JP2019507791A5 - - Google Patents

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Publication number
JP2019507791A5
JP2019507791A5 JP2018547929A JP2018547929A JP2019507791A5 JP 2019507791 A5 JP2019507791 A5 JP 2019507791A5 JP 2018547929 A JP2018547929 A JP 2018547929A JP 2018547929 A JP2018547929 A JP 2018547929A JP 2019507791 A5 JP2019507791 A5 JP 2019507791A5
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JP
Japan
Prior art keywords
compound
pharmaceutically acceptable
dihydroxybutan
sulfonamide
thio
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Application number
JP2018547929A
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English (en)
Japanese (ja)
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JP6883917B2 (ja
JP2019507791A (ja
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Priority claimed from PCT/US2017/021570 external-priority patent/WO2017156270A1/en
Publication of JP2019507791A publication Critical patent/JP2019507791A/ja
Publication of JP2019507791A5 publication Critical patent/JP2019507791A5/ja
Priority to JP2021078242A priority Critical patent/JP7126014B2/ja
Application granted granted Critical
Publication of JP6883917B2 publication Critical patent/JP6883917B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2018547929A 2016-03-11 2017-03-09 結晶性関節障害を処置するためのcxcr−2阻害剤 Expired - Fee Related JP6883917B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2021078242A JP7126014B2 (ja) 2016-03-11 2021-05-05 結晶性関節障害を処置するためのcxcr-2阻害剤

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662307348P 2016-03-11 2016-03-11
US62/307,348 2016-03-11
PCT/US2017/021570 WO2017156270A1 (en) 2016-03-11 2017-03-09 Cxcr-2 inhibitors for treating crystal arthropathy disorders

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2021078242A Division JP7126014B2 (ja) 2016-03-11 2021-05-05 結晶性関節障害を処置するためのcxcr-2阻害剤

Publications (3)

Publication Number Publication Date
JP2019507791A JP2019507791A (ja) 2019-03-22
JP2019507791A5 true JP2019507791A5 (https=) 2020-04-30
JP6883917B2 JP6883917B2 (ja) 2021-06-09

Family

ID=59789863

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2018547929A Expired - Fee Related JP6883917B2 (ja) 2016-03-11 2017-03-09 結晶性関節障害を処置するためのcxcr−2阻害剤
JP2021078242A Active JP7126014B2 (ja) 2016-03-11 2021-05-05 結晶性関節障害を処置するためのcxcr-2阻害剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2021078242A Active JP7126014B2 (ja) 2016-03-11 2021-05-05 結晶性関節障害を処置するためのcxcr-2阻害剤

Country Status (10)

Country Link
US (1) US10772886B2 (https=)
EP (1) EP3426253A4 (https=)
JP (2) JP6883917B2 (https=)
CN (2) CN109152780B (https=)
AU (1) AU2017231832B2 (https=)
BR (1) BR112018068393A2 (https=)
CA (1) CA3017345A1 (https=)
CO (1) CO2018010880A2 (https=)
MX (1) MX386771B (https=)
WO (1) WO2017156270A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109152780B (zh) 2016-03-11 2021-10-01 阿迪亚生命科学公司 用于治疗结晶性关节病症的cxcr-2抑制剂
BR112020004697A2 (pt) * 2017-09-12 2020-10-27 Ardea Biosciences, Inc. inibidores de cxcr-2 para tratamento de distúrbios
EP3738956B1 (en) * 2018-01-11 2023-03-01 Shenzhen Optimum Biological Technology Co., Ltd Cxcr2 antagonist
CN114286819B (zh) 2019-07-11 2024-03-05 深圳嘉科生物科技有限公司 一种cxcr2拮抗剂的晶型及其应用
KR102260478B1 (ko) * 2019-08-19 2021-06-02 연세대학교 산학협력단 일나트륨 요소화물 결정 용해용 조성물
TW202210068A (zh) * 2020-06-05 2022-03-16 美商雅力思提雅治療公司 用於治療家族性地中海型發熱病的cxcr-2抑制劑
WO2022162021A1 (en) * 2021-01-27 2022-08-04 Astrazeneca Ab Verinurad compositions and methods of use

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AU2005210504B2 (en) 2004-01-30 2009-01-08 Merck Sharp & Dohme Corp. Crystalline polymorphs of a CXC-chemokine receptor ligand
KR101280095B1 (ko) 2004-08-28 2013-09-09 아스트라제네카 아베 케모킨 수용체 조절제로서의 피리미딘 술폰아미드 유도체
AU2008206231A1 (en) * 2007-01-19 2008-07-24 Takeda Pharmaceuticals U.S.A., Inc. Methods for preventing or reducing the number of gout flares using xanthine oxidoreductase inhibitors and anti-inflammatory agents
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CN102088993A (zh) 2008-03-20 2011-06-08 卡罗勒斯治疗公司 炎症的治疗方法
CA2730477A1 (en) 2008-07-16 2010-01-21 Astrazeneca Ab Pyrimidyl sulfonaminde derivative and its use for the treatment of chemokine mediated diseases
JP2012505160A (ja) 2008-10-06 2012-03-01 カロラス セラピューティクス, インク. 炎症を処置する方法
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CN103097377A (zh) 2010-07-13 2013-05-08 阿斯利康(瑞典)有限公司 N-[2-[[(2,3-二氟苯基)甲基]硫基]-6-{[(1r,2s)-2,3-二羟基-1-甲基丙基]氧基}-4-嘧啶基]-1-氮杂环丁烷磺酰胺的新晶形
CA2811990C (en) * 2010-08-23 2023-03-21 Dean Y. Maeda Aminopyridine- and aminopyrimidinecarboxamides as cxcr2 modulators
ES2861927T3 (es) * 2011-07-12 2021-10-06 Astrazeneca Ab N-(6-((2R,3S)-3,4-Dihidroxibutan-2-iloxi)-2-(4-fluorobenciltio)pirimidin-4-il)-3-metilacetidina-1-sulfonamida como modulador del receptor de quimiocina
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US20180221312A1 (en) 2016-03-11 2018-08-09 Ardea Biosciences, Inc. Cxcr-2 inhibitors for treating disorders
CN109152780B (zh) 2016-03-11 2021-10-01 阿迪亚生命科学公司 用于治疗结晶性关节病症的cxcr-2抑制剂
BR112020004697A2 (pt) 2017-09-12 2020-10-27 Ardea Biosciences, Inc. inibidores de cxcr-2 para tratamento de distúrbios

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