JP2019529543A5 - - Google Patents

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Publication number
JP2019529543A5
JP2019529543A5 JP2019535434A JP2019535434A JP2019529543A5 JP 2019529543 A5 JP2019529543 A5 JP 2019529543A5 JP 2019535434 A JP2019535434 A JP 2019535434A JP 2019535434 A JP2019535434 A JP 2019535434A JP 2019529543 A5 JP2019529543 A5 JP 2019529543A5
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JP
Japan
Prior art keywords
pharmaceutical composition
injectable pharmaceutical
once
group
acyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2019535434A
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English (en)
Japanese (ja)
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JP6929367B2 (ja
JP2019529543A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/CN2017/101327 external-priority patent/WO2018050043A1/en
Publication of JP2019529543A publication Critical patent/JP2019529543A/ja
Publication of JP2019529543A5 publication Critical patent/JP2019529543A5/ja
Application granted granted Critical
Publication of JP6929367B2 publication Critical patent/JP6929367B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2019535434A 2016-09-13 2017-09-12 ブプレノルフィン徐放性製剤 Active JP6929367B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662394168P 2016-09-13 2016-09-13
US62/394,168 2016-09-13
PCT/CN2017/101327 WO2018050043A1 (en) 2016-09-13 2017-09-12 Sustained-release buprenorphine formulations background of invention

Publications (3)

Publication Number Publication Date
JP2019529543A JP2019529543A (ja) 2019-10-17
JP2019529543A5 true JP2019529543A5 (https=) 2020-08-06
JP6929367B2 JP6929367B2 (ja) 2021-09-01

Family

ID=61619029

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2019535434A Active JP6929367B2 (ja) 2016-09-13 2017-09-12 ブプレノルフィン徐放性製剤

Country Status (31)

Country Link
US (1) US10744132B2 (https=)
EP (1) EP3512518B1 (https=)
JP (1) JP6929367B2 (https=)
KR (1) KR102244500B1 (https=)
CN (1) CN109789137B (https=)
AR (1) AR110468A1 (https=)
AU (1) AU2017325910B2 (https=)
BR (1) BR112019004923A2 (https=)
CA (1) CA3033046C (https=)
CL (1) CL2019000624A1 (https=)
CO (1) CO2019003632A2 (https=)
DK (1) DK3512518T3 (https=)
ES (1) ES2934721T3 (https=)
FI (1) FI3512518T3 (https=)
HR (1) HRP20230062T8 (https=)
HU (1) HUE060906T2 (https=)
LT (1) LT3512518T (https=)
MX (1) MX374304B (https=)
MY (1) MY196269A (https=)
PE (1) PE20190707A1 (https=)
PH (1) PH12019500466A1 (https=)
PL (1) PL3512518T3 (https=)
PT (1) PT3512518T (https=)
RS (1) RS63894B1 (https=)
RU (1) RU2747306C2 (https=)
SG (1) SG11201901294QA (https=)
SI (1) SI3512518T1 (https=)
SM (1) SMT202300006T1 (https=)
TW (1) TWI743193B (https=)
WO (1) WO2018050043A1 (https=)
ZA (1) ZA201900890B (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1057075C (zh) * 1997-09-10 2000-10-04 中国石油化工总公司 低碳烯烃直接水合连续生产低碳醇的方法
BR112020016576A2 (pt) 2018-05-11 2020-12-15 Alar Pharmaceuticals Inc. Formulações injetáveis de ação prolongada e formas cristalinas de derivados de buprenorfina
KR102898979B1 (ko) * 2018-12-27 2025-12-10 에일러 파마슈티컬스 아이엔씨. 주사가능한 날트렉손 서방형 약학 제제
EP3936112A1 (en) * 2020-07-07 2022-01-12 Occlugel Hydrophilic degradable microspheres for delivering buprenorphine
IL308211A (en) * 2021-05-05 2024-01-01 Lyndra Therapeutics Inc Gastric residence systems comprising methadone

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RO121631B1 (ro) 1999-08-27 2008-01-30 Southern Research Institute Compoziţie cu buprenorfină şi utilizarea acesteia pentru reducerea consumului de heroină şi/sau alcool
DE60329515D1 (de) 2002-10-25 2009-11-12 Euro Celtique Sa Analoga und prodrugs von buprenorphin
CN1263760C (zh) * 2002-11-12 2006-07-12 财团法人奇美医院 新颖的丁丙诺啡酯衍生物及其制备方法,以及长效作用镇痛药学组合物
TWI226830B (en) * 2002-11-12 2005-01-21 Chi Mei Foundation Medical Ct Novel ester derivatives of buprenorphine and their preparation processes, and long acting analgesic pharmaceutical compositions
DE60224288T2 (de) 2002-11-25 2009-04-16 Chi Mei Foundation Medical Center Buprenorphinesterderivate, Verfahren zu ihrer Herstellung, und langwirksame analgetische Arzneimittel
WO2005117830A1 (en) 2004-06-04 2005-12-15 Camurus Ab Liquid depot formulations
RU2008124805A (ru) * 2005-11-21 2009-12-27 Шеринг-Плоу Лтд. (CH) Фармацевтические композиции, содержащие бупренорфин
GB0606124D0 (en) 2006-03-28 2006-05-03 Reckitt Benckiser Healthcare Buprenorphine derivatives and uses thereof
ES2549115T3 (es) * 2006-09-22 2015-10-23 Zynerba Pharmaceuticals, Inc. Profármacos de buprenorfina administrables por vía transdérmica y composiciones resistentes al consumo excesivo de los mismos
US20090181068A1 (en) * 2008-01-14 2009-07-16 Dunn Richard L Low Viscosity Liquid Polymeric Delivery System
GB2481017B (en) 2010-06-08 2015-01-07 Rb Pharmaceuticals Ltd Microparticle buprenorphine suspension
GB2481018B (en) 2010-06-08 2015-03-18 Rb Pharmaceuticals Ltd Injectable flowable composition comprising buprenorphine
FR2975912B1 (fr) 2011-05-30 2013-06-14 Flamel Tech Sa Composition a liberation controlee de buprenorphine
US9393211B2 (en) 2013-03-15 2016-07-19 Oakwood Laboratories LLC High drug load buprenorphine microspheres and method of producing same
GB201404139D0 (en) * 2014-03-10 2014-04-23 Rb Pharmaceuticals Ltd Sustained release buprenorphine solution formulations
GB201419091D0 (en) * 2014-10-27 2014-12-10 Camurus Ab Formulations

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