JP2015531365A5 - - Google Patents

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Publication number
JP2015531365A5
JP2015531365A5 JP2015533717A JP2015533717A JP2015531365A5 JP 2015531365 A5 JP2015531365 A5 JP 2015531365A5 JP 2015533717 A JP2015533717 A JP 2015533717A JP 2015533717 A JP2015533717 A JP 2015533717A JP 2015531365 A5 JP2015531365 A5 JP 2015531365A5
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JP
Japan
Prior art keywords
solid dispersion
thienotriazolodiazepine compound
formula
concentration
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2015533717A
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English (en)
Japanese (ja)
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JP2015531365A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/IB2013/003026 external-priority patent/WO2014068402A2/en
Publication of JP2015531365A publication Critical patent/JP2015531365A/ja
Publication of JP2015531365A5 publication Critical patent/JP2015531365A5/ja
Ceased legal-status Critical Current

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JP2015533717A 2012-09-28 2013-09-27 チエノトリアゾロジアゼピン化合物を含む医薬製剤 Ceased JP2015531365A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201261707465P 2012-09-28 2012-09-28
US61/707,465 2012-09-28
US201361782882P 2013-03-14 2013-03-14
US61/782,882 2013-03-14
US201361831811P 2013-06-06 2013-06-06
US61/831,811 2013-06-06
PCT/IB2013/003026 WO2014068402A2 (en) 2012-09-28 2013-09-27 Pharmaceutical formulation containing thienotriazolodiazepine compounds

Publications (2)

Publication Number Publication Date
JP2015531365A JP2015531365A (ja) 2015-11-02
JP2015531365A5 true JP2015531365A5 (https=) 2018-04-12

Family

ID=50475880

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015533717A Ceased JP2015531365A (ja) 2012-09-28 2013-09-27 チエノトリアゾロジアゼピン化合物を含む医薬製剤

Country Status (13)

Country Link
US (1) US20140107107A1 (https=)
EP (1) EP2900221B1 (https=)
JP (1) JP2015531365A (https=)
KR (1) KR20150100613A (https=)
CN (1) CN104968334B (https=)
AU (1) AU2013340483B2 (https=)
BR (1) BR112015006537A2 (https=)
CA (1) CA2885944A1 (https=)
HK (2) HK1210434A1 (https=)
IN (1) IN2015DN03135A (https=)
MX (1) MX2015003771A (https=)
RU (1) RU2015115634A (https=)
WO (1) WO2014068402A2 (https=)

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WO2015018522A1 (en) * 2013-08-06 2015-02-12 Oncoethix Sa Bet-bromodomain inhibitor shows synergism with several anti-cancer agents in pre-clinical models of diffuse large b-cell lymphoma (dlbcl)
RU2016122654A (ru) 2013-11-08 2017-12-14 Дана-Фарбер Кэнсер Инститьют, Инк. Комбинированная терапия злокачественной опухоли с использованием ингибиторов бромодоменового и экстратерминального (вет) белка
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TWI672141B (zh) 2014-02-20 2019-09-21 美商醫科泰生技 投予ros1突變癌細胞之分子
JP2017506666A (ja) 2014-02-28 2017-03-09 テンシャ セラピューティクス,インコーポレイテッド 高インスリン血症に関連した症状の処置
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WO2015168587A1 (en) * 2014-05-02 2015-11-05 Oncoethix Sa Method of treating resistant multiple myeloma and mantle cell lymphoma using thienotriazolodiazepine compounds
WO2015169953A1 (en) * 2014-05-08 2015-11-12 Oncoethix Gmbh Method of treating glioma using thienotriazolodiazepine compounds
AU2015257658A1 (en) * 2014-05-08 2016-11-10 Oncoethix Gmbh Method of treating triple-negative breast cancer using thienotriazolodiazepine compounds
BR112016029012A2 (pt) 2014-06-13 2017-08-22 Oncoethix Gmbh método de tratamento de câncer de pulmão de células não pequenas e/ou câncer de pulmão de células pequenas usando compostos de tienotriazolodiazepina
KR20170037670A (ko) * 2014-08-19 2017-04-04 온코에틱스 게엠베하 티에노트리아졸로디아제핀 화합물을 사용한 림프종의 치료 방법
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JP6599979B2 (ja) 2014-09-15 2019-10-30 インサイト・コーポレイション Betタンパク質阻害剤として用いるための三環式複素環化合物
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CN107207471B (zh) 2014-12-02 2020-06-26 伊尼塔公司 用于治疗神经母细胞瘤的组合
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CN111225662B (zh) * 2017-10-17 2022-11-22 伊尼塔公司 药物组合物和剂型
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JP7812785B2 (ja) * 2019-09-18 2026-02-10 ブリストル-マイヤーズ スクイブ カンパニー Tyk2阻害薬の剤形
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DK4245298T3 (en) * 2020-12-18 2026-03-30 Daewoong Pharmaceutical Co Ltd Hidtil ukendt formulering til oral administration, som omfatter 1-(5-(2,4-difluorphenyl)-1-((3-fluorphenyl)sulfonyl)-4-methoxy-1h-pyrrol-3-yl)-n-methylmethanamin
CN116098870B (zh) * 2023-04-10 2023-07-25 上海赛默罗生物科技有限公司 α5-GABAA受体调节剂的固体分散体及其制备方法

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