JP2018535235A5 - - Google Patents
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- Publication number
- JP2018535235A5 JP2018535235A5 JP2018527201A JP2018527201A JP2018535235A5 JP 2018535235 A5 JP2018535235 A5 JP 2018535235A5 JP 2018527201 A JP2018527201 A JP 2018527201A JP 2018527201 A JP2018527201 A JP 2018527201A JP 2018535235 A5 JP2018535235 A5 JP 2018535235A5
- Authority
- JP
- Japan
- Prior art keywords
- amino
- pyridazin
- acetamide
- thiadiazol
- ylpyrrolidin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562260784P | 2015-11-30 | 2015-11-30 | |
| US62/260,784 | 2015-11-30 | ||
| PCT/EP2016/079253 WO2017093301A1 (en) | 2015-11-30 | 2016-11-30 | 1,3,4-thiadiazole compounds and their use in treating cancer |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2018535235A JP2018535235A (ja) | 2018-11-29 |
| JP2018535235A5 true JP2018535235A5 (enExample) | 2020-01-16 |
| JP6821680B2 JP6821680B2 (ja) | 2021-01-27 |
Family
ID=57460503
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018527201A Active JP6821680B2 (ja) | 2015-11-30 | 2016-11-30 | １，３，４−チアジアゾール化合物およびがんの治療におけるその使用 |
Country Status (28)
| Country | Link |
|---|---|
| US (1) | US10040789B2 (enExample) |
| EP (1) | EP3383872B1 (enExample) |
| JP (1) | JP6821680B2 (enExample) |
| KR (1) | KR20180083411A (enExample) |
| CN (1) | CN108349965B (enExample) |
| AR (1) | AR106875A1 (enExample) |
| AU (1) | AU2016361834B2 (enExample) |
| BR (1) | BR112018008330B1 (enExample) |
| CA (1) | CA3005517C (enExample) |
| CL (1) | CL2018001409A1 (enExample) |
| CO (1) | CO2018006930A2 (enExample) |
| DK (1) | DK3383872T3 (enExample) |
| DO (1) | DOP2018000135A (enExample) |
| EA (1) | EA035519B9 (enExample) |
| ES (1) | ES2796562T3 (enExample) |
| IL (1) | IL259508A (enExample) |
| MX (1) | MX2018006483A (enExample) |
| MY (1) | MY195680A (enExample) |
| NI (1) | NI201800063A (enExample) |
| NZ (1) | NZ743699A (enExample) |
| PE (1) | PE20181522A1 (enExample) |
| PH (1) | PH12018501133A1 (enExample) |
| SG (1) | SG11201803808VA (enExample) |
| SV (1) | SV2018005700A (enExample) |
| TN (1) | TN2018000118A1 (enExample) |
| TW (1) | TW201731511A (enExample) |
| WO (1) | WO2017093301A1 (enExample) |
| ZA (1) | ZA201804361B (enExample) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201520959D0 (en) | 2015-11-27 | 2016-01-13 | Astrazeneca Ab And Cancer Res Technology Ltd | Bis-pyridazine compounds and their use in treating cancer |
| TW201730188A (zh) | 2015-11-30 | 2017-09-01 | 阿斯特捷利康公司 | 1,3,4-噻二唑化合物及其在治療癌症中之用途 |
| US10323028B2 (en) | 2015-11-30 | 2019-06-18 | Astrazeneca Ab | 1,3,4-thiadiazole compounds and their use in treating cancer |
| ES2939506T3 (es) * | 2018-10-16 | 2023-04-24 | Medshine Discovery Inc | Derivado de tiadiazol y usos del mismo como inhibidor de GLS1 para el tratamiento de cáncer |
| CN114560855B (zh) * | 2021-03-26 | 2023-05-23 | 成都苑东生物制药股份有限公司 | 环烷基甲酰胺类衍生物、其制备方法及用途 |
| WO2025196446A1 (en) | 2024-03-22 | 2025-09-25 | Sitryx Therapeutics Limited | Thiadiazoles as glutaminase 1 inhibitors |
| WO2025196447A1 (en) | 2024-03-22 | 2025-09-25 | Sitryx Therapeutics Limited | Thiadiazoles as glutaminase 1 inhibitors |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2012340866B2 (en) * | 2011-11-21 | 2017-03-16 | Calithera Biosciences Inc. | Heterocyclic inhibitors of glutaminase |
| US9029531B2 (en) | 2012-11-22 | 2015-05-12 | Agios Pharmaceuticals, Inc. | Compounds and their methods of use |
| WO2014079011A1 (en) * | 2012-11-22 | 2014-05-30 | Agios Pharmaceuticals, Inc. | Heterocyclic compounds for inhibiting glutaminase and their methods of use |
| CN105960405B (zh) | 2014-01-06 | 2021-02-19 | 理森制药股份公司 | 谷氨酰胺酶抑制剂 |
| GB201409624D0 (en) * | 2014-05-30 | 2014-07-16 | Astrazeneca Ab | 1,3,4-thiadiazole compounds and their use in treating cancer |
| TW201730188A (zh) * | 2015-11-30 | 2017-09-01 | 阿斯特捷利康公司 | 1,3,4-噻二唑化合物及其在治療癌症中之用途 |
| US10323028B2 (en) * | 2015-11-30 | 2019-06-18 | Astrazeneca Ab | 1,3,4-thiadiazole compounds and their use in treating cancer |
-
2016
- 2016-11-29 TW TW105139334A patent/TW201731511A/zh unknown
- 2016-11-29 US US15/362,989 patent/US10040789B2/en active Active
- 2016-11-30 NZ NZ743699A patent/NZ743699A/en unknown
- 2016-11-30 TN TNP/2018/000118A patent/TN2018000118A1/en unknown
- 2016-11-30 DK DK16805078.9T patent/DK3383872T3/da active
- 2016-11-30 WO PCT/EP2016/079253 patent/WO2017093301A1/en not_active Ceased
- 2016-11-30 CN CN201680067210.XA patent/CN108349965B/zh active Active
- 2016-11-30 BR BR112018008330-5A patent/BR112018008330B1/pt active IP Right Grant
- 2016-11-30 MY MYPI2018702070A patent/MY195680A/en unknown
- 2016-11-30 MX MX2018006483A patent/MX2018006483A/es unknown
- 2016-11-30 CA CA3005517A patent/CA3005517C/en active Active
- 2016-11-30 KR KR1020187017163A patent/KR20180083411A/ko not_active Withdrawn
- 2016-11-30 AR ARP160103664A patent/AR106875A1/es unknown
- 2016-11-30 JP JP2018527201A patent/JP6821680B2/ja active Active
- 2016-11-30 SG SG11201803808VA patent/SG11201803808VA/en unknown
- 2016-11-30 AU AU2016361834A patent/AU2016361834B2/en active Active
- 2016-11-30 EA EA201891239A patent/EA035519B9/ru not_active IP Right Cessation
- 2016-11-30 EP EP16805078.9A patent/EP3383872B1/en active Active
- 2016-11-30 ES ES16805078T patent/ES2796562T3/es active Active
- 2016-11-30 PE PE2018001012A patent/PE20181522A1/es unknown
-
2018
- 2018-05-22 IL IL259508A patent/IL259508A/en active IP Right Grant
- 2018-05-24 CL CL2018001409A patent/CL2018001409A1/es unknown
- 2018-05-29 DO DO2018000135A patent/DOP2018000135A/es unknown
- 2018-05-29 SV SV2018005700A patent/SV2018005700A/es unknown
- 2018-05-29 NI NI201800063A patent/NI201800063A/es unknown
- 2018-05-29 PH PH12018501133A patent/PH12018501133A1/en unknown
- 2018-06-28 ZA ZA2018/04361A patent/ZA201804361B/en unknown
- 2018-06-29 CO CONC2018/0006930A patent/CO2018006930A2/es unknown
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