JP2019524844A5 - - Google Patents
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- Publication number
- JP2019524844A5 JP2019524844A5 JP2019509528A JP2019509528A JP2019524844A5 JP 2019524844 A5 JP2019524844 A5 JP 2019524844A5 JP 2019509528 A JP2019509528 A JP 2019509528A JP 2019509528 A JP2019509528 A JP 2019509528A JP 2019524844 A5 JP2019524844 A5 JP 2019524844A5
- Authority
- JP
- Japan
- Prior art keywords
- hexahydro
- pyrazino
- diazanaphthalene
- compound according
- hydrogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662377119P | 2016-08-19 | 2016-08-19 | |
| US62/377,119 | 2016-08-19 | ||
| PCT/US2017/047644 WO2018035477A1 (en) | 2016-08-19 | 2017-08-18 | 5-ht2c receptor agonists and compositions and methods of use |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2019524844A JP2019524844A (ja) | 2019-09-05 |
| JP2019524844A5 true JP2019524844A5 (enExample) | 2020-09-24 |
| JP6977024B2 JP6977024B2 (ja) | 2021-12-08 |
Family
ID=59799461
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019509528A Expired - Fee Related JP6977024B2 (ja) | 2016-08-19 | 2017-08-18 | ５−ｈｔ２ｃ受容体アゴニストおよび組成物ならびに使用方法 |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US10836764B2 (enExample) |
| EP (1) | EP3500570B1 (enExample) |
| JP (1) | JP6977024B2 (enExample) |
| KR (1) | KR20190049732A (enExample) |
| CN (1) | CN109952301B (enExample) |
| AU (1) | AU2017313908C1 (enExample) |
| BR (1) | BR112019003142A2 (enExample) |
| CA (1) | CA3033142A1 (enExample) |
| EA (1) | EA038219B1 (enExample) |
| IL (1) | IL264682B (enExample) |
| MA (1) | MA45987A (enExample) |
| MX (1) | MX391442B (enExample) |
| NZ (1) | NZ750469A (enExample) |
| WO (1) | WO2018035477A1 (enExample) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3500570B1 (en) * | 2016-08-19 | 2022-10-05 | Arena Pharmaceuticals, Inc. | 5-ht2c receptor agonists and compositions and methods of use |
| US12459965B2 (en) | 2017-10-09 | 2025-11-04 | Compass Pathfinder Limited | Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use |
| GB2571696B (en) | 2017-10-09 | 2020-05-27 | Compass Pathways Ltd | Large scale method for the preparation of Psilocybin and formulations of Psilocybin so produced |
| US20210052600A1 (en) | 2017-12-27 | 2021-02-25 | Takeda Pharmaceutical Company Limited | Therapeutic agents for stress urinary incontinence and incotinence of feces |
| WO2020061103A1 (en) | 2018-09-18 | 2020-03-26 | Nikang Therapeutics, Inc. | Fused tricyclic ring derivatives as src homology-2 phosphatase inhibitors |
| EP3860996A4 (en) | 2018-10-02 | 2022-08-31 | Northwestern University | BETA-CARBOLINES AS POSITIVE ALLOSTERIC MODULATORS OF HUMAN SEROTONIN RECEPTOR 2C (5-HT2C) |
| WO2020212951A1 (en) | 2019-04-17 | 2020-10-22 | Compass Pathfinder Limited | Methods for treating anxiety disorders, headache disorders, and eating disorders with psilocybin |
| US20230277568A1 (en) * | 2020-07-10 | 2023-09-07 | Eleusis Therapeutics Us, Inc. | Method of treatment for psilocybin or psilocin infusion |
| US11312684B1 (en) | 2021-02-10 | 2022-04-26 | Eleusis Therapeutics Us, Inc. | Pharmaceutically acceptable salts of psilocin and uses thereof |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4597961A (en) | 1985-01-23 | 1986-07-01 | Etscorn Frank T | Transcutaneous application of nicotine |
| US4920989A (en) | 1985-04-25 | 1990-05-01 | Regents Of The University Of California | Method and apparatus for aiding in the reduction of incidence of tobacco smoking |
| IL86170A (en) | 1987-05-01 | 1992-12-01 | Elan Transdermal Ltd | Preparations and compositions comprising nicotine for percutaneous administration |
| US5004610A (en) | 1988-06-14 | 1991-04-02 | Alza Corporation | Subsaturated nicotine transdermal therapeutic system |
| AU8057491A (en) | 1990-07-03 | 1992-02-04 | Quaker Chemical Corporation (A Delaware Corporation) | Aqueous coolant |
| WO1992018005A1 (en) | 1991-04-16 | 1992-10-29 | National Institutes Of Health | Method of treating trichotillomania and onychophagia |
| GB0202015D0 (en) * | 2002-01-29 | 2002-03-13 | Hoffmann La Roche | Piperazine Derivatives |
| EP1494533A2 (en) | 2002-04-12 | 2005-01-12 | The University of Chicago | Farnesoid x-activated receptor agonists |
| JP5520051B2 (ja) * | 2007-11-15 | 2014-06-11 | 武田薬品工業株式会社 | 縮合ピリジン誘導体およびその用途 |
| US8518933B2 (en) * | 2009-04-23 | 2013-08-27 | Abbvie Inc. | Modulators of 5-HT receptors and methods of use thereof |
| JP6272695B2 (ja) * | 2010-09-01 | 2018-01-31 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 体重管理のために有用な５−ｈｔ２ｃアゴニストの改変放出剤形 |
| WO2015066344A1 (en) | 2013-11-01 | 2015-05-07 | Arena Pharmaceuticals, Inc. | 5-ht2c receptor agonists and compositions and methods of use |
| WO2015161285A1 (en) * | 2014-04-17 | 2015-10-22 | G1 Therapeutics, Inc. | Tricyclic lactams for use in the protection of hematopoietic stem and progenitor cells against ionizing radiation |
| EP3500570B1 (en) * | 2016-08-19 | 2022-10-05 | Arena Pharmaceuticals, Inc. | 5-ht2c receptor agonists and compositions and methods of use |
-
2017
- 2017-08-18 EP EP17762266.9A patent/EP3500570B1/en active Active
- 2017-08-18 CN CN201780062933.5A patent/CN109952301B/zh not_active Expired - Fee Related
- 2017-08-18 EA EA201990527A patent/EA038219B1/ru not_active IP Right Cessation
- 2017-08-18 AU AU2017313908A patent/AU2017313908C1/en not_active Ceased
- 2017-08-18 BR BR112019003142-1A patent/BR112019003142A2/pt not_active IP Right Cessation
- 2017-08-18 JP JP2019509528A patent/JP6977024B2/ja not_active Expired - Fee Related
- 2017-08-18 WO PCT/US2017/047644 patent/WO2018035477A1/en not_active Ceased
- 2017-08-18 KR KR1020197007503A patent/KR20190049732A/ko not_active Withdrawn
- 2017-08-18 US US16/326,522 patent/US10836764B2/en active Active
- 2017-08-18 MX MX2019002020A patent/MX391442B/es unknown
- 2017-08-18 NZ NZ750469A patent/NZ750469A/en not_active IP Right Cessation
- 2017-08-18 MA MA045987A patent/MA45987A/fr unknown
- 2017-08-18 CA CA3033142A patent/CA3033142A1/en active Pending
-
2019
- 2019-02-06 IL IL264682A patent/IL264682B/en unknown
-
2020
- 2020-10-19 US US17/073,458 patent/US11608339B2/en active Active
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