MX2013004427A - Preparacion de los compuestos de biciclo [2.2.2] octan-2-ona. - Google Patents

Preparacion de los compuestos de biciclo [2.2.2] octan-2-ona.

Info

Publication number
MX2013004427A
MX2013004427A MX2013004427A MX2013004427A MX2013004427A MX 2013004427 A MX2013004427 A MX 2013004427A MX 2013004427 A MX2013004427 A MX 2013004427A MX 2013004427 A MX2013004427 A MX 2013004427A MX 2013004427 A MX2013004427 A MX 2013004427A
Authority
MX
Mexico
Prior art keywords
compounds
formula
present
octan
preparation
Prior art date
Application number
MX2013004427A
Other languages
English (en)
Spanish (es)
Inventor
Stefan Abele
Jacques-Alexis Funel
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of MX2013004427A publication Critical patent/MX2013004427A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/385Saturated compounds containing a keto group being part of a ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C29/00Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
    • C07C29/132Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group
    • C07C29/136Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group of >C=O containing groups, e.g. —COOH
    • C07C29/147Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group of >C=O containing groups, e.g. —COOH of carboxylic acids or derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/63Esters of sulfonic acids
    • C07C309/64Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms
    • C07C309/65Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms of a saturated carbon skeleton
    • C07C309/66Methanesulfonates
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/27Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation
    • C07C45/29Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation of hydroxy groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/27Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation
    • C07C45/30Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation with halogen containing compounds, e.g. hypohalogenation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/51Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by pyrolysis, rearrangement or decomposition
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/56Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds
    • C07C45/57Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with oxygen as the only heteroatom
    • C07C45/59Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with oxygen as the only heteroatom in five-membered rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/65Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by splitting-off hydrogen atoms or functional groups; by hydrogenolysis of functional groups
    • C07C45/66Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by splitting-off hydrogen atoms or functional groups; by hydrogenolysis of functional groups by dehydration
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/78Separation; Purification; Stabilisation; Use of additives
    • C07C45/81Separation; Purification; Stabilisation; Use of additives by change in the physical state, e.g. crystallisation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00Preparation of carboxylic acid esters
    • C07C67/30Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C07C67/313Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by introduction of doubly bound oxygen containing functional groups, e.g. carboxyl groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D317/00Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/72Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 spiro-condensed with carbocyclic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/12Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14The ring being saturated
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00Systems containing two condensed rings
    • C07C2602/36Systems containing two condensed rings the rings having more than two atoms in common
    • C07C2602/44Systems containing two condensed rings the rings having more than two atoms in common the bicyclo ring system containing eight carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
MX2013004427A 2010-10-20 2011-10-19 Preparacion de los compuestos de biciclo [2.2.2] octan-2-ona. MX2013004427A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IB2010054747 2010-10-20
PCT/IB2011/054660 WO2012052939A2 (en) 2010-10-20 2011-10-19 Preparation of bicyclo[2.2.2]octan-2-one compounds

Publications (1)

Publication Number Publication Date
MX2013004427A true MX2013004427A (es) 2013-07-17

Family

ID=45757740

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2013004427A MX2013004427A (es) 2010-10-20 2011-10-19 Preparacion de los compuestos de biciclo [2.2.2] octan-2-ona.

Country Status (13)

Country Link
US (1) US9296673B2 (enExample)
EP (1) EP2630111B1 (enExample)
JP (1) JP5909237B2 (enExample)
KR (1) KR101876594B1 (enExample)
CN (1) CN103168019B (enExample)
CA (1) CA2813131C (enExample)
DK (1) DK2630111T3 (enExample)
ES (1) ES2536897T3 (enExample)
HU (1) HUE025195T2 (enExample)
IL (1) IL225763A (enExample)
MX (1) MX2013004427A (enExample)
TW (2) TWI511949B (enExample)
WO (1) WO2012052939A2 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2692656T3 (es) 2010-10-20 2018-12-04 Idorsia Pharmaceuticals Ltd Preparación diastereoselectiva de los compuestos de biciclo[2.2.2]octan-2-ona
US9296673B2 (en) * 2010-10-20 2016-03-29 Actelion Pharmaceuticals Ltd. Preparation of bicyclo[2.2.2]octan-2-one compounds

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3046106A1 (de) * 1980-12-06 1982-07-15 Studiengesellschaft Kohle mbH, 4330 Mülheim Optisch reine bicyclo(2.2.2)oct-5-en-2.one, verfahren zu ihrer herstellung und ihre verwendung
JP3439255B2 (ja) * 1994-03-31 2003-08-25 長瀬産業株式会社 不斉マイケル反応を触媒する金属錯体
AR066148A1 (es) * 2007-04-27 2009-07-29 Actelion Pharmaceuticals Ltd Derivados puenteados de ciclohexeno bloqueadores del canal de calcio
KR101364909B1 (ko) 2008-04-25 2014-02-21 액테리온 파마슈티칼 리미티드 칼슘 채널 차단제로서의 벤지미다졸 유도체
ES2692656T3 (es) 2010-10-20 2018-12-04 Idorsia Pharmaceuticals Ltd Preparación diastereoselectiva de los compuestos de biciclo[2.2.2]octan-2-ona
US9296673B2 (en) * 2010-10-20 2016-03-29 Actelion Pharmaceuticals Ltd. Preparation of bicyclo[2.2.2]octan-2-one compounds

Also Published As

Publication number Publication date
JP2013544796A (ja) 2013-12-19
KR101876594B1 (ko) 2018-08-02
ES2536897T3 (es) 2015-05-29
TW201217324A (en) 2012-05-01
TWI551583B (zh) 2016-10-01
CN103168019B (zh) 2015-05-27
DK2630111T3 (en) 2015-04-20
WO2012052939A2 (en) 2012-04-26
EP2630111B1 (en) 2015-02-25
EP2630111A2 (en) 2013-08-28
TWI511949B (zh) 2015-12-11
JP5909237B2 (ja) 2016-04-26
CA2813131C (en) 2019-02-12
US9296673B2 (en) 2016-03-29
CN103168019A (zh) 2013-06-19
WO2012052939A3 (en) 2012-06-21
HUE025195T2 (en) 2016-02-29
IL225763A0 (en) 2013-06-27
IL225763A (en) 2016-04-21
US20130211104A1 (en) 2013-08-15
TW201217325A (en) 2012-05-01
KR20130138268A (ko) 2013-12-18
CA2813131A1 (en) 2012-04-26

Similar Documents

Publication Publication Date Title
WO2012049666A3 (en) Data word analysis by spectroscopy
Parella et al. Long-range proton–carbon coupling constants: NMR methods and applications
EA201490932A1 (ru) Связывающие молекулы в отношении всма и cd3
WO2007109211A3 (en) 1-oxo-isoindoline compounds for the treatment of spinal muscular atrophy and other uses
SG194233A1 (en) Identification of polynucleotides associated with a sample
MY167795A (en) Tdp-43 specefic binding molecules
NO20083153L (no) Kjemiske forbindelser
EA201070256A1 (ru) Способ и промежуточные соединения для получения ингибиторов интегразы
EP2546654A3 (en) Heroin detection by raman spectroscopy from impure compositions comprising an interfering fluorescent contaminant
MX349925B (es) Un método y aparato para probar materiales de circulación perdidos para formaciones subterráneas.
TW201206878A (en) A method of producing ingenol-3-angelate
EP2668659A2 (en) Timing device and method in a mass spectrometer
WO2009149072A3 (en) Identification of body fluids using raman spectroscopy
WO2010144151A3 (en) Single-molecule real-time analysis of protein synthesis
Muthu et al. Vibrational and UV spectra, first order hyperpolarizability, NBO and HOMO–LUMO analysis of 4-chloro-N-(2-methyl-2, 3-dihydroindol-1-yl)-3-sulfamoyl-benzamide
MX2013004427A (es) Preparacion de los compuestos de biciclo [2.2.2] octan-2-ona.
WO2011081296A3 (ko) 검색 결과 제공 시스템 및 방법
WO2012168344A8 (en) BINDING COMPOUNDS TO HUMAN β1-ADRENORECEPTOR (β1-AR) AND THEIR USE IN THE MEASUREMENT OF AUTO-ANTI-βA1-AR ANTIBODIES
PH12014502846A1 (en) Colorant compound derived from genipa americana genipin and glycine
EA201270390A1 (ru) 1,2,4-триазин, который может быть использован в качестве ускорителя вулканизации, и способ его получения
Liu et al. A selective colorimetric sensor for Cu2+ in aqueous solution
WO2009108949A3 (en) Cold shock protein compositions and methods and kits for the use thereof
Arjunan et al. Structural, vibrational, electronic investigations and quantum chemical studies of 2-amino-4-methoxybenzothiazole
MX2012003994A (es) Radiosintesis automatizada.
AR088678A1 (es) Procedimiento de sintesis de la ivabradina y de sus sales de adicion a un acido farmaceuticamente aceptable

Legal Events

Date Code Title Description
FG Grant or registration