JP2017500338A5 - - Google Patents
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- JP2017500338A5 JP2017500338A5 JP2016541373A JP2016541373A JP2017500338A5 JP 2017500338 A5 JP2017500338 A5 JP 2017500338A5 JP 2016541373 A JP2016541373 A JP 2016541373A JP 2016541373 A JP2016541373 A JP 2016541373A JP 2017500338 A5 JP2017500338 A5 JP 2017500338A5
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- JP
- Japan
- Prior art keywords
- cancer
- compound
- formula
- methyl
- tumors
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB1322755.8 | 2013-12-20 | ||
| GBGB1322755.8A GB201322755D0 (en) | 2013-12-20 | 2013-12-20 | Bicyclic heterocycle compounds and their uses in therapy |
| GB201406986A GB201406986D0 (en) | 2014-04-17 | 2014-04-17 | Bicyclic heterocycle compounds and their uses in therapy |
| GB1406986.8 | 2014-04-17 | ||
| PCT/GB2014/053778 WO2015092420A1 (en) | 2013-12-20 | 2014-12-19 | Bicyclic heterocycle compounds and their uses in therapy |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019005876A Division JP6735369B2 (ja) | 2013-12-20 | 2019-01-17 | 二環式複素環化合物および治療におけるそれらの使用 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017500338A JP2017500338A (ja) | 2017-01-05 |
| JP2017500338A5 true JP2017500338A5 (Direct) | 2018-02-01 |
| JP6470756B2 JP6470756B2 (ja) | 2019-02-13 |
Family
ID=52134239
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016541373A Active JP6470756B2 (ja) | 2013-12-20 | 2014-12-19 | 二環式複素環化合物および治療におけるそれらの使用 |
| JP2019005876A Active JP6735369B2 (ja) | 2013-12-20 | 2019-01-17 | 二環式複素環化合物および治療におけるそれらの使用 |
| JP2020119260A Active JP7110279B2 (ja) | 2013-12-20 | 2020-07-10 | 二環式複素環化合物および治療におけるそれらの使用 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019005876A Active JP6735369B2 (ja) | 2013-12-20 | 2019-01-17 | 二環式複素環化合物および治療におけるそれらの使用 |
| JP2020119260A Active JP7110279B2 (ja) | 2013-12-20 | 2020-07-10 | 二環式複素環化合物および治療におけるそれらの使用 |
Country Status (29)
| Country | Link |
|---|---|
| US (6) | US9783538B2 (Direct) |
| EP (2) | EP3083616B1 (Direct) |
| JP (3) | JP6470756B2 (Direct) |
| KR (1) | KR102408262B1 (Direct) |
| CN (3) | CN115368356B (Direct) |
| AU (2) | AU2014369446C1 (Direct) |
| BR (2) | BR122022015241B1 (Direct) |
| CA (1) | CA2933939C (Direct) |
| CY (1) | CY1124436T1 (Direct) |
| DK (1) | DK3083616T3 (Direct) |
| ES (1) | ES2883289T3 (Direct) |
| HR (1) | HRP20211406T1 (Direct) |
| HU (1) | HUE056297T2 (Direct) |
| IL (1) | IL246239B (Direct) |
| LT (1) | LT3083616T (Direct) |
| MX (1) | MX380469B (Direct) |
| MY (2) | MY186311A (Direct) |
| NZ (2) | NZ719905A (Direct) |
| PH (1) | PH12016501139A1 (Direct) |
| PL (1) | PL3083616T3 (Direct) |
| PT (1) | PT3083616T (Direct) |
| RS (1) | RS62301B1 (Direct) |
| RU (1) | RU2696310C1 (Direct) |
| SA (1) | SA516371360B1 (Direct) |
| SG (2) | SG11201604795RA (Direct) |
| SI (1) | SI3083616T1 (Direct) |
| SM (1) | SMT202100497T1 (Direct) |
| TW (1) | TWI649319B (Direct) |
| WO (1) | WO2015092420A1 (Direct) |
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| CN120247907A (zh) | 2020-05-04 | 2025-07-04 | 大塚制药株式会社 | Iap拮抗剂化合物和中间体及其合成方法 |
| EP4146617B8 (en) | 2020-05-04 | 2025-10-15 | Taiho Pharmaceutical Co., Ltd. | Methods for synthesizing anhydrous lactic acid |
| WO2023168394A1 (en) | 2022-03-04 | 2023-09-07 | Otsuka Pharmaceutical Co., Ltd. | Methods of treating cancer with iap antagonist compounds and combination therapies |
| KR20250053870A (ko) | 2022-08-31 | 2025-04-22 | 다이호야쿠힌고교 가부시키가이샤 | 톨리나판트, 세다주리딘 및 데시타빈을 사용한 t 세포 림프종의 치료를 위한 조합 요법 |
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