JP2013500977A5 - - Google Patents

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Publication number
JP2013500977A5
JP2013500977A5 JP2012523011A JP2012523011A JP2013500977A5 JP 2013500977 A5 JP2013500977 A5 JP 2013500977A5 JP 2012523011 A JP2012523011 A JP 2012523011A JP 2012523011 A JP2012523011 A JP 2012523011A JP 2013500977 A5 JP2013500977 A5 JP 2013500977A5
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JP
Japan
Prior art keywords
compound
pharmaceutically acceptable
pharmaceutical composition
acceptable salt
salt form
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JP2012523011A
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English (en)
Japanese (ja)
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JP2013500977A (ja
JP5738292B2 (ja
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Priority claimed from PCT/US2010/043592 external-priority patent/WO2011017178A1/en
Publication of JP2013500977A publication Critical patent/JP2013500977A/ja
Publication of JP2013500977A5 publication Critical patent/JP2013500977A5/ja
Application granted granted Critical
Publication of JP5738292B2 publication Critical patent/JP5738292B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2012523011A 2009-07-28 2010-07-28 Jak経路の阻害のための組成物および方法 Expired - Fee Related JP5738292B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22919109P 2009-07-28 2009-07-28
US61/229,191 2009-07-28
PCT/US2010/043592 WO2011017178A1 (en) 2009-07-28 2010-07-28 Compositions and methods for inhibition of the jak pathway

Publications (3)

Publication Number Publication Date
JP2013500977A JP2013500977A (ja) 2013-01-10
JP2013500977A5 true JP2013500977A5 (https=) 2013-09-12
JP5738292B2 JP5738292B2 (ja) 2015-06-24

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ID=42676842

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012523011A Expired - Fee Related JP5738292B2 (ja) 2009-07-28 2010-07-28 Jak経路の阻害のための組成物および方法

Country Status (11)

Country Link
US (1) US20110028503A1 (https=)
EP (1) EP2459195A1 (https=)
JP (1) JP5738292B2 (https=)
KR (1) KR101740076B1 (https=)
CN (2) CN102470135A (https=)
AU (3) AU2010281404A1 (https=)
BR (1) BR112012002001A2 (https=)
CA (1) CA2768543C (https=)
MX (1) MX337849B (https=)
RU (1) RU2557982C2 (https=)
WO (1) WO2011017178A1 (https=)

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HK1252685A1 (zh) 2015-11-03 2019-05-31 Theravance Biopharma R&D Ip, Llc 用於治疗呼吸疾病的jak激酶抑制剂化合物
US10406148B2 (en) 2017-05-01 2019-09-10 Theravance Biopharma R&D Ip, Llc Methods of treatment using a JAK inhibitor compound
CN107805212B (zh) * 2017-11-03 2021-08-20 宿迁德威化工股份有限公司 一种2-甲基-5-氨基苯磺酰胺的制备方法
BR112022001418A2 (pt) 2019-08-08 2022-06-07 Rigel Pharmaceuticals Inc Compostos e método para tratar a síndrome de liberação de citocinas
CN111973599A (zh) * 2020-08-07 2020-11-24 杭州邦顺制药有限公司 用于眼部疾病治疗的化合物
TW202317550A (zh) 2021-06-25 2023-05-01 美商施萬生物製藥研發 Ip有限責任公司 作為jak抑制劑之咪唑吲唑化合物

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