (2) IL296379B2 (https=)
LT (1) LT3625233T (https=)
MX (2) MX385265B (https=)
PL (1) PL3625233T3 (https=)
PT (1) PT3625233T (https=)
RS (1) RS64547B9 (https=)
RU (1) RU2753401C2 (https=)
SG (2) SG11201909429VA (https=)
SI (1) SI3625233T1 (https=)
WO (1) WO2018208557A1 (https=)

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CN114206851B (zh) 2019-04-26 2025-02-11 默沙东有限责任公司 可用于制备(2s,5r)-7-氧代-n-哌啶-4-基-6-(硫酸基)-1,6-二氮杂双环[3.2.1]辛烷-2-甲酰胺的中间体的制备方法
CA3152300C (en) * 2019-08-29 2024-04-30 Arixa Pharmaceuticals, Inc. Orally administered combinations of beta lactam antibiotics and avibactam derivatives for treating bacterial infections
US20210186983A1 (en) * 2019-12-20 2021-06-24 Arixa Pharmaceuticals, Inc. Orally administered combinations of amoxicillin and avibactam derivatives for treating mycobacterial infections
AU2021266715A1 (en) 2020-05-05 2022-11-17 Qpex Biopharma, Inc. Boronic acid derivatives and synthesis, polymorphic forms, and therapeutic uses thereof
CN111943950B (zh) * 2020-09-10 2022-03-29 山东安信制药有限公司 一种瑞来巴坦的制备方法
JP2024512793A (ja) * 2021-04-05 2024-03-19 キューペックス バイオファーマ, インコーポレイテッド セフチブテン投与レジメン
CN115448920B (zh) * 2022-10-14 2025-01-03 广州楷石医药有限公司 一种β-内酰胺酶抑制剂及其应用
GB202306833D0 (en) 2023-05-09 2023-06-21 Adjutec Pharma As Therapy
GB202306826D0 (en) 2023-05-09 2023-06-21 Adjutec Pharma As Therapy
CN119431373B (zh) * 2024-07-24 2025-08-08 科睿迪(南京)医药科技有限公司 一种β-内酰胺酶抑制剂及其用途
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CN119841826B (zh) * 2024-09-30 2026-04-10 科睿迪(南京)医药科技有限公司 二氮杂二环类β-内酰胺酶抑制剂及其应用

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