JP2013544796A5 - - Google Patents
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- Publication number
- JP2013544796A5 JP2013544796A5 JP2013534440A JP2013534440A JP2013544796A5 JP 2013544796 A5 JP2013544796 A5 JP 2013544796A5 JP 2013534440 A JP2013534440 A JP 2013534440A JP 2013534440 A JP2013534440 A JP 2013534440A JP 2013544796 A5 JP2013544796 A5 JP 2013544796A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- phenyl
- group
- dioxaspiro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 CN(C)C(CC#O)(CCC1)CC1(*)*=C Chemical compound CN(C)C(CC#O)(CCC1)CC1(*)*=C 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IBPCT/IB2010/054747 | 2010-10-20 | ||
| IB2010054747 | 2010-10-20 | ||
| PCT/IB2011/054660 WO2012052939A2 (en) | 2010-10-20 | 2011-10-19 | Preparation of bicyclo[2.2.2]octan-2-one compounds |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013544796A JP2013544796A (ja) | 2013-12-19 |
| JP2013544796A5 true JP2013544796A5 (enExample) | 2014-12-04 |
| JP5909237B2 JP5909237B2 (ja) | 2016-04-26 |
Family
ID=45757740
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013534440A Expired - Fee Related JP5909237B2 (ja) | 2010-10-20 | 2011-10-19 | ビシクロ［２．２．２］オクタン−２−オン化合物の製造 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US9296673B2 (enExample) |
| EP (1) | EP2630111B1 (enExample) |
| JP (1) | JP5909237B2 (enExample) |
| KR (1) | KR101876594B1 (enExample) |
| CN (1) | CN103168019B (enExample) |
| CA (1) | CA2813131C (enExample) |
| DK (1) | DK2630111T3 (enExample) |
| ES (1) | ES2536897T3 (enExample) |
| HU (1) | HUE025195T2 (enExample) |
| IL (1) | IL225763A (enExample) |
| MX (1) | MX2013004427A (enExample) |
| TW (2) | TWI511949B (enExample) |
| WO (1) | WO2012052939A2 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2692656T3 (es) | 2010-10-20 | 2018-12-04 | Idorsia Pharmaceuticals Ltd | Preparación diastereoselectiva de los compuestos de biciclo[2.2.2]octan-2-ona |
| US9296673B2 (en) * | 2010-10-20 | 2016-03-29 | Actelion Pharmaceuticals Ltd. | Preparation of bicyclo[2.2.2]octan-2-one compounds |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3046106A1 (de) * | 1980-12-06 | 1982-07-15 | Studiengesellschaft Kohle mbH, 4330 Mülheim | Optisch reine bicyclo(2.2.2)oct-5-en-2.one, verfahren zu ihrer herstellung und ihre verwendung |
| JP3439255B2 (ja) * | 1994-03-31 | 2003-08-25 | 長瀬産業株式会社 | 不斉マイケル反応を触媒する金属錯体 |
| AR066148A1 (es) * | 2007-04-27 | 2009-07-29 | Actelion Pharmaceuticals Ltd | Derivados puenteados de ciclohexeno bloqueadores del canal de calcio |
| KR101364909B1 (ko) | 2008-04-25 | 2014-02-21 | 액테리온 파마슈티칼 리미티드 | 칼슘 채널 차단제로서의 벤지미다졸 유도체 |
| ES2692656T3 (es) | 2010-10-20 | 2018-12-04 | Idorsia Pharmaceuticals Ltd | Preparación diastereoselectiva de los compuestos de biciclo[2.2.2]octan-2-ona |
| US9296673B2 (en) * | 2010-10-20 | 2016-03-29 | Actelion Pharmaceuticals Ltd. | Preparation of bicyclo[2.2.2]octan-2-one compounds |
-
2011
- 2011-10-19 US US13/880,520 patent/US9296673B2/en not_active Expired - Fee Related
- 2011-10-19 WO PCT/IB2011/054660 patent/WO2012052939A2/en not_active Ceased
- 2011-10-19 HU HUE11820867A patent/HUE025195T2/en unknown
- 2011-10-19 TW TW100137956A patent/TWI511949B/zh not_active IP Right Cessation
- 2011-10-19 DK DK11820867.7T patent/DK2630111T3/en active
- 2011-10-19 JP JP2013534440A patent/JP5909237B2/ja not_active Expired - Fee Related
- 2011-10-19 EP EP11820867.7A patent/EP2630111B1/en active Active
- 2011-10-19 TW TW100137955A patent/TWI551583B/zh not_active IP Right Cessation
- 2011-10-19 CA CA2813131A patent/CA2813131C/en active Active
- 2011-10-19 KR KR1020137012606A patent/KR101876594B1/ko not_active Expired - Fee Related
- 2011-10-19 CN CN201180050144.2A patent/CN103168019B/zh not_active Expired - Fee Related
- 2011-10-19 MX MX2013004427A patent/MX2013004427A/es active IP Right Grant
- 2011-10-19 ES ES11820867.7T patent/ES2536897T3/es active Active
-
2013
- 2013-04-15 IL IL225763A patent/IL225763A/en active IP Right Grant
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