JP2018524339A5 - - Google Patents

Download PDF

Info

Publication number
JP2018524339A5
JP2018524339A5 JP2017567655A JP2017567655A JP2018524339A5 JP 2018524339 A5 JP2018524339 A5 JP 2018524339A5 JP 2017567655 A JP2017567655 A JP 2017567655A JP 2017567655 A JP2017567655 A JP 2017567655A JP 2018524339 A5 JP2018524339 A5 JP 2018524339A5
Authority
JP
Japan
Prior art keywords
ring
alkyl
compound
optionally
fluoro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2017567655A
Other languages
English (en)
Japanese (ja)
Other versions
JP2018524339A (ja
JP7099824B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2016/065499 external-priority patent/WO2017001660A1/en
Publication of JP2018524339A publication Critical patent/JP2018524339A/ja
Publication of JP2018524339A5 publication Critical patent/JP2018524339A5/ja
Priority to JP2021194493A priority Critical patent/JP7516338B2/ja
Application granted granted Critical
Publication of JP7099824B2 publication Critical patent/JP7099824B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2017567655A 2015-07-02 2016-07-01 抗菌化合物 Active JP7099824B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2021194493A JP7516338B2 (ja) 2015-07-02 2021-11-30 抗菌化合物

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
EP15174936 2015-07-02
EP15174936.3 2015-07-02
EP16174713 2016-06-16
EP16174713.4 2016-06-16
EP16174718.3 2016-06-16
EP16174718 2016-06-16
PCT/EP2016/065499 WO2017001660A1 (en) 2015-07-02 2016-07-01 Antibacterial compounds

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2021194493A Division JP7516338B2 (ja) 2015-07-02 2021-11-30 抗菌化合物

Publications (3)

Publication Number Publication Date
JP2018524339A JP2018524339A (ja) 2018-08-30
JP2018524339A5 true JP2018524339A5 (cg-RX-API-DMAC10.html) 2019-08-08
JP7099824B2 JP7099824B2 (ja) 2022-07-12

Family

ID=56289523

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2017567655A Active JP7099824B2 (ja) 2015-07-02 2016-07-01 抗菌化合物
JP2017567289A Pending JP2018519302A (ja) 2015-07-02 2016-07-01 抗菌化合物
JP2021194493A Active JP7516338B2 (ja) 2015-07-02 2021-11-30 抗菌化合物

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2017567289A Pending JP2018519302A (ja) 2015-07-02 2016-07-01 抗菌化合物
JP2021194493A Active JP7516338B2 (ja) 2015-07-02 2021-11-30 抗菌化合物

Country Status (29)

Country Link
US (6) US20180155341A1 (cg-RX-API-DMAC10.html)
EP (3) EP3316969B1 (cg-RX-API-DMAC10.html)
JP (3) JP7099824B2 (cg-RX-API-DMAC10.html)
KR (2) KR102710552B1 (cg-RX-API-DMAC10.html)
CN (3) CN107708809A (cg-RX-API-DMAC10.html)
AU (3) AU2016287478B2 (cg-RX-API-DMAC10.html)
BR (1) BR112017028318B1 (cg-RX-API-DMAC10.html)
CA (1) CA2986331A1 (cg-RX-API-DMAC10.html)
CL (1) CL2017003404A1 (cg-RX-API-DMAC10.html)
CO (1) CO2017013408A2 (cg-RX-API-DMAC10.html)
DK (1) DK3316969T3 (cg-RX-API-DMAC10.html)
EA (2) EA201890201A1 (cg-RX-API-DMAC10.html)
ES (1) ES2914681T3 (cg-RX-API-DMAC10.html)
HK (1) HK1249468A1 (cg-RX-API-DMAC10.html)
HR (1) HRP20220339T1 (cg-RX-API-DMAC10.html)
IL (2) IL256391B (cg-RX-API-DMAC10.html)
LT (1) LT3316969T (cg-RX-API-DMAC10.html)
MA (1) MA42293A (cg-RX-API-DMAC10.html)
MD (1) MD3316969T2 (cg-RX-API-DMAC10.html)
MX (2) MX386598B (cg-RX-API-DMAC10.html)
PE (1) PE20180520A1 (cg-RX-API-DMAC10.html)
PH (2) PH12017502297A1 (cg-RX-API-DMAC10.html)
PL (1) PL3316969T3 (cg-RX-API-DMAC10.html)
RS (1) RS63201B1 (cg-RX-API-DMAC10.html)
SI (1) SI3316969T1 (cg-RX-API-DMAC10.html)
SM (1) SMT202200220T1 (cg-RX-API-DMAC10.html)
UA (1) UA125171C2 (cg-RX-API-DMAC10.html)
WO (2) WO2017001660A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA201708692B (cg-RX-API-DMAC10.html)

Families Citing this family (46)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG11201701315VA (en) 2014-08-28 2017-03-30 Asceneuron Sa Glycosidase inhibitors
WO2017001660A1 (en) * 2015-07-02 2017-01-05 Janssen Sciences Ireland Uc Antibacterial compounds
JP6785252B2 (ja) 2015-07-02 2020-11-18 エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft 二環式ラクタム及びその使用方法
JP7055378B2 (ja) 2015-09-17 2022-04-18 ユニバーシティ・オブ・ノートル・ダム・デュ・ラック マイコバクテリア感染症に対して有用なベンジルアミン含有複素環化合物及び組成物
MX381953B (es) 2016-02-25 2025-03-13 Asceneuron S A Sales de derivados de piperazina obtenidas por adicion de acidos.
CN108884078A (zh) 2016-02-25 2018-11-23 阿森纽荣股份公司 糖苷酶抑制剂
AU2017222958B2 (en) 2016-02-25 2019-07-18 Asceneuron S. A. Glycosidase inhibitors
US11261183B2 (en) 2016-02-25 2022-03-01 Asceneuron Sa Sulfoximine glycosidase inhibitors
SMT202300273T1 (it) 2016-03-16 2023-09-06 Kura Oncology Inc Derivati di tieno[2,3–d]pirimidina sostituiti come inibitori di menina–mll e metodi d’uso
CA3026010A1 (en) 2016-06-16 2017-12-21 Janssen Sciences Ireland Unlimited Company Heterocyclic compounds as antibacterials
JP7349359B2 (ja) 2016-10-17 2023-09-22 エフ. ホフマン-ラ ロシュ アーゲー 二環式ピリドンラクタム及びその使用方法。
US11072607B2 (en) 2016-12-16 2021-07-27 Genentech, Inc. Inhibitors of RIP1 kinase and methods of use thereof
US20200048267A1 (en) * 2017-02-06 2020-02-13 Janssen Pharmaceutica Nv Oga inhibitor compounds
MA47676A (fr) * 2017-03-01 2021-06-02 Janssen Sciences Ireland Unlimited Co Polythérapie
EP3672959A1 (en) 2017-08-24 2020-07-01 Asceneuron SA Linear glycosidase inhibitors
EP3684361A4 (en) * 2017-09-20 2021-09-08 Kura Oncology, Inc. SUBSTITUTED INHIBITORS OF MENIN-MLL AND METHOD OF USING
WO2019079410A1 (en) 2017-10-17 2019-04-25 Vanderbilt University ANTAGONISTS OF THE MUSCARINIC RECEPTOR OF ACETYLCHOLINE M4
US11325896B2 (en) 2017-12-20 2022-05-10 Vanderbilt University Antagonists of the muscarinic acetylcholine receptor M4
RU2680972C1 (ru) * 2018-02-13 2019-03-01 Федеральное государственное бюджетное научное учреждение "Центральный научно-исследовательский институт туберкулеза" Способ определения длительности химиотерапии туберкулеза органов дыхания с множественной и широкой лекарственной устойчивостью МБТ у детей и подростков
WO2019175737A1 (en) * 2018-03-12 2019-09-19 University Of Notre Dame Du Lac Deuterated imidazopyridines
WO2019204537A1 (en) 2018-04-20 2019-10-24 Genentech, Inc. N-[4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-5,6-dihydro-4h-pyrrolo[1,2-b]pyrazol e-2-carboxamide derivatives and related compounds as rip1 kinase inhibitors for treating e.g. irritable bowel syndrome (ibs)
BR112021003022A2 (pt) 2018-08-22 2021-05-11 Asceneuron Sa sais de adição de ácido de ácido succínico ou ácido fumárico, de ácido monossuccínico, de ácido monofumárico e de adição de ácido succínico ou sal de adição de ácido fumárico, métodos para preparar um sal de adição de ácido do ácido succínico ou ácido fumárico, para tratar uma tauopatia e para inibir uma glicosidase, e, forma de dosagem oral sólida
US11731972B2 (en) 2018-08-22 2023-08-22 Asceneuron Sa Spiro compounds as glycosidase inhibitors
US12016852B2 (en) 2018-08-22 2024-06-25 Asceneuron Sa Pyrrolidine glycosidase inhibitors
WO2020039028A1 (en) 2018-08-22 2020-02-27 Asceneuron S. A. Tetrahydro-benzoazepine glycosidase inhibitors
CN109503631A (zh) * 2018-12-29 2019-03-22 中国医学科学院医药生物技术研究所 含有二氮杂螺环片段的咪唑并[1,2-a]吡啶-3-酰胺类化合物及其制备方法和应用
EP3976031A4 (en) * 2019-05-28 2023-07-12 Shionogi & Co., Ltd MEDICINAL PRODUCT INTENDED FOR THE TREATMENT OF A MYCOBACTERIAL INFECTION CHARACTERIZED BY THE COMBINATION OF A BC1 INHIBITOR WITH CLARITHROMYCIN OR AZITHROMYCIN AND CLOFAZIMINE
KR102076958B1 (ko) 2019-06-24 2020-02-13 엘티소재주식회사 헤테로고리 화합물 및 이를 이용한 유기 발광 소자
CA3149868A1 (en) 2019-09-13 2021-03-18 Jerome Emile Georges Guillemont Antibacterial compounds
CN114450288A (zh) 2019-09-30 2022-05-06 爱尔兰詹森科学公司 4-喹啉酮抗细菌化合物
US20220372033A1 (en) 2019-09-30 2022-11-24 Janssen Sciences Ireland Unlimited Company Antibacterial compounds
EP4081304B1 (en) 2019-12-27 2024-03-06 Tecnimede, Sociedade Técnico-Medicinal, SA Antibacterial quinolines
CA3211532A1 (en) 2021-03-16 2022-09-22 Janssen Sciences Ireland Unlimited Company Antibacterial compounds
AU2022236404A1 (en) 2021-03-17 2023-11-02 Janssen Sciences Ireland Unlimited Company Antibacterial compounds
JP2024509997A (ja) 2021-03-17 2024-03-05 ヤンセン・サイエンシズ・アイルランド・アンリミテッド・カンパニー 抗菌化合物
WO2022214520A1 (en) 2021-04-07 2022-10-13 Janssen Sciences Ireland Unlimited Company Antibacterial compounds
WO2022214519A1 (en) 2021-04-07 2022-10-13 Janssen Sciences Ireland Unlimited Company Antibacterial compounds
WO2023275744A1 (en) 2021-06-29 2023-01-05 TECNIMEDE - Sociedade Técnico-medicinal, SA Heterocyclic compounds for the treatment of tuberculosis
CA3234515A1 (en) 2021-10-28 2023-05-04 Jose Manuel Bartolome-Nebreda Imidazopyridine amides and related compounds for use in the treatment of bacterial infections
CN114957954B (zh) * 2022-05-16 2024-08-20 万华化学集团股份有限公司 一种用于光学透镜的热塑性树脂组合物及其制备方法和应用
CN119300832A (zh) * 2022-06-15 2025-01-10 C4医药公司 用于靶向降解smarca2的化合物
TW202409040A (zh) 2022-07-19 2024-03-01 大陸商西藏海思科製藥有限公司 作為激酶抑制劑的喹唑啉酮衍生物的製備及其用途
WO2024089170A1 (en) 2022-10-27 2024-05-02 Janssen Sciences Ireland Unlimited Company Antibacterial compounds
WO2024223859A1 (en) 2023-04-26 2024-10-31 Janssen Pharmaceutica Nv Antibacterial compounds
WO2025017047A1 (en) 2023-07-18 2025-01-23 Janssen Pharmaceutica Nv Combination products of at least three antibiotics comprising bedaquiline, pretomanid or delamanid, and a cytochrome bc1 inhibitor, and their use in the treatment of mycobacterial infections
WO2025129116A1 (en) * 2023-12-14 2025-06-19 C4 Therapeutics, Inc. Compounds for the targeted degradation of smarca2

Family Cites Families (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1046520C (zh) 1994-11-15 1999-11-17 法玛西雅厄普约翰美国公司 二环噁嗪及噻嗪噁唑烷酮抗菌剂
DE69614847T2 (de) 1995-05-11 2002-04-04 Pharmacia & Upjohn Co., Kalamazoo Spirocyclische und bicyclische diazinyl- und carbazinyloxazolidinone
ATE463482T1 (de) 2002-07-25 2010-04-15 Janssen Pharmaceutica Nv Chinolinderivate und deren verwendung als mycobakterielle inhibitoren
AR042956A1 (es) 2003-01-31 2005-07-13 Vertex Pharma Inhibidores de girasa y usos de los mismos
MA27360A1 (fr) 2004-11-23 2005-06-01 Brahim Bennani Synthese et application des spiro-isoxazolines comme agents anti-tuberculeux
CN101631786A (zh) 2006-12-20 2010-01-20 先灵公司 新颖的jnk抑制剂
CL2008001631A1 (es) * 2007-06-06 2009-01-02 Smithkline Beecham Corp Compuestos derivados de heterociclos sustituidos, con la presencia de un grupo fenoxi, inhibidores de transcriptasa inversa; composicion farmaceutica; y uso en el tratamiento de infecciones virales por vih.
TWI498115B (zh) 2007-12-27 2015-09-01 Daiichi Sankyo Co Ltd 咪唑羰基化合物
JP5613656B2 (ja) 2008-03-26 2014-10-29 グローバル、アライアンス、フォア、ティービー、ドラッグ、ディベロップメント 置換されたフェニルオキサゾリジノンと共有結合した二環式ニトロイミダゾール
US8658350B2 (en) 2008-09-22 2014-02-25 Oregon Health & Science University Methods for detecting Mycobacterium tuberculosis disease
AU2009334997A1 (en) 2008-12-30 2011-08-04 Millennium Pharmaceuticals, Inc. Heteroaryl compounds useful as Raf kinase inhibitors
BR112012010752B1 (pt) 2009-11-05 2021-07-20 University Of Notre Dame Du Lac Compostos imidazo[1,2-a]piridina
CN102869661B (zh) 2010-03-18 2015-08-05 韩国巴斯德研究所 抗感染化合物
KR102104125B1 (ko) 2011-04-21 2020-05-29 재단법인 한국파스퇴르연구소 소염 화합물
US20150011508A1 (en) 2011-09-01 2015-01-08 Irm Llc Compounds and compositions as c-kit kinase inhibitors
AU2012302042B2 (en) 2011-09-01 2016-03-31 Novartis Ag Compounds and compositions as c-kit kinase inhibitors
US9199981B2 (en) 2011-09-01 2015-12-01 Novartis Ag Compounds and compositions as C-kit kinase inhibitors
SG11201405056UA (en) * 2012-03-02 2014-09-26 Genentech Inc Amido spirocyclic amide and sulfonamide derivatives
KR101918469B1 (ko) 2012-06-04 2018-11-15 한국화학연구원 바이사이클릭 니트로이미다졸 유도체 또는 이들의 광학이성질체, 이의 약학적으로 허용가능한 염, 이의 제조방법 및 이를 유효성분으로 함유하는 약제학적 조성물
BR112015001201B1 (pt) * 2012-07-18 2022-02-22 University Of Notre Dame Du Lac Compostos anti-infecciosos 5,5-heteroaromáticos e composição
KR101650716B1 (ko) 2012-11-22 2016-08-24 한국화학연구원 바이시클릭니트로이미다졸 유도체, 이의 제조방법 및 이를 유효성분으로 함유하는 결핵의 예방 또는 치료용 약학적 조성물
HUE056198T2 (hu) * 2013-08-02 2022-02-28 Pasteur Institut Korea Fertõzés elleni vegyületek
KR101564425B1 (ko) 2013-11-26 2015-10-30 한국화학연구원 신규한 바이사이클릭 니트로이미다졸 카바메이트 화합물, 이를 제조하는 방법 및 이를 유효성분으로 함유하는 결핵 질환의 예방 또는 치료용 약제학적 조성물
CN105524058B (zh) 2014-10-21 2018-03-27 广州艾格生物科技有限公司 吡唑并[1,5‑a]吡啶类化合物及其应用
JP2017533220A (ja) 2014-11-03 2017-11-09 ザ リージェンツ オブ ザ ユニバーシティ オブ カリフォルニア 結核処置のための多剤療法
WO2017001660A1 (en) 2015-07-02 2017-01-05 Janssen Sciences Ireland Uc Antibacterial compounds
CA3026010A1 (en) 2016-06-16 2017-12-21 Janssen Sciences Ireland Unlimited Company Heterocyclic compounds as antibacterials
MX2018015657A (es) 2016-06-16 2019-03-14 Janssen Sciences Ireland Unlimited Co Compuestos heterociclico como antibacterianos.
MA47676A (fr) 2017-03-01 2021-06-02 Janssen Sciences Ireland Unlimited Co Polythérapie

Similar Documents

Publication Publication Date Title
JP2018524339A5 (cg-RX-API-DMAC10.html)
JP2018519302A5 (cg-RX-API-DMAC10.html)
JP2019518046A5 (cg-RX-API-DMAC10.html)
JP2019518050A5 (cg-RX-API-DMAC10.html)
JP2018536648A5 (cg-RX-API-DMAC10.html)
JP2008195730A5 (cg-RX-API-DMAC10.html)
JP2019094345A5 (cg-RX-API-DMAC10.html)
JP2012524053A5 (cg-RX-API-DMAC10.html)
JP2006507265A5 (cg-RX-API-DMAC10.html)
CN111836814A (zh) 稠环化合物、其制备方法及用途
JP2014500295A5 (cg-RX-API-DMAC10.html)
JP2004517099A5 (cg-RX-API-DMAC10.html)
JP2008201787A5 (cg-RX-API-DMAC10.html)
RU2007101653A (ru) Производные 1-азабицикло[3.3.1]нонанов
JP2013542267A5 (cg-RX-API-DMAC10.html)
JP2019519616A5 (cg-RX-API-DMAC10.html)
JP2019520344A5 (cg-RX-API-DMAC10.html)
JP2024539645A (ja) インテグリン阻害剤及び他の薬剤と組み合わせたその使用
RU2016104437A (ru) Соединения хинина, способ их получения и их медицинское применение
JPWO2021030556A5 (cg-RX-API-DMAC10.html)
EP2124930B1 (en) Isosorbide mononitrate derivatives for the treatment of intestinal disorders
JP2015522592A5 (cg-RX-API-DMAC10.html)
ITMI980442A1 (it) Sali nitrati di farmaci antiulcera
JPWO2019213445A5 (cg-RX-API-DMAC10.html)
JP2006516643A5 (cg-RX-API-DMAC10.html)