JP2016504330A5 - - Google Patents

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Publication number
JP2016504330A5
JP2016504330A5 JP2015548841A JP2015548841A JP2016504330A5 JP 2016504330 A5 JP2016504330 A5 JP 2016504330A5 JP 2015548841 A JP2015548841 A JP 2015548841A JP 2015548841 A JP2015548841 A JP 2015548841A JP 2016504330 A5 JP2016504330 A5 JP 2016504330A5
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JP
Japan
Prior art keywords
group
compound
range
pharmaceutically acceptable
hydrogen
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JP2015548841A
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English (en)
Japanese (ja)
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JP6533466B2 (ja
JP2016504330A (ja
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Priority claimed from PCT/IB2013/061090 external-priority patent/WO2014097178A1/en
Publication of JP2016504330A publication Critical patent/JP2016504330A/ja
Publication of JP2016504330A5 publication Critical patent/JP2016504330A5/ja
Application granted granted Critical
Publication of JP6533466B2 publication Critical patent/JP6533466B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2015548841A 2012-12-18 2013-12-18 抗菌性化合物、その合成およびその適用 Expired - Fee Related JP6533466B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN5299CH2012 2012-12-18
IN5299/CHE/2012 2012-12-18
PCT/IB2013/061090 WO2014097178A1 (en) 2012-12-18 2013-12-18 Antimicrobial compounds, their synthesis and applications thereof

Publications (3)

Publication Number Publication Date
JP2016504330A JP2016504330A (ja) 2016-02-12
JP2016504330A5 true JP2016504330A5 (https=) 2017-01-26
JP6533466B2 JP6533466B2 (ja) 2019-06-19

Family

ID=54148251

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015548841A Expired - Fee Related JP6533466B2 (ja) 2012-12-18 2013-12-18 抗菌性化合物、その合成およびその適用

Country Status (9)

Country Link
US (1) US9783490B2 (https=)
EP (1) EP2934563B1 (https=)
JP (1) JP6533466B2 (https=)
CN (1) CN104981249B (https=)
AU (1) AU2013365769B2 (https=)
BR (1) BR112015014391B1 (https=)
CA (1) CA2894202A1 (https=)
HK (1) HK1210437A1 (https=)
WO (1) WO2014097178A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105566149B (zh) * 2016-03-02 2017-05-24 郑州大学 具有抗菌活性的查尔酮阳离子抗菌肽模拟物及其制备方法
CN106995384B (zh) * 2017-04-21 2018-12-11 郑州大学 具有抗菌活性的二烷基阳离子两亲性抗菌肽模拟物及其制备方法
EP3724216A1 (en) 2017-12-15 2020-10-21 Dana Farber Cancer Institute, Inc. Stabilized peptide-mediated targeted protein degradation

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK0610487T3 (da) 1992-09-03 2000-05-15 Boehringer Ingelheim Pharma Nye aminosyrederivater, fremgangsmåde til deres fremstilling og farmaceutiske præparater indeholdende disse forbindelser
US5654451B1 (en) * 1993-01-14 2000-02-22 Magainin Pharma Amino acids and peptides having modified c-terminals and modified n-terminals
JPH09507846A (ja) * 1993-12-30 1997-08-12 スミスクライン・ビーチャム・コーポレイション フェニルメチルヘキサンアミドおよびその使用
US5663148A (en) 1994-07-12 1997-09-02 Abbott Laboratories Anaphylatoxin receptor ligands containing lipophilic residues
US6071890A (en) * 1994-12-09 2000-06-06 Genzyme Corporation Organ-specific targeting of cationic amphiphile/DNA complexes for gene therapy
JP3338452B2 (ja) 1995-12-12 2002-10-28 大鵬薬品工業株式会社 エポキシコハク酸アミド誘導体又はその塩及びこれを含有する医薬
CA2217550A1 (en) * 1996-10-22 1998-04-22 F. Hoffmann-La Roche Ag Cationic lipids for gene therapy
WO1999031052A1 (fr) * 1997-12-12 1999-06-24 Fuji Yakuhin Kogyo Kabushiki Kaisha Nouveaux inhibiteurs de metalloproteinases
AU2180201A (en) * 1999-11-30 2001-06-12 Aventis Pharma S.A. Hydroxamic acid macrocyclic derivatives, preparation method and compositions containing same
JP2002161084A (ja) * 2000-11-28 2002-06-04 Sumitomo Pharmaceut Co Ltd 複素環誘導体
US7393836B2 (en) 2004-07-06 2008-07-01 Boehringer Ingelheim International Gmbh D-xylopyranosyl-substituted phenyl derivatives, medicaments containing such compounds, their use and process for their manufacture
GB0512751D0 (en) * 2005-06-22 2005-07-27 Glaxo Group Ltd New adjuvant
EP2019819A4 (en) * 2006-05-09 2011-01-19 Neobiotics Ab INNOVATIVE PEPTIDE DERIVATIVES AS ANTIMICROBIAL AGENTS FOR THE TREATMENT OF INJURIES
SG175573A1 (en) * 2006-10-04 2011-11-28 Inimex Pharmaceuticals Inc Novel peptides for treating and preventing immune-related disorders, including treating and preventing infection by modulating innate immunity
JP2010512417A (ja) * 2006-12-11 2010-04-22 ワイス エルエルシー イオンチャネルモジュレータ−
CN102757477B (zh) * 2011-04-27 2014-09-03 首都医科大学 烯丙基半胱氨酰氨基酸甲酯衍生物及其合成方法和应用
DK2709619T3 (en) * 2011-05-16 2018-01-15 Cellceutix Corp RELATIONSHIPS FOR USING THE TREATMENT OF MUCOSITIS

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