JP2014500252A5 - - Google Patents

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Publication number
JP2014500252A5
JP2014500252A5 JP2013538052A JP2013538052A JP2014500252A5 JP 2014500252 A5 JP2014500252 A5 JP 2014500252A5 JP 2013538052 A JP2013538052 A JP 2013538052A JP 2013538052 A JP2013538052 A JP 2013538052A JP 2014500252 A5 JP2014500252 A5 JP 2014500252A5
Authority
JP
Japan
Prior art keywords
pyridin
methyl
ylamino
phenoxy
methylsulfonyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2013538052A
Other languages
English (en)
Japanese (ja)
Other versions
JP6038037B2 (ja
JP2014500252A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2011/082004 external-priority patent/WO2012062210A1/en
Publication of JP2014500252A publication Critical patent/JP2014500252A/ja
Publication of JP2014500252A5 publication Critical patent/JP2014500252A5/ja
Application granted granted Critical
Publication of JP6038037B2 publication Critical patent/JP6038037B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2013538052A 2010-11-09 2011-11-09 キナーゼ活性を増加させるための化合物とその応用 Expired - Fee Related JP6038037B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201010535640 2010-11-09
CN201010535640.4 2010-11-09
PCT/CN2011/082004 WO2012062210A1 (en) 2010-11-09 2011-11-09 Compound for increasing kinase active and application thereof

Publications (3)

Publication Number Publication Date
JP2014500252A JP2014500252A (ja) 2014-01-09
JP2014500252A5 true JP2014500252A5 (enExample) 2014-12-25
JP6038037B2 JP6038037B2 (ja) 2016-12-07

Family

ID=46050413

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013538052A Expired - Fee Related JP6038037B2 (ja) 2010-11-09 2011-11-09 キナーゼ活性を増加させるための化合物とその応用

Country Status (8)

Country Link
US (1) US9409900B2 (enExample)
EP (1) EP2638036B1 (enExample)
JP (1) JP6038037B2 (enExample)
KR (2) KR101643721B1 (enExample)
CN (1) CN103502244B (enExample)
AU (1) AU2011328673B2 (enExample)
SG (2) SG190784A1 (enExample)
WO (1) WO2012062210A1 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR127073A1 (es) 2021-09-17 2023-12-13 Flagship Pioneering Innovations Vi Llc Composiciones y métodos para producir polirribonucleótidos circulares

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3632042A1 (de) 1986-03-08 1987-09-10 Bayer Ag Diarylsulfidderivate
JPS62212378A (ja) * 1986-03-08 1987-09-18 バイエル・アクチエンゲゼルシヤフト ジアリ−ルスルフイド誘導体
US6719520B2 (en) 1998-10-08 2004-04-13 Smithkline Beecham Corporation Method and compounds
JP2002527419A (ja) * 1998-10-08 2002-08-27 スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー Gsk−3阻害物質としてのピロール−2,5−ジオン類
UA71945C2 (en) * 1999-01-27 2005-01-17 Pfizer Prod Inc Substituted bicyclic derivatives being used as anticancer agents
EP1127882A1 (en) * 2000-01-25 2001-08-29 Pfizer Products Inc. Tetrazole compounds as thyroid receptor ligands
GB0008264D0 (en) * 2000-04-04 2000-05-24 Smithkline Beecham Plc Novel method and compounds
JP3598994B2 (ja) * 2000-07-10 2004-12-08 セイコーエプソン株式会社 電気光学装置の製造方法
ES2263743T3 (es) * 2001-04-13 2006-12-16 Pfizer Products Inc. Derivados de 4-aminopiridopirimidina sustituidos con un grupo biciclico.
WO2003026665A1 (en) * 2001-09-26 2003-04-03 Bayer Pharmaceuticals Corporation 2-phenylamino-4-(5-pyrazolylamino)-pyrimidine derivatives as kinase inhibitors, in particular, src kinase inhibitors
DE10153396A1 (de) * 2001-11-01 2003-05-28 Siemens Ag Einrichtung zur Ansteuerung einer elektrischen Kraftstoffpumpe
KR100768609B1 (ko) * 2003-07-09 2007-10-18 에프. 호프만-라 로슈 아게 티오페닐아미노이미다졸린
BRPI0517232A (pt) * 2004-11-02 2008-10-07 Banyu Pharma Co Ltd composto ou um sal farmaceuticamente aceitável do mesmo, composição farmacêutica, ativador da glicocinase, e, agentes terapêuticos e/ou profiláticos para diabetes e para obesidade
US20120052061A1 (en) * 2007-09-24 2012-03-01 Tragara Pharmaceuticals Inc. Therapies for treating cancer using combinations of cox-2 inhibitors and anti-her2(erbb2) antibodies or combinations of cox-2 inhibitors and her2(erbb2) receptor tyrosine kinase inhibitors
WO2010090875A1 (en) * 2009-01-21 2010-08-12 Rigel Pharmaceuticals, Inc. Derivatives of n2-(3-pyridil or phenyl)-n4-(4-piperidyl)-2,4-pyrimidinediamine useful in the treatment of inflammatory, autoimmune or proliferative diseases

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