JP2014520898A5 - - Google Patents

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JP2014520898A5
JP2014520898A5 JP2014521840A JP2014521840A JP2014520898A5 JP 2014520898 A5 JP2014520898 A5 JP 2014520898A5 JP 2014521840 A JP2014521840 A JP 2014521840A JP 2014521840 A JP2014521840 A JP 2014521840A JP 2014520898 A5 JP2014520898 A5 JP 2014520898A5
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pharmaceutically acceptable
tautomer
stereoisomer
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JP2014521840A
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JP6105578B2 (ja
JP2014520898A (ja
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Priority claimed from PCT/US2012/047685 external-priority patent/WO2013013188A1/en
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JP2014521840A 2011-07-21 2012-07-20 複素環式プロテインキナーゼ阻害剤 Active JP6105578B2 (ja)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US201161510207P 2011-07-21 2011-07-21
US201161632834P 2011-07-21 2011-07-21
US61/632,834 2011-07-21
US61/510,207 2011-07-21
US201261632826P 2012-03-01 2012-03-01
US61/632,826 2012-03-01
US201261608028P 2012-03-07 2012-03-07
US61/608,028 2012-03-07
PCT/US2012/047685 WO2013013188A1 (en) 2011-07-21 2012-07-20 Heterocyclic protein kinase inhibitors

Publications (3)

Publication Number Publication Date
JP2014520898A JP2014520898A (ja) 2014-08-25
JP2014520898A5 true JP2014520898A5 (OSRAM) 2015-09-10
JP6105578B2 JP6105578B2 (ja) 2017-03-29

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JP2014521840A Active JP6105578B2 (ja) 2011-07-21 2012-07-20 複素環式プロテインキナーゼ阻害剤

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US (7) US9416132B2 (OSRAM)
EP (3) EP3409278B8 (OSRAM)
JP (1) JP6105578B2 (OSRAM)
CY (1) CY1123626T1 (OSRAM)
DK (2) DK2734205T3 (OSRAM)
ES (2) ES2834093T3 (OSRAM)
HU (1) HUE052198T2 (OSRAM)
PL (1) PL3409278T3 (OSRAM)
PT (1) PT3409278T (OSRAM)
WO (1) WO2013013188A1 (OSRAM)

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BR112022020114A2 (pt) * 2020-04-15 2022-11-29 Pyramid Biosciences Inc Métodos para preparar inibidores do receptor tirosina quinase
CN112430632B (zh) * 2020-11-18 2022-09-13 上海合全药物研发有限公司 2-((反式)-4-氨基环己烷基)异丙醇的制备方法
WO2022166860A1 (zh) 2021-02-08 2022-08-11 杭州邦顺制药有限公司 Pim激酶抑制剂
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CN116262753A (zh) * 2021-12-13 2023-06-16 杭州邦顺制药有限公司 一种新颖的pim激酶抑制剂
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