JP2013544811A5 - - Google Patents

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Publication number
JP2013544811A5
JP2013544811A5 JP2013537774A JP2013537774A JP2013544811A5 JP 2013544811 A5 JP2013544811 A5 JP 2013544811A5 JP 2013537774 A JP2013537774 A JP 2013537774A JP 2013537774 A JP2013537774 A JP 2013537774A JP 2013544811 A5 JP2013544811 A5 JP 2013544811A5
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JP
Japan
Prior art keywords
phenyl
isoxazol
trifluoromethyl
chroman
oxadiazol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2013537774A
Other languages
English (en)
Japanese (ja)
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JP2013544811A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2011/058891 external-priority patent/WO2012061459A1/en
Publication of JP2013544811A publication Critical patent/JP2013544811A/ja
Publication of JP2013544811A5 publication Critical patent/JP2013544811A5/ja
Ceased legal-status Critical Current

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JP2013537774A 2010-11-03 2011-11-02 自己免疫疾患および血管疾患の治療用のs1p1アゴニストとしての複素環式化合物 Ceased JP2013544811A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US40968210P 2010-11-03 2010-11-03
US61/409,682 2010-11-03
PCT/US2011/058891 WO2012061459A1 (en) 2010-11-03 2011-11-02 Heterocyclic compounds as s1p1 agonists for the treatment of autoimmune and vascular diseases

Publications (2)

Publication Number Publication Date
JP2013544811A JP2013544811A (ja) 2013-12-19
JP2013544811A5 true JP2013544811A5 (enExample) 2014-11-06

Family

ID=44983720

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013537774A Ceased JP2013544811A (ja) 2010-11-03 2011-11-02 自己免疫疾患および血管疾患の治療用のs1p1アゴニストとしての複素環式化合物

Country Status (6)

Country Link
US (1) US8629282B2 (enExample)
EP (1) EP2635573B1 (enExample)
JP (1) JP2013544811A (enExample)
CN (1) CN103298807A (enExample)
ES (1) ES2525298T3 (enExample)
WO (1) WO2012061459A1 (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2539256T3 (es) 2010-07-20 2015-06-29 Bristol-Myers Squibb Company Compuestos de 3-fenil-1,2,4-oxadiazol sustituidos
JP5869579B2 (ja) 2010-09-24 2016-02-24 ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company 置換オキサジアゾール化合物およびそれらのs1p1アゴニストとしての使用
TWI613182B (zh) 2013-02-21 2018-02-01 必治妥美雅史谷比公司 雙環化合物
TWI689487B (zh) 2014-08-20 2020-04-01 美商必治妥美雅史谷比公司 經取代雙環化合物
JP6883882B2 (ja) * 2016-07-22 2021-06-09 シージャーズォアン サガシティ ニュー ドラッグ デベロップメント カンパニー リミテッド S1p1アゴニスト及びその応用
IL271149B2 (en) 2017-06-14 2024-05-01 Trevena Inc Compounds for modulating s1p1 activity and methods of using the same
CA3088460A1 (en) 2018-01-18 2019-07-25 Shijiazhuang Sagacity New Drug Development Company, Ltd. Crystal and salt forms of tricyclic compound and preparation process thereof
EP4061352A4 (en) * 2019-11-19 2024-02-28 Trevena, Inc. Compounds and methods of preparing compounds s1p1 modulators
EP4061358B1 (en) * 2019-11-20 2025-05-28 Arena Pharmaceuticals, Inc. Etrasimod for use in the treatment of eosinophilic esophagitis

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ES2539256T3 (es) 2010-07-20 2015-06-29 Bristol-Myers Squibb Company Compuestos de 3-fenil-1,2,4-oxadiazol sustituidos
JP5869579B2 (ja) 2010-09-24 2016-02-24 ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company 置換オキサジアゾール化合物およびそれらのs1p1アゴニストとしての使用

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